[go: up one dir, main page]

DE60305460D1 - Verwendung von 4-(4-methylpiperazin-1-ylmethyl)-n 4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl benzamid zur behandlung von seminomen - Google Patents

Verwendung von 4-(4-methylpiperazin-1-ylmethyl)-n 4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl benzamid zur behandlung von seminomen

Info

Publication number
DE60305460D1
DE60305460D1 DE60305460T DE60305460T DE60305460D1 DE 60305460 D1 DE60305460 D1 DE 60305460D1 DE 60305460 T DE60305460 T DE 60305460T DE 60305460 T DE60305460 T DE 60305460T DE 60305460 D1 DE60305460 D1 DE 60305460D1
Authority
DE
Germany
Prior art keywords
ylamino
pyrimidin
ylmethyl
pyridin
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60305460T
Other languages
English (en)
Inventor
C Heinrich
Christopher Corless
Kathleen Kemmer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Oregon Health and Science University
Government of the United States of America
Original Assignee
Oregon Health and Science University
Government of the United States of America
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Oregon Health and Science University, Government of the United States of America filed Critical Oregon Health and Science University
Application granted granted Critical
Publication of DE60305460D1 publication Critical patent/DE60305460D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE60305460T 2002-02-22 2003-02-17 Verwendung von 4-(4-methylpiperazin-1-ylmethyl)-n 4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl benzamid zur behandlung von seminomen Expired - Lifetime DE60305460D1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US35904902P 2002-02-22 2002-02-22
PCT/IB2003/000622 WO2003070248A1 (en) 2002-02-22 2003-02-17 Use of 4-(4-methylpiperazin-1-ylmethyl)-n[4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl]-benzamide for treating seminomas

Publications (1)

Publication Number Publication Date
DE60305460D1 true DE60305460D1 (de) 2006-06-29

Family

ID=27757766

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60305460T Expired - Lifetime DE60305460D1 (de) 2002-02-22 2003-02-17 Verwendung von 4-(4-methylpiperazin-1-ylmethyl)-n 4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl benzamid zur behandlung von seminomen

Country Status (7)

Country Link
US (1) US20050153975A1 (de)
EP (1) EP1487452B1 (de)
JP (1) JP2005523282A (de)
AT (1) ATE326970T1 (de)
AU (1) AU2003209521A1 (de)
DE (1) DE60305460D1 (de)
WO (1) WO2003070248A1 (de)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW225528B (de) * 1992-04-03 1994-06-21 Ciba Geigy Ag
CO4940418A1 (es) * 1997-07-18 2000-07-24 Novartis Ag Modificacion de cristal de un derivado de n-fenil-2- pirimidinamina, procesos para su fabricacion y su uso
DE60017179T2 (de) * 1999-10-19 2006-01-05 Merck & Co., Inc. Tyrosin kinaseinhibitoren
MY128450A (en) * 2000-05-24 2007-02-28 Upjohn Co 1-(pyrrolidin-1-ylmethyl)-3-(pyrrol-2-ylmethylidene)-2-indolinone derivatives
WO2002028409A2 (en) * 2000-10-05 2002-04-11 Whitehead Institute For Biomedical Research Effects of combined administration of farnesyl transferase inhibitors and signal transduction inhibitors

Also Published As

Publication number Publication date
US20050153975A1 (en) 2005-07-14
EP1487452B1 (de) 2006-05-24
EP1487452A1 (de) 2004-12-22
WO2003070248A1 (en) 2003-08-28
JP2005523282A (ja) 2005-08-04
ATE326970T1 (de) 2006-06-15
AU2003209521A1 (en) 2003-09-09

Similar Documents

Publication Publication Date Title
ATE321556T1 (de) Behandlung gastrointestinaler stroma-tumoren
MY128664A (en) Crystal modification of a n-phenyl-2-pyrimidineamine derivative, processes for its manufacture and its use
TWI347186B (en) Salt forms of 4-(4-methylpiperazin-1-ylmethyl)-n-[4-methyl-3-(4-pyridin-3-yl)pyrimidin-2-ylamino)phenyl]-benzamide
ATE399555T1 (de) Behandlung der rheumatoiden arthritis mit imitanib
BR0316126A (pt) Combinação de compostos para o tratamento de leucemia linfocìtica crÈnica
DE60305460D1 (de) Verwendung von 4-(4-methylpiperazin-1-ylmethyl)-n 4-methyl-3-(4-pyridin-3-yl) pyrimidin-2-ylamino) phenyl benzamid zur behandlung von seminomen
DE602004022540D1 (de) Verwendung von tyrosin-kinase-hemmern zur behandlung von diabetes
BR0312242A (pt) 4-(4-metilpiperazin-1-ilmetil)-n-[4-metil-3-(4-piridin-3-il) pirimidin-2-ilamino)fenil]-benzamida para o tratamento da fibrose pulmonar
WO2004026930A3 (en) The method for reducing inflammation using sti-571 or its salt
UY28498A1 (es) Modificación de cristal de un derivado de n-fenil-2-pirimidinamina, procesos para su fabricación y su uso.
ECSP982588A (es) Modificacion de cristal de un derivado de n-fenil -2-pirimidinamina procesos para su fabricacion y su uso

Legal Events

Date Code Title Description
8332 No legal effect for de