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DK0672031T3 - Catecholdiethere som selektive PDE IV-inhibitorer - Google Patents

Catecholdiethere som selektive PDE IV-inhibitorer

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Publication number
DK0672031T3
DK0672031T3 DK94900390T DK94900390T DK0672031T3 DK 0672031 T3 DK0672031 T3 DK 0672031T3 DK 94900390 T DK94900390 T DK 94900390T DK 94900390 T DK94900390 T DK 94900390T DK 0672031 T3 DK0672031 T3 DK 0672031T3
Authority
DK
Denmark
Prior art keywords
inhibitors
dieters
catechol
compounds
selective pde
Prior art date
Application number
DK94900390T
Other languages
Danish (da)
English (en)
Inventor
Allen J Duplantier
James F Eggler
Anthony Marfat
Hiroko Masamune
Original Assignee
Pfizer
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Publication date
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Application granted granted Critical
Publication of DK0672031T3 publication Critical patent/DK0672031T3/da

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    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
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    • C07C65/21—Compounds having carboxyl groups bound to carbon atoms of six—membered aromatic rings and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups containing ether groups, groups, groups, or groups
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NO952178D0 (no) 1995-06-01
AU673569B2 (en) 1996-11-14
NZ257955A (en) 1996-05-28
EP0672031B1 (en) 2003-03-12
HU9303423D0 (en) 1994-04-28
CZ141795A3 (en) 1995-11-15
IL107758A (en) 1997-11-20
NO952178L (no) 1995-08-01
ES2192192T3 (es) 2003-10-01
EP0672031A1 (en) 1995-09-20
FI935379L (fi) 1994-06-03
PL309257A1 (en) 1995-10-02
RU95113454A (ru) 1997-06-10
HUT65928A (en) 1994-07-28
WO1994012461A1 (en) 1994-06-09
CN1094028A (zh) 1994-10-26
JPH08501318A (ja) 1996-02-13
ZA938978B (en) 1995-06-01
DE69332762D1 (de) 2003-04-17
FI935379A0 (fi) 1993-12-01
CA2400368A1 (en) 1994-06-09
CA2150812A1 (en) 1994-06-09
JP3100984B2 (ja) 2000-10-23
AU5539694A (en) 1994-06-22
BR9307570A (pt) 1999-05-25
DE69332762T2 (de) 2003-08-14
PT672031E (pt) 2003-06-30
FI935379A7 (fi) 1994-06-03
KR950704228A (ko) 1995-11-17
CA2150812C (en) 2002-12-24
ATE234270T1 (de) 2003-03-15

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