DK0708105T3 - 5-HT4-receptoragonister - Google Patents
5-HT4-receptoragonisterInfo
- Publication number
- DK0708105T3 DK0708105T3 DK95307480T DK95307480T DK0708105T3 DK 0708105 T3 DK0708105 T3 DK 0708105T3 DK 95307480 T DK95307480 T DK 95307480T DK 95307480 T DK95307480 T DK 95307480T DK 0708105 T3 DK0708105 T3 DK 0708105T3
- Authority
- DK
- Denmark
- Prior art keywords
- receptor agonists
- agonists
- receptor
- Prior art date
Links
- 108091005482 5-HT4 receptors Proteins 0.000 title 1
- 239000000018 receptor agonist Substances 0.000 title 1
- 229940044601 receptor agonist Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/08—Bridged systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP25490794 | 1994-10-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK0708105T3 true DK0708105T3 (da) | 1999-08-23 |
Family
ID=17271511
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK95307480T DK0708105T3 (da) | 1994-10-20 | 1995-10-20 | 5-HT4-receptoragonister |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US5684003A (da) |
| EP (1) | EP0708105B1 (da) |
| KR (1) | KR960014128A (da) |
| CA (1) | CA2160420A1 (da) |
| DE (1) | DE69506826T2 (da) |
| DK (1) | DK0708105T3 (da) |
| ES (1) | ES2128668T3 (da) |
| TW (1) | TW403747B (da) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR19990022096A (ko) * | 1995-05-31 | 1999-03-25 | 쇼다 오사무 | 모노시클릭 아미노기를 갖는 인다졸 유도체 |
| US6069152A (en) * | 1997-10-07 | 2000-05-30 | Eli Lilly And Company | 5-HT4 agonists and antagonists |
| US5914405A (en) * | 1997-10-07 | 1999-06-22 | Eli Lilly And Company | Process for preparing 3-substituted indazoles |
| FR2792318B1 (fr) * | 1999-04-16 | 2001-06-15 | Synthelabo | Derives d'indazole, leur preparation et leur application en therapeutique |
| US7671097B2 (en) * | 2005-05-24 | 2010-03-02 | Georgia-Pacific Chemicals Llc | Stable phenolic resin polymer dispersions having low free aldehyde content |
| EP1448557A4 (en) | 2001-10-26 | 2005-02-02 | Univ Connecticut | HETEROINDANE: A NEW CLASS OF HIGH-ACTIVITY CANNABIMIMETIC LIGANDS |
| TW200533348A (en) * | 2004-02-18 | 2005-10-16 | Theravance Inc | Indazole-carboxamide compounds as 5-ht4 receptor agonists |
| US7728006B2 (en) * | 2004-04-07 | 2010-06-01 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
| US8309575B2 (en) | 2004-04-07 | 2012-11-13 | Theravance, Inc. | Quinolinone-carboxamide compounds as 5-HT4 receptor agonists |
| TWI351282B (en) | 2004-04-07 | 2011-11-01 | Theravance Inc | Quinolinone-carboxamide compounds as 5-ht4 recepto |
| JP5042028B2 (ja) * | 2004-11-05 | 2012-10-03 | セラヴァンス, インコーポレーテッド | キノリノン−カルボキサミド化合物 |
| ES2332808T3 (es) * | 2004-11-05 | 2010-02-12 | Theravance, Inc. | Compuestos agonistas del receptor 5-ht4. |
| MX2007007818A (es) * | 2004-12-22 | 2007-09-11 | Theravance Inc | Compuestos de indazol-carboxamida. |
| KR20070107807A (ko) * | 2005-03-02 | 2007-11-07 | 세라밴스 인코포레이티드 | 5-ht4 수용체 아고니스트인 퀴놀리논 화합물 |
| JOP20130213B1 (ar) | 2012-07-17 | 2021-08-17 | Takeda Pharmaceuticals Co | معارضات لمستقبلht3-5 |
| PT3201203T (pt) | 2014-09-29 | 2021-08-09 | Takeda Pharmaceuticals Co | Forma cristalina de 1-(1-metil-1h-pirazol-4-il)-n-((1r,5s,7s)-9-metil-3-oxa-9-azabiciclo[3.3.1]nonan-7-il)-1hindol-3-carboxamida |
| GB201511382D0 (en) | 2015-06-29 | 2015-08-12 | Imp Innovations Ltd | Novel compounds and their use in therapy |
| TW202412782A (zh) * | 2022-05-25 | 2024-04-01 | 天主教魯汶大學 | 用於治療trpm3介導之病症的吲唑衍生物 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8829079D0 (en) * | 1988-12-13 | 1989-01-25 | Beecham Group Plc | Novel compounds |
| GB9009389D0 (en) * | 1990-04-26 | 1990-06-20 | Smith Kline French Lab | Treatment |
| US5256656A (en) * | 1990-07-31 | 1993-10-26 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives |
| US5187166A (en) * | 1990-07-31 | 1993-02-16 | Nisshin Flour Milling Co., Ltd. | Azabicyclo derivatives and their use as antiemetics |
| TW251287B (da) * | 1993-04-30 | 1995-07-11 | Nissei Co Ltd |
-
1995
- 1995-10-12 US US08/543,853 patent/US5684003A/en not_active Expired - Lifetime
- 1995-10-12 CA CA002160420A patent/CA2160420A1/en not_active Abandoned
- 1995-10-20 KR KR1019950036424A patent/KR960014128A/ko not_active Withdrawn
- 1995-10-20 DK DK95307480T patent/DK0708105T3/da active
- 1995-10-20 TW TW084111089A patent/TW403747B/zh not_active IP Right Cessation
- 1995-10-20 EP EP95307480A patent/EP0708105B1/en not_active Expired - Lifetime
- 1995-10-20 ES ES95307480T patent/ES2128668T3/es not_active Expired - Lifetime
- 1995-10-20 DE DE69506826T patent/DE69506826T2/de not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| KR960014128A (ko) | 1996-05-22 |
| DE69506826T2 (de) | 1999-08-05 |
| EP0708105B1 (en) | 1998-12-23 |
| ES2128668T3 (es) | 1999-05-16 |
| EP0708105A1 (en) | 1996-04-24 |
| TW403747B (en) | 2000-09-01 |
| US5684003A (en) | 1997-11-04 |
| CA2160420A1 (en) | 1996-04-21 |
| DE69506826D1 (de) | 1999-02-04 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| DK0802910T3 (da) | Estrogenagonister/antagonister | |
| EP0934305A4 (en) | INTEGRINANTAGONISTS | |
| FI964576L (fi) | Uusia agonistiyhdisteitä | |
| NO972016D0 (no) | Indolyl-Y-reseptorantagonister | |
| ID24836A (id) | Agonis prostaglandin | |
| DE69734833D1 (de) | Vitronektin rezeptor antagonisten | |
| DK0708105T3 (da) | 5-HT4-receptoragonister | |
| NO961887L (no) | -adrenergiske agonister | |
| FI951249L (fi) | Serotiinireseptoriaineita | |
| EP0885205A4 (en) | Fibrinogen Receptor Antagonists | |
| DK0906294T3 (da) | Benzoxazinon-dopamin D4-receptor-antagonister | |
| FI974170A0 (fi) | B-adrenergisiä agonisteja | |
| TR199501389A2 (tr) | Adesyon reseptörü antagonistleri (karsitlari). | |
| ID17561A (id) | Komposisi untuk pemakaian luar | |
| NO985970D0 (no) | Indolinderivater anvendelige som 5_HT-2C-reseptor-antagonister | |
| BR9709521A (pt) | "3-Cianoaril-pirazóis" | |
| FI971492L (fi) | Indolijohdannaiset 5-HT1-tyyppisinä agonisteina | |
| MA23795A1 (fr) | Derives d'indole substitues | |
| DE69431672D1 (de) | Adrenergischer rezeptor | |
| NO973624D0 (no) | Vasokonstriktive substituerte 2,3-dihydro-1,4-dioksinopiperidiner | |
| FR2758444B1 (fr) | Boucles d'oreille | |
| FI972558A7 (fi) | Uusi reseptori | |
| GB9715018D0 (en) | 3-Fluoro-4-aminopiperidine derivatives as 5-HT receptor agonists | |
| KR960012039U (ko) | 모니터용 서류고정대 | |
| NO962290L (no) | Uthaler for fiskeliner |