DK106090A - Fremgangsmaade til fremstilling af 1-aetoxykarbonyloxyaetylesteren af 6-(d-(-)-alfa-amino-alfa-fenylacetamido)-penicillansyre - Google Patents

Fremgangsmaade til fremstilling af 1-aetoxykarbonyloxyaetylesteren af 6-(d-(-)-alfa-amino-alfa-fenylacetamido)-penicillansyre Download PDF

Info

Publication number: DK106090A
Authority: DK; Denmark
Prior art keywords: alfa; carbonyloxya; aetoxy; phenylacetamido; amino
Prior art date: 1982-06-29

Application number

DK106090A

Other languages

English (en)

Other versions

DK167807B1 (da

DK106090D0 (da

Inventor

Luigi Ratti

Derek Reginald Palmer

Robert Graham Tyson

Original Assignee

Astra Laekemedel Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-06-29

Filing date

1990-04-30

Publication date

1990-04-30

1982-06-29 Priority claimed from IT22141/82A external-priority patent/IT1190897B/it

1983-01-07 Priority claimed from GB838300331A external-priority patent/GB8300331D0/en

1990-04-30 Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab

1990-04-30 Publication of DK106090A publication Critical patent/DK106090A/da

1990-04-30 Publication of DK106090D0 publication Critical patent/DK106090D0/da

1993-12-20 Application granted granted Critical

1993-12-20 Publication of DK167807B1 publication Critical patent/DK167807B1/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C68/00—Preparation of esters of carbonic or haloformic acids
- C07C68/02—Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/96—Esters of carbonic or haloformic acids
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Communicable Diseases (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)

DK106090A 1982-06-29 1990-04-30 Fremgangsmaade til fremstilling af 1-ethoxycarbonyloxyethylesteren af 6-(d-(-)-alfa-amino-alfa-phenylacetamido)-penicillansyre DK167807B1 (da)

Applications Claiming Priority (10)

Application Number	Priority Date	Filing Date	Title
IT2214182		1982-06-29
IT22141/82A IT1190897B (it)	1982-06-29	1982-06-29	Procedimento per la preparazione dell'estere 1-etossicarbonilossietilico dell'acido 6-(d(-)-alfa aminoalfa fenilacetamido)-penicillanico
GB8226751		1982-09-20
GB8226751		1982-09-20
GB8228622		1982-10-06
GB8228622		1982-10-06
GB8232629		1982-11-16
GB8232629		1982-11-16
GB8300331		1983-01-07
GB838300331A GB8300331D0 (en)	1983-01-07	1983-01-07	Preparation of bromo carbonates

Publications (3)

Publication Number	Publication Date
DK106090A true DK106090A (da)	1990-04-30
DK106090D0 DK106090D0 (da)	1990-04-30
DK167807B1 DK167807B1 (da)	1993-12-20

Family

ID=27516485

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
DK296683A DK160039C (da)	1982-06-29	1983-06-28	Forbindelsen alfa-bromidaetylkarbonat og anvendelse af alfa-bromidaetylkarbonat ved fremstilling af aetoxykarbonyloxyaetylesteren af penicillin g
DK105990A DK159821C (da)	1982-06-29	1990-04-30	Fremgangsmaade til fremstilling af 1-aetoxykarbonyloxyaetylesteren af 6-(d-(-)-alfa-amino-alfa-fenylacetamido)-penicillansyre
DK106090A DK167807B1 (da)	1982-06-29	1990-04-30	Fremgangsmaade til fremstilling af 1-ethoxycarbonyloxyethylesteren af 6-(d-(-)-alfa-amino-alfa-phenylacetamido)-penicillansyre

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
DK296683A DK160039C (da)	1982-06-29	1983-06-28	Forbindelsen alfa-bromidaetylkarbonat og anvendelse af alfa-bromidaetylkarbonat ved fremstilling af aetoxykarbonyloxyaetylesteren af penicillin g
DK105990A DK159821C (da)	1982-06-29	1990-04-30	Fremgangsmaade til fremstilling af 1-aetoxykarbonyloxyaetylesteren af 6-(d-(-)-alfa-amino-alfa-fenylacetamido)-penicillansyre

Country Status (23)

Country	Link
JP (2)	JPH0819052B2 (da)
AT (1)	AT383128B (da)
AU (1)	AU566803B2 (da)
BG (3)	BG38335A3 (da)
CH (2)	CH657620B (da)
CY (2)	CY1519A (da)
DD (1)	DD211561A5 (da)
DE (2)	DE3348299C2 (da)
DK (3)	DK160039C (da)
FI (1)	FI79115C (da)
FR (1)	FR2543957B1 (da)
GB (3)	GB2168050A (da)
GR (1)	GR78585B (da)
HU (1)	HU191534B (da)
IE (1)	IE56712B1 (da)
IL (1)	IL68992A (da)
IS (1)	IS1361B6 (da)
NL (1)	NL194081C (da)
NO (3)	NO157696C (da)
NZ (1)	NZ204736A (da)
PT (1)	PT76944B (da)
SE (2)	SE454879B (da)
YU (2)	YU43926B (da)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2573756B1 (fr) *	1984-11-23	1987-01-16	Poudres & Explosifs Ste Nale	Procede de preparation des carbonates de bromo-1 ethyle et d'hydrocarbyle et nouveaux carbonates de bromo-1 ethyle et d'hydrocarbyle

Family Cites Families (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CH516593A (de) *	1967-09-29	1971-12-15	Leo Pharm Prod Ltd	Verfahren zur Herstellung von neuen Estern von a-Aminobenzyl-penicillin
US3873521A (en) *	1970-09-17	1975-03-25	Astra Laekemedel Ab	Esters of {60 -amino penicillins
IE35648B1 (en) *	1970-09-25	1976-04-14	Beecham Group Ltd	Penicillins
DE2161420A1 (de) *	1970-12-30	1972-07-27	Toyama Chemical Co. Ltd., Tokio	Penicillinderivate und Verfahren zu deren Herstellung
DE2228670A1 (de) *	1971-06-15	1973-01-11	Yamanouchi Pharma Co Ltd	Neue oxymethylesterderivate von penicillin und cephalosporin
IL48514A (en) *	1972-02-15	1976-08-31	Mckenna A	Hexapeptide intermediate for the preparation of the lh-and fsh-releasing hormone
GB1426717A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1426869A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1425571A (en) *	1972-03-13	1976-02-18	Astra Laekemedel Ab	Penicillins and cephaosporins
SE397981B (sv) *	1973-02-19	1977-11-28	Astra Laekemedel Ab	Nya tetraalkylammoniumsalter av 6-aminopenicillansyra och av bensylpenicillin avsedda att anvendas som mellanprodukter vid framstellning av vissa estrar av 6-aminopenicillansyra och av bensylpenicillin
GB1565656A (en) *	1975-12-13	1980-04-23	Beecham Group Ltd	Preparation of substituted penicillin acid esters
GB1598568A (en) *	1977-04-19	1981-09-23	Glaxo Lab Ltd	Esters of(6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl)-2-methoxyiminoacetamido)-ceph-3-em-4-carboxylic acid
JPS5444694A (en) *	1977-09-06	1979-04-09	Kou Kamata	Aminobenzylpenicillin derivative
AU1637983A (en) *	1982-06-30	1984-01-05	Glaxo Group Limited	Cephalosporin antibiotics
ATE43833T1 (de) *	1982-11-04	1989-06-15	Astra Laekemedel Ab	Verfahren zur herstellung des 1'ethoxycarbonyloxyethylestersvon benzylpenicillin.

1983
- 1983-06-15 IL IL68992A patent/IL68992A/xx not_active IP Right Cessation
- 1983-06-15 SE SE8303414A patent/SE454879B/sv not_active IP Right Cessation
- 1983-06-20 IE IE1445/83A patent/IE56712B1/en not_active IP Right Cessation
- 1983-06-24 DE DE3348299A patent/DE3348299C2/de not_active Expired - Lifetime
- 1983-06-24 DE DE3322783A patent/DE3322783A1/de active Granted
- 1983-06-27 GB GB08528958A patent/GB2168050A/en not_active Withdrawn
- 1983-06-28 BG BG068052A patent/BG38335A3/xx unknown
- 1983-06-28 BG BG061516A patent/BG37527A3/xx unknown
- 1983-06-28 CH CH527585A patent/CH657620B/de not_active IP Right Cessation
- 1983-06-28 AU AU16328/83A patent/AU566803B2/en not_active Expired
- 1983-06-28 FI FI832363A patent/FI79115C/fi not_active IP Right Cessation
- 1983-06-28 DK DK296683A patent/DK160039C/da not_active IP Right Cessation
- 1983-06-28 HU HU832325A patent/HU191534B/hu unknown
- 1983-06-28 NO NO832351A patent/NO157696C/no not_active IP Right Cessation
- 1983-06-28 NZ NZ204736A patent/NZ204736A/en unknown
- 1983-06-28 GR GR71790A patent/GR78585B/el unknown
- 1983-06-28 CH CH3540/83A patent/CH656377A5/de not_active IP Right Cessation
- 1983-06-28 NL NL8302286A patent/NL194081C/nl not_active IP Right Cessation
- 1983-06-28 BG BG068053A patent/BG38336A3/xx unknown
- 1983-06-28 PT PT76944A patent/PT76944B/pt unknown
- 1983-06-29 IS IS2825A patent/IS1361B6/is unknown
- 1983-06-29 YU YU1415/83A patent/YU43926B/xx unknown
- 1983-06-29 DD DD83252531A patent/DD211561A5/de unknown
- 1983-06-29 AT AT0238483A patent/AT383128B/de not_active IP Right Cessation
- 1983-12-30 FR FR8321138A patent/FR2543957B1/fr not_active Expired
1985
- 1985-03-28 NO NO851255A patent/NO851255L/no unknown
- 1985-03-28 NO NO851254A patent/NO851254L/no unknown
- 1985-09-16 GB GB08522826A patent/GB2168699B/en not_active Expired
- 1985-09-16 GB GB08522827A patent/GB2169287B/en not_active Expired
1986
- 1986-02-14 YU YU218/86A patent/YU43693B/xx unknown
1990
- 1990-04-30 DK DK105990A patent/DK159821C/da not_active IP Right Cessation
- 1990-04-30 DK DK106090A patent/DK167807B1/da not_active IP Right Cessation
- 1990-11-16 CY CY1519A patent/CY1519A/en unknown
- 1990-11-16 CY CY1520A patent/CY1520A/en unknown
1991
- 1991-02-26 SE SE9100548A patent/SE503843C2/xx not_active IP Right Cessation
- 1991-04-30 JP JP3124442A patent/JPH0819052B2/ja not_active Expired - Lifetime
- 1991-04-30 JP JP3124441A patent/JPH0730082B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
BG38335A3 (en)	1985-11-15
DK160039C (da)	1991-06-10
CY1519A (en)	1990-11-16
SE8303414D0 (sv)	1983-06-15
DE3322783C2 (da)	1991-01-31
FI832363L (fi)	1983-12-30
GB8522827D0 (en)	1985-10-23
DK167807B1 (da)	1993-12-20
BG37527A3 (en)	1985-06-14
NL8302286A (nl)	1984-01-16
YU141583A (en)	1986-06-30
AU566803B2 (en)	1987-10-29
GB2168050A (en)	1986-06-11
JPH0730082B2 (ja)	1995-04-05
PT76944A (en)	1983-07-01
DE3348299C2 (da)	1990-12-20
DK296683A (da)	1983-12-30
SE9100548D0 (sv)	1991-02-26
JPH0717918A (ja)	1995-01-20
IS2825A7 (is)	1984-07-08
DK159821C (da)	1991-04-29
SE8303414L (sv)	1983-12-30
JPH0543583A (ja)	1993-02-23
SE454879B (sv)	1988-06-06
SE503843C2 (sv)	1996-09-16
FI79115B (fi)	1989-07-31
FI79115C (fi)	1989-11-10
PT76944B (en)	1986-04-09
DK105990D0 (da)	1990-04-30
BG38336A3 (en)	1985-11-15
FR2543957A1 (fr)	1984-10-12
ATA238483A (de)	1986-10-15
CH657620B (da)	1986-09-15
FR2543957B1 (fr)	1986-10-24
AU1632883A (en)	1984-01-05
DK296683D0 (da)	1983-06-28
YU43926B (en)	1989-12-31
NO851255L (no)	1983-12-30
NO157696B (no)	1988-01-25
DE3322783A1 (de)	1984-02-09
NL194081C (nl)	2001-06-05
IL68992A (en)	1991-06-10
DK159821B (da)	1990-12-10
NO851254L (no)	1983-12-30
NO157696C (no)	1988-05-04
YU21886A (en)	1987-10-31
CY1520A (en)	1990-11-16
IS1361B6 (is)	1989-05-25
DK105990A (da)	1990-04-30
FI832363A0 (fi)	1983-06-28
GR78585B (da)	1984-09-27
IE831445L (en)	1983-12-29
GB2169287B (en)	1987-04-08
GB8522826D0 (en)	1985-10-23
GB2168699A (en)	1986-06-25
NL194081B (nl)	2001-02-01
GB8528958D0 (en)	1986-01-02
HU191534B (en)	1987-03-30
GB2169287A (en)	1986-07-09
NZ204736A (en)	1986-11-12
SE9100548L (sv)	1991-02-26
GB2168699B (en)	1987-04-15
JPH0819052B2 (ja)	1996-02-28
DD211561A5 (de)	1984-07-18
CH656377A5 (de)	1986-06-30
NO832351L (no)	1983-12-30
DK160039B (da)	1991-01-21
YU43693B (en)	1989-10-31
AT383128B (de)	1987-05-25
DK106090D0 (da)	1990-04-30
IE56712B1 (en)	1991-11-20

Publication	Publication Date	Title
DK336783D0 (da)	1983-07-22	Fremgangsmade til fremstilling af methylendiphosphonsyrederivater
RO86355A (ro)	1985-03-15	Procedeu pentru prepararea(s)-epimerului esterului acidului 7-beta-malonamida-7-alfa-meto0i-3-tetrazoliltiometil-1-detia-1-o0a-3-cefem-4-carbo0ilic
DK156828C (da)	1990-02-19	Fremgangsmaade til fremstilling af cyclopropancarboxylsyreesterderivater
DK265783A (da)	1983-12-15	Fremgangsmaade til fremstilling af vinylkarboxylsyrederivater
DK159109C (da)	1991-02-18	Fremgangsmaade til fremstilling af l-ascorbinsyre
DK357782A (da)	1983-02-11	Fremgangsmaade til fremstilling af tetrahydrofurancarboxylsyrederivater
DK159122C (da)	1991-02-11	Fremgangsmaade til fremstilling af 2-keto-l-gulonsyre
DK161106C (da)	1991-11-11	Fremgangsmaade til fremstilling af 2-keto-l-gulonsyre
DK98684D0 (da)	1984-02-24	Fremgangsmade til fremstilling af fedtsyreestere af ascorbinsyre
DK157673C (da)	1990-07-16	Analogifremgangsmaade til fremstilling af phenylaliphatiske carboxylsyrederivater
DK554481A (da)	1982-06-16	Fremgangsmaade til fremstilling af cephalosporansyrederivater
DK262982A (da)	1982-12-13	Fremgangsmaade til fremstilling af apovincaminsyreestere
DK157677C (da)	1990-06-18	Fremgangsmaade til fremstilling af cyclopropancarboxylsyreesterderivater
DK354680A (da)	1981-02-19	Fremgangsmaade til fremstilling af substituerede (cyclo) alkancarboxylsyre-(alfa-cyano-3-phenoxy-benzyl)-estere
DK408782A (da)	1983-03-31	Fremgangsmaade til fremstilling af antranilsyreestere
DK159821C (da)	1991-04-29	Fremgangsmaade til fremstilling af 1-aetoxykarbonyloxyaetylesteren af 6-(d-(-)-alfa-amino-alfa-fenylacetamido)-penicillansyre
DK139983A (da)	1984-06-04	Fremgangsmaade til fremstilling af 2-thiopheneddikesyrederivater
DK157613C (da)	1990-06-11	Fremgangsmaade til fremstilling af cyclopropancarboxylsyreesterderivater
DK488088D0 (da)	1988-09-02	Fremgangsmaade til fremstilling af 1-aryl-3-pyrazol-3-carboxylsyreestere
DK179183D0 (da)	1983-04-22	Fremgangsmade til fremstilling af hydroxymethylbutensyrer
DK467381A (da)	1982-04-24	Fremgangsmaade til fremstilling af chlor-fluoralkenyl-substituerede cyclopropancarboxylsyreestere
DK153760C (da)	1989-01-09	Analogifremgangsmaade til fremstilling af estre af 2-thenoylmercaptopropionylglycin
DK20782A (da)	1982-07-20	Fremgangsmaade til fremstilling af cephalosporansyrederivater
DK151020C (da)	1988-02-29	Fremgangsmaade til fremstilling af apovincaminsyreestere
DK196883D0 (da)	1983-05-03	Fremgangsmade til fremstilling af cyanhydrincarboxylsyreestere

Legal Events

Date	Code	Title	Description
1993-12-20	B1	Patent granted (law 1993)
2003-07-14	PUP	Patent expired