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DE60306534D1 - Neue derivate von cycloalkanodionen, verfahren zu deren herstellung und deren pharmakologische anwendungen - Google Patents

Neue derivate von cycloalkanodionen, verfahren zu deren herstellung und deren pharmakologische anwendungen

Info

Publication number
DE60306534D1
DE60306534D1 DE60306534T DE60306534T DE60306534D1 DE 60306534 D1 DE60306534 D1 DE 60306534D1 DE 60306534 T DE60306534 T DE 60306534T DE 60306534 T DE60306534 T DE 60306534T DE 60306534 D1 DE60306534 D1 DE 60306534D1
Authority
DE
Germany
Prior art keywords
cycloalkanodiones
preparation
new derivatives
treatment
pharmacological applications
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60306534T
Other languages
English (en)
Other versions
DE60306534T2 (de
Inventor
Rio Zambrana Joaquin Del
Manso Diana Frechilla
Rodriguez M Lopez
Salama Bellinda Benhamu
Cubero Angel Fuentes
Wallace Mercedes Delgado
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
UCB Pharma SA Spain
Original Assignee
Cepa Schwarz Pharma SL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cepa Schwarz Pharma SL filed Critical Cepa Schwarz Pharma SL
Application granted granted Critical
Publication of DE60306534D1 publication Critical patent/DE60306534D1/de
Publication of DE60306534T2 publication Critical patent/DE60306534T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/381Heterocyclic compounds having sulfur as a ring hetero atom having five-membered rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/41641,3-Diazoles
    • A61K31/41881,3-Diazoles condensed with other heterocyclic ring systems, e.g. biotin, sorbinil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/04Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D277/00Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/34Oxygen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Epidemiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
DE60306534T 2002-07-31 2003-07-29 Neue derivate von cycloalkanodionen, verfahren zu deren herstellung und deren pharmakologische anwendungen Expired - Fee Related DE60306534T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
ES200201811A ES2199086B1 (es) 2002-07-31 2002-07-31 Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
ES200201811 2002-07-31
PCT/ES2003/000394 WO2004014915A1 (es) 2002-07-31 2003-07-29 Nuevos derivados de cicloalcanodionas procedimiento para su preparación y sus aplicaciones farmacológicas

Publications (2)

Publication Number Publication Date
DE60306534D1 true DE60306534D1 (de) 2006-08-10
DE60306534T2 DE60306534T2 (de) 2007-04-19

Family

ID=31198114

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60306534T Expired - Fee Related DE60306534T2 (de) 2002-07-31 2003-07-29 Neue derivate von cycloalkanodionen, verfahren zu deren herstellung und deren pharmakologische anwendungen

Country Status (23)

Country Link
US (1) US7351732B2 (de)
EP (1) EP1544201B1 (de)
JP (1) JP2005539017A (de)
KR (1) KR20050042471A (de)
CN (2) CN101172977A (de)
AT (1) ATE331717T1 (de)
AU (1) AU2003254512A1 (de)
BR (1) BR0313375A (de)
CA (1) CA2492837A1 (de)
CY (1) CY1106170T1 (de)
DE (1) DE60306534T2 (de)
DK (1) DK1544201T3 (de)
ES (2) ES2199086B1 (de)
IL (1) IL166469A0 (de)
MX (1) MXPA05001245A (de)
NO (1) NO20051068L (de)
NZ (1) NZ538489A (de)
PL (1) PL373644A1 (de)
PT (1) PT1544201E (de)
RU (1) RU2322445C2 (de)
UA (1) UA79801C2 (de)
WO (1) WO2004014915A1 (de)
ZA (1) ZA200500784B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2199086B1 (es) 2002-07-31 2005-06-01 Cepa Schwarz Pharma Sl Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
ES2238015B1 (es) * 2004-01-30 2006-11-01 Cepa Schwarz Pharma, S.L. Derivados de cicloalcanodionas con actividad neuroprotectora.
WO2008015538A2 (en) * 2006-07-31 2008-02-07 Schwarz Pharma S.L. Use of diaza- and thiaza-cycloalkanediones for preventing and/or treating pain and /or migraine
EP2338873A1 (de) 2009-12-22 2011-06-29 Gmeiner, Peter Neue Aminotetralinderivate

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4055410A (en) * 1976-03-15 1977-10-25 E. I. Du Pont De Nemours And Company Substituted bromo- or chloroacetamide herbicides
EP0002978B1 (de) * 1977-12-29 1982-10-06 Synthelabo Thiazolidindion-2,4 Derivate, deren Herstellung und Verwendung als Arzneimittel
DE3901814A1 (de) * 1988-07-28 1990-02-01 Bayer Ag Substituierte aminomethylzetraline sowie ihre heterocyclischen analoga
EP0510691B1 (de) * 1991-04-26 2004-11-03 Osaka Bioscience Institute Für ein menschliches Zelloberflächen-Antigen kodierende DNS
TW288010B (de) * 1992-03-05 1996-10-11 Pfizer
AP486A (en) * 1993-04-27 1996-04-16 Pfizer Indole derivatives.
WO1996006846A1 (es) 1994-09-01 1996-03-07 Universidad Complutense De Madrid Nuevos derivados de arilpiperazinas
ES2082727B1 (es) 1994-09-01 1996-10-16 Univ Madrid Complutense Nuevos derivados de arilpiperazinas.
ES2094690B1 (es) 1994-11-22 1997-08-01 Univ Madrid Complutense Nuevos derivados de imida-piperazinas.
ES2109190B1 (es) 1996-03-22 1998-07-01 Univ Madrid Complutense Nuevos derivados de bencimidazol con afinidad por los receptores serotoninergicos 5-ht /5-ht
ES2129370B1 (es) 1997-09-23 2000-03-01 Univ Madrid Complutense Procedimiento para la obtencion del 2-(4-(4-(m-etilsulfonamidofenil)p iperazin-1-il(butil)-1,3-dioxoperhidropirrolo)1,2-c(imidazol
US6133277A (en) 1997-12-05 2000-10-17 Janssen Pharmaceutica N.V. (Benzodioxan, benzofuran or benzopyran) derivatives having fundic relaxation properties
ES2154605B1 (es) 1999-09-14 2001-11-16 Univ Madrid Complutense Nuevos derivados mixtos de bencimidazol-arilpiperazina con afinidad por los receptores serotoninergicos 5-ht1a y 5-ht3
DE10148425A1 (de) 2001-10-01 2003-04-17 Bayer Ag Chromane
ES2199086B1 (es) 2002-07-31 2005-06-01 Cepa Schwarz Pharma Sl Nuevos derivados de cicloalcanodionas, procedimiento para su preparacion y sus aplicaciones farmacologicas.
ES2238015B1 (es) 2004-01-30 2006-11-01 Cepa Schwarz Pharma, S.L. Derivados de cicloalcanodionas con actividad neuroprotectora.
EP1674103A1 (de) 2004-12-27 2006-06-28 Cepa Schwarz Pharma s.l. Arylpiperazine Derivative als 5-HT1A Rezeptor Liganden

Also Published As

Publication number Publication date
RU2322445C2 (ru) 2008-04-20
ES2199086A1 (es) 2004-02-01
NZ538489A (en) 2006-09-29
ES2271673T3 (es) 2007-04-16
CN1671708A (zh) 2005-09-21
EP1544201B1 (de) 2006-06-28
KR20050042471A (ko) 2005-05-09
DE60306534T2 (de) 2007-04-19
US20050250777A1 (en) 2005-11-10
CN101172977A (zh) 2008-05-07
PL373644A1 (en) 2005-09-05
ZA200500784B (en) 2006-08-30
NO20051068L (no) 2005-02-25
AU2003254512A1 (en) 2004-02-25
BR0313375A (pt) 2005-06-21
ES2199086B1 (es) 2005-06-01
JP2005539017A (ja) 2005-12-22
MXPA05001245A (es) 2005-09-12
IL166469A0 (en) 2006-01-15
UA79801C2 (en) 2007-07-25
CY1106170T1 (el) 2011-06-08
RU2005102821A (ru) 2005-10-10
US7351732B2 (en) 2008-04-01
ATE331717T1 (de) 2006-07-15
EP1544201A1 (de) 2005-06-22
WO2004014915A1 (es) 2004-02-19
CN100422185C (zh) 2008-10-01
PT1544201E (pt) 2006-11-30
DK1544201T3 (da) 2006-10-30
CA2492837A1 (en) 2004-02-19

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Legal Events

Date Code Title Description
8327 Change in the person/name/address of the patent owner

Owner name: SCHWARZ PHARMA, S.L., MADRID, ES

8364 No opposition during term of opposition
8328 Change in the person/name/address of the agent

Representative=s name: HOEFER & PARTNER, 81543 MUENCHEN

8339 Ceased/non-payment of the annual fee