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DE60335869D1 - 1h-benzo(f)indazol-5-yl-derivate als selektive glucocorticoid-rezeptor-modulatoren - Google Patents

1h-benzo(f)indazol-5-yl-derivate als selektive glucocorticoid-rezeptor-modulatoren

Info

Publication number
DE60335869D1
DE60335869D1 DE60335869T DE60335869T DE60335869D1 DE 60335869 D1 DE60335869 D1 DE 60335869D1 DE 60335869 T DE60335869 T DE 60335869T DE 60335869 T DE60335869 T DE 60335869T DE 60335869 D1 DE60335869 D1 DE 60335869D1
Authority
DE
Germany
Prior art keywords
glucocorticoid receptor
indazol
benzo
derivatives
receptor modulators
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60335869T
Other languages
English (en)
Inventor
Amjad Ali
James M Balkovec
Donald W Graham
Christopher F Thompson
Nazia Quraishi
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Organon Pharma UK Ltd
Merck Sharp and Dohme LLC
Original Assignee
Merck Sharp and Dohme Ltd
Merck Sharp and Dohme LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Sharp and Dohme Ltd, Merck Sharp and Dohme LLC filed Critical Merck Sharp and Dohme Ltd
Application granted granted Critical
Publication of DE60335869D1 publication Critical patent/DE60335869D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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  • Transplantation (AREA)
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  • Child & Adolescent Psychology (AREA)
DE60335869T 2002-04-11 2003-04-08 1h-benzo(f)indazol-5-yl-derivate als selektive glucocorticoid-rezeptor-modulatoren Expired - Lifetime DE60335869D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US37194802P 2002-04-11 2002-04-11
PCT/US2003/010867 WO2003086294A2 (en) 2002-04-11 2003-04-08 1h-benzo[f]indazol-5-yl derivatives as selective glucocorticoid receptor modulators

Publications (1)

Publication Number Publication Date
DE60335869D1 true DE60335869D1 (de) 2011-03-10

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DE60335869T Expired - Lifetime DE60335869D1 (de) 2002-04-11 2003-04-08 1h-benzo(f)indazol-5-yl-derivate als selektive glucocorticoid-rezeptor-modulatoren

Country Status (8)

Country Link
US (2) US7282591B2 (de)
EP (1) EP1496892B1 (de)
JP (1) JP4570878B2 (de)
AT (1) ATE496620T1 (de)
AU (1) AU2003221706B2 (de)
CA (1) CA2481320A1 (de)
DE (1) DE60335869D1 (de)
WO (1) WO2003086294A2 (de)

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