DE602004009030D1 - Phenyltetrazol-Verbindungen - Google Patents
Phenyltetrazol-VerbindungenInfo
- Publication number
- DE602004009030D1 DE602004009030D1 DE602004009030T DE602004009030T DE602004009030D1 DE 602004009030 D1 DE602004009030 D1 DE 602004009030D1 DE 602004009030 T DE602004009030 T DE 602004009030T DE 602004009030 T DE602004009030 T DE 602004009030T DE 602004009030 D1 DE602004009030 D1 DE 602004009030D1
- Authority
- DE
- Germany
- Prior art keywords
- phenyltetrazole
- connections
- angiotensin
- antagonists
- intermediates
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired - Lifetime
Links
- MARUHZGHZWCEQU-UHFFFAOYSA-N 5-phenyl-2h-tetrazole Chemical compound C1=CC=CC=C1C1=NNN=N1 MARUHZGHZWCEQU-UHFFFAOYSA-N 0.000 title abstract 2
- 229940123413 Angiotensin II antagonist Drugs 0.000 abstract 1
- 239000002333 angiotensin II receptor antagonist Substances 0.000 abstract 1
- 238000006243 chemical reaction Methods 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D257/04—Five-membered rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT002338A ITMI20032338A1 (it) | 2003-11-28 | 2003-11-28 | Composti feniltetrazolici. |
| ITMI20032338 | 2003-11-28 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DE602004009030D1 true DE602004009030D1 (de) | 2007-10-31 |
| DE602004009030T2 DE602004009030T2 (de) | 2008-06-12 |
Family
ID=34611237
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE602004009030T Expired - Lifetime DE602004009030T2 (de) | 2003-11-28 | 2004-11-19 | Phenyltetrazolverbindungen |
Country Status (9)
| Country | Link |
|---|---|
| US (2) | US7345072B2 (de) |
| EP (1) | EP1555260B1 (de) |
| JP (1) | JP2005162751A (de) |
| AT (1) | ATE373645T1 (de) |
| DE (1) | DE602004009030T2 (de) |
| ES (1) | ES2273617T3 (de) |
| IT (1) | ITMI20032338A1 (de) |
| PL (1) | PL1555260T3 (de) |
| PT (1) | PT1555260E (de) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1706401A1 (de) | 2004-09-02 | 2006-10-04 | Teva Pharmaceutical Industries Ltd. | Herstellung von olmesartan-medoxomil |
| DE102004060699A1 (de) * | 2004-12-16 | 2006-06-22 | Ratiopharm Gmbh | Verfahren zur Herstellung von Candesartan |
| WO2006067216A2 (en) * | 2004-12-22 | 2006-06-29 | Enantia, S. L. | Intermediate compounds for the preparation of an angiotensin ii receptor and process for the preparation of valsartan |
| JP2007526342A (ja) | 2005-01-03 | 2007-09-13 | テバ ファーマシューティカル インダストリーズ リミティド | 低レベルの不純物を有するオルメサルタンメドキソミル |
| WO2007005967A2 (en) * | 2005-07-05 | 2007-01-11 | Teva Pharmaceutical Industries Ltd. | Process for preparing valsartan |
| EP1816131A1 (de) * | 2006-02-06 | 2007-08-08 | KRKA, tovarna zdravil, d.d., Novo mesto | Verfahren zur Herstellung von Olmesartan Medoxomil |
| CA2616466A1 (en) * | 2005-07-29 | 2007-02-15 | Krka | Process for the preparation of olmesartan medoxomil |
| WO2007071750A1 (en) * | 2005-12-22 | 2007-06-28 | Enantia, S.L. | Intermediates and processes for the preparation of valsartan |
| ES2300175B1 (es) * | 2006-02-14 | 2009-06-08 | Inke, S.A. | Procedimiento para la obtencion de intermedios utiles en la obtencion de un compuesto farmaceuticamente activo. |
| ITMI20061848A1 (it) * | 2006-09-27 | 2008-03-28 | Dipharma Spa | Procedimento per la preparazione di composti feniltetrazolici |
| BRPI0815111A2 (pt) * | 2007-08-08 | 2015-01-27 | Lek Pharmaceuticals | Processo para a preparação ou purificação de olmesartan medoxomil, sais de olmesartan medoxomil e seus usos e composições farmacêuticas |
| EP2432777A1 (de) | 2009-05-20 | 2012-03-28 | Ranbaxy Laboratories Limited | Verfahren zur herstellung von olmesartan-medoxomil |
| KR101117128B1 (ko) * | 2009-06-02 | 2012-03-14 | 한국화학연구원 | 페닐테트라졸 유도체 또는 이의 약학적으로 허용가능한 염을 유효성분으로 포함하는 골다공증 또는 비만의 예방 또는 치료용 약학적 조성물 |
| WO2011080684A1 (en) | 2009-12-31 | 2011-07-07 | Ranbaxy Laboratories Limited | Process for the preparation of candesartan cilexetil |
| WO2011092666A1 (en) | 2010-01-29 | 2011-08-04 | Ranbaxy Laboratories Limited | An improved process for the preparation of candesartan cilexetil, polymorphic forms of n-trityl candesartan and their uses thereof |
| CN102675294A (zh) * | 2012-05-17 | 2012-09-19 | 浙江天宇药业股份有限公司 | 一种合成氯沙坦及其中间体的方法 |
| CN105001209A (zh) * | 2015-06-29 | 2015-10-28 | 千辉药业(安徽)有限责任公司 | 一种厄贝沙坦的合成方法 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5412102A (en) * | 1994-05-27 | 1995-05-02 | Syntex (U.S.A.) Inc. | Processes for preparing 1-butyl-2-[2'-(2H-tetrazol-5-yl) biphenyl-4-ylmethyl]-1H-indole-3-carboxylic acid |
| TW409125B (en) * | 1996-04-22 | 2000-10-21 | Novartis Ag | Antivirally active heterocyclic azahexane derivatives |
| ATE314097T1 (de) * | 1996-10-28 | 2006-01-15 | Amersham Health As | Kontrastmittel |
| JP2002145770A (ja) * | 2000-08-30 | 2002-05-22 | Sankyo Co Ltd | 心不全の予防又は治療のための医薬組成物 |
-
2003
- 2003-11-28 IT IT002338A patent/ITMI20032338A1/it unknown
-
2004
- 2004-11-19 ES ES04027599T patent/ES2273617T3/es not_active Expired - Lifetime
- 2004-11-19 EP EP04027599A patent/EP1555260B1/de not_active Expired - Lifetime
- 2004-11-19 DE DE602004009030T patent/DE602004009030T2/de not_active Expired - Lifetime
- 2004-11-19 AT AT04027599T patent/ATE373645T1/de active
- 2004-11-19 PL PL04027599T patent/PL1555260T3/pl unknown
- 2004-11-19 PT PT04027599T patent/PT1555260E/pt unknown
- 2004-11-24 US US10/995,135 patent/US7345072B2/en not_active Expired - Fee Related
- 2004-11-25 JP JP2004340068A patent/JP2005162751A/ja active Pending
-
2008
- 2008-01-29 US US12/021,313 patent/US20080119657A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP1555260B1 (de) | 2007-09-19 |
| ES2273617T3 (es) | 2008-03-16 |
| ITMI20032338A1 (it) | 2005-05-29 |
| ES2273617T1 (es) | 2007-05-16 |
| PL1555260T3 (pl) | 2008-02-29 |
| EP1555260A1 (de) | 2005-07-20 |
| US20080119657A1 (en) | 2008-05-22 |
| ATE373645T1 (de) | 2007-10-15 |
| US20050119488A1 (en) | 2005-06-02 |
| PT1555260E (pt) | 2007-12-04 |
| DE602004009030T2 (de) | 2008-06-12 |
| US7345072B2 (en) | 2008-03-18 |
| JP2005162751A (ja) | 2005-06-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8364 | No opposition during term of opposition |