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DE69531934D1 - Hydrophobe arzneistoffabgabesysteme - Google Patents

Hydrophobe arzneistoffabgabesysteme

Info

Publication number
DE69531934D1
DE69531934D1 DE69531934T DE69531934T DE69531934D1 DE 69531934 D1 DE69531934 D1 DE 69531934D1 DE 69531934 T DE69531934 T DE 69531934T DE 69531934 T DE69531934 T DE 69531934T DE 69531934 D1 DE69531934 D1 DE 69531934D1
Authority
DE
Germany
Prior art keywords
drug delivery
delivery systems
hydrophobic drug
dosage form
unit dosage
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE69531934T
Other languages
English (en)
Other versions
DE69531934T2 (de
Inventor
Edward M Rudnic
John A Mccarty
George W Belenduik
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Supernus Pharmaceuticals Inc
Original Assignee
Shire Laboratories Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Shire Laboratories Inc filed Critical Shire Laboratories Inc
Application granted granted Critical
Publication of DE69531934D1 publication Critical patent/DE69531934D1/de
Publication of DE69531934T2 publication Critical patent/DE69531934T2/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/23—Calcitonins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
    • A61K38/13—Cyclosporins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/31—Somatostatins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1617—Organic compounds, e.g. phospholipids, fats
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/5005—Wall or coating material
    • A61K9/5021—Organic macromolecular compounds
    • A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
    • A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Immunology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Endocrinology (AREA)
  • Zoology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Infusion, Injection, And Reservoir Apparatuses (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DE69531934T 1994-03-18 1995-03-15 Hydrophobe arzneistoffabgabesysteme Expired - Lifetime DE69531934T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/210,014 US5430021A (en) 1994-03-18 1994-03-18 Hydrophobic drug delivery systems
US210014 1994-03-18
PCT/US1995/003212 WO1995025505A1 (en) 1994-03-18 1995-03-15 Hydrophobic drug delivery systems

Publications (2)

Publication Number Publication Date
DE69531934D1 true DE69531934D1 (de) 2003-11-20
DE69531934T2 DE69531934T2 (de) 2004-09-02

Family

ID=22781263

Family Applications (1)

Application Number Title Priority Date Filing Date
DE69531934T Expired - Lifetime DE69531934T2 (de) 1994-03-18 1995-03-15 Hydrophobe arzneistoffabgabesysteme

Country Status (10)

Country Link
US (1) US5430021A (de)
EP (1) EP0750494B1 (de)
JP (1) JPH09510708A (de)
AT (1) ATE251895T1 (de)
AU (1) AU703950B2 (de)
CA (1) CA2185802C (de)
DE (1) DE69531934T2 (de)
DK (1) DK0750494T3 (de)
ES (1) ES2210286T3 (de)
WO (1) WO1995025505A1 (de)

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Also Published As

Publication number Publication date
ATE251895T1 (de) 2003-11-15
CA2185802A1 (en) 1995-09-28
AU1992595A (en) 1995-10-09
JPH09510708A (ja) 1997-10-28
WO1995025505A1 (en) 1995-09-28
ES2210286T3 (es) 2004-07-01
DE69531934T2 (de) 2004-09-02
DK0750494T3 (da) 2004-01-19
EP0750494A4 (de) 1998-05-20
EP0750494A1 (de) 1997-01-02
CA2185802C (en) 2009-12-22
AU703950B2 (en) 1999-04-01
US5430021A (en) 1995-07-04
EP0750494B1 (de) 2003-10-15

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