DE60101386D1 - PIPERAZINE AND PIPERIDINE COMPOUNDS - Google Patents

PIPERAZINE AND PIPERIDINE COMPOUNDS

Info

Publication number: DE60101386D1
Authority: DE; Germany
Prior art keywords: piperazine; piperidine compounds; piperidine; compounds
Prior art date: 2000-05-12
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired - Lifetime

Application number

DE60101386T

Other languages

German (de)

Other versions

DE60101386T2 (en

Inventor

W Feenstra

Der Heijden A Van

G Kruse

K Long

Scharrenburg J Van

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Abbott Healthcare Products BV

Original Assignee

Solvay Pharmaceuticals BV

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-12

Filing date

2001-05-10

Publication date

2004-01-15

2001-05-10 Application filed by Solvay Pharmaceuticals BV filed Critical Solvay Pharmaceuticals BV

2004-01-15 Publication of DE60101386D1 publication Critical patent/DE60101386D1/en

2004-05-27 Application granted granted Critical

2004-05-27 Publication of DE60101386T2 publication Critical patent/DE60101386T2/en

2021-05-11 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Chemical Kinetics & Catalysis (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Neurosurgery (AREA)
Medicinal Chemistry (AREA)
Biomedical Technology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Addiction (AREA)
Psychology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DE60101386T 2000-05-12 2001-05-10 PIPERAZINE AND PIPERIDINE COMPOUNDS Expired - Lifetime DE60101386T2 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP00201699		2000-05-12
EP00201699		2000-05-12
PCT/EP2001/005320 WO2001085725A1 (en)	2000-05-12	2001-05-10	Piperazine and piperidine compounds

Publications (2)

Publication Number	Publication Date
DE60101386D1 true DE60101386D1 (en)	2004-01-15
DE60101386T2 DE60101386T2 (en)	2004-05-27

Family

ID=8171488

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DE60101386T Expired - Lifetime DE60101386T2 (en)	2000-05-12	2001-05-10	PIPERAZINE AND PIPERIDINE COMPOUNDS

Country Status (27)

Country	Link
US (2)	US6911448B2 (en)
EP (1)	EP1283838B1 (en)
JP (1)	JP2003532729A (en)
CN (1)	CN1174979C (en)
AR (1)	AR028443A1 (en)
AT (1)	ATE255578T1 (en)
AU (2)	AU6392701A (en)
BR (1)	BR0110592A (en)
CA (1)	CA2405971C (en)
CZ (1)	CZ301464B6 (en)
DE (1)	DE60101386T2 (en)
DK (1)	DK1283838T3 (en)
DZ (1)	DZ3370A1 (en)
ES (1)	ES2211809T3 (en)
HU (1)	HUP0302016A2 (en)
IL (2)	IL152177A0 (en)
MX (1)	MXPA02011084A (en)
NO (1)	NO323778B1 (en)
NZ (1)	NZ522116A (en)
PL (1)	PL198857B1 (en)
PT (1)	PT1283838E (en)
RU (1)	RU2261250C2 (en)
SK (1)	SK286778B6 (en)
TR (1)	TR200302294T4 (en)
UA (1)	UA72337C2 (en)
WO (1)	WO2001085725A1 (en)
ZA (1)	ZA200208537B (en)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
CA2405971C (en) *	2000-05-12	2010-03-30	Solvay Pharmaceuticals B.V.	New piperazine and piperidine compounds
EP1408976B3 (en) *	2001-07-20	2010-08-25	Psychogenics Inc.	Treatment for attention-deficit hyperactivity disorder
WO2004000837A1 (en) *	2002-06-25	2003-12-31	Sumitomo Pharmaceuticals Co., Ltd.	Novel benzoxazolinone derivative
ES2232292B1 (en) *	2003-07-30	2006-11-01	Laboratorios Del Dr. Esteve, S.A.	SULFONAMIDIC COMPOUNDS DERIVED FROM BENZOXAZINONA, ITS PREPARATION AND USE AS MEDICATIONS.
US7596407B2 (en)	2004-03-26	2009-09-29	Solvay Pharmaceuticals, B.V.	Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
EP1595542A1 (en) *	2004-03-26	2005-11-16	Solvay Pharmaceuticals B.V.	Transdermal iontophoretic delivery of piperazinyl-2(3H)-benzoxazolone compounds
AR058022A1 (en) *	2005-08-22	2008-01-23	Solvay Pharm Bv	DERIVATIVES OF BENZOOXAZOLES, PHARMACEUTICAL COMPOSITIONS AND ITS USE FOR THE TREATMENT OF NERVOUS SYSTEM DISORDERS.
US7750013B2 (en)	2005-08-22	2010-07-06	Solvay Pharmaceuticals, B.V.	N-oxides as prodrugs of piperazine and piperidine derivatives
SI1919883T1 (en) *	2005-08-22	2009-04-30	Solvay Pharm Bv	N-oxides as prodrugs of piperazine&piperidine derivatives
US20070275977A1 (en) *	2006-05-02	2007-11-29	Van Aar Marcel P	N-oxides of pyridylmethyl -piperazine and -piperidine derivatives
US8106056B2 (en)	2006-06-16	2012-01-31	Solvay Pharmaceuticals B.V.	Combination preparations comprising bifeprunox and a dopamine agonist
ES2344131T3 (en)	2006-12-07	2010-08-18	F. Hoffmann-La Roche Ag	DERIVATIVES OF ESPIRO-PIPERIDINE AS ANTAGONISTS OF RECEIVER V1A.
MX2009005507A (en)	2006-12-07	2009-06-03	Hoffmann La Roche	Spiro-piperidine derivatives.
US20080139617A1 (en)	2006-12-08	2008-06-12	Caterina Bissantz	Indoles
CA2670139A1 (en)	2006-12-08	2008-06-12	F. Hoffmann-La Roche Ag	Indoles
MX2009006454A (en)	2006-12-22	2009-06-26	Hoffmann La Roche	Spiro-piperidine derivatives.
WO2009090177A1 (en) *	2008-01-15	2009-07-23	Solvay Pharmaceuticals B.V.	Bifeprunox derivatives
EP3503879A4 (en)	2016-08-26	2020-04-29	EXCIVA GmbH	COMPOSITIONS AND RELATED METHODS
EP3831898A4 (en) *	2018-07-27	2022-04-06	Chugoku Marine Paints, Ltd.	ANTI-ROITING PAINT COMPOSITION, ANTI-ROITING COATING, SUBSTRATE WITH ANTI-ROITING COATING, MANUFACTURING METHOD THEREOF AND REPAIRING METHOD

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60126275A (en) *	1983-12-13	1985-07-05	Otsuka Pharmaceut Co Ltd	Benzothiazole derivative
FR2567884B1 (en)	1984-07-19	1987-03-06	Roussel Uclaf	NEW INDOLE DERIVATIVES, THEIR PREPARATION, THEIR APPLICATION AS MEDICAMENTS AND THE COMPOSITIONS CONTAINING THEM
DE3571436D1 (en)	1984-12-21	1989-08-17	Duphar Int Res	New pharmaceutical compositions having anti-psychotic properties
EP0189612B1 (en) *	1984-12-21	1992-11-04	Duphar International Research B.V	New pharmaceutical compositions having a psychotropic activity
DE4127849A1 (en) *	1991-08-22	1993-02-25	Merck Patent Gmbh	BENZODIOXAN DERIVATIVES
BRPI9708389B8 (en) *	1996-03-29	2015-12-08	Duphar Int Res	piperazine and piperidine compounds, pharmaceutical compositions.
TW530054B (en) *	1997-09-24	2003-05-01	Duphar Int Res	New piperazine and piperidine compounds
GB9811879D0 (en) *	1998-06-03	1998-07-29	Knoll Ag	Therapeutic agents
UA71590C2 (en) *	1998-11-13	2004-12-15	Duphar Int Res	Piperazine and piperidine derivatives
CA2405758A1 (en) *	2000-05-12	2001-11-15	Solvay Pharmaceuticals B.V.	Use of compounds having combined dopamine d2, 5-ht1a and alpha adrenoreceptor agonistic action for treating cns disorders
CA2405971C (en) *	2000-05-12	2010-03-30	Solvay Pharmaceuticals B.V.	New piperazine and piperidine compounds

2001
- 2001-05-10 CA CA2405971A patent/CA2405971C/en not_active Expired - Fee Related
- 2001-05-10 AT AT01938214T patent/ATE255578T1/en active
- 2001-05-10 US US10/257,677 patent/US6911448B2/en not_active Expired - Fee Related
- 2001-05-10 TR TR2003/02294T patent/TR200302294T4/en unknown
- 2001-05-10 DK DK01938214T patent/DK1283838T3/en active
- 2001-05-10 NZ NZ522116A patent/NZ522116A/en not_active IP Right Cessation
- 2001-05-10 BR BR0110592-2A patent/BR0110592A/en not_active IP Right Cessation
- 2001-05-10 AU AU6392701A patent/AU6392701A/en active Pending
- 2001-05-10 MX MXPA02011084A patent/MXPA02011084A/en active IP Right Grant
- 2001-05-10 IL IL15217701A patent/IL152177A0/en unknown
- 2001-05-10 HU HU0302016A patent/HUP0302016A2/en unknown
- 2001-05-10 EP EP01938214A patent/EP1283838B1/en not_active Expired - Lifetime
- 2001-05-10 CZ CZ20023721A patent/CZ301464B6/en not_active IP Right Cessation
- 2001-05-10 AU AU2001263927A patent/AU2001263927B2/en not_active Ceased
- 2001-05-10 WO PCT/EP2001/005320 patent/WO2001085725A1/en not_active Ceased
- 2001-05-10 JP JP2001582326A patent/JP2003532729A/en not_active Ceased
- 2001-05-10 PT PT01938214T patent/PT1283838E/en unknown
- 2001-05-10 CN CNB018093302A patent/CN1174979C/en not_active Expired - Fee Related
- 2001-05-10 RU RU2002133458/04A patent/RU2261250C2/en not_active IP Right Cessation
- 2001-05-10 ES ES01938214T patent/ES2211809T3/en not_active Expired - Lifetime
- 2001-05-10 DZ DZ013370A patent/DZ3370A1/en active
- 2001-05-10 DE DE60101386T patent/DE60101386T2/en not_active Expired - Lifetime
- 2001-05-10 PL PL358201A patent/PL198857B1/en not_active IP Right Cessation
- 2001-05-10 SK SK1587-2002A patent/SK286778B6/en not_active IP Right Cessation
- 2001-05-11 AR ARP010102239A patent/AR028443A1/en active IP Right Grant
- 2001-10-05 UA UA2002129990A patent/UA72337C2/en unknown
2002
- 2002-10-08 IL IL152177A patent/IL152177A/en not_active IP Right Cessation
- 2002-10-22 ZA ZA200208537A patent/ZA200208537B/en unknown
- 2002-11-08 NO NO20025365A patent/NO323778B1/en not_active IP Right Cessation
2005
- 2005-05-16 US US11/129,465 patent/US7297699B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
NO20025365D0 (en)	2002-11-08
US7297699B2 (en)	2007-11-20
US6911448B2 (en)	2005-06-28
US20060089366A1 (en)	2006-04-27
RU2261250C2 (en)	2005-09-27
PT1283838E (en)	2004-04-30
CZ20023721A3 (en)	2003-02-12
CA2405971C (en)	2010-03-30
SK15872002A3 (en)	2003-04-01
AU2001263927B2 (en)	2004-09-30
PL358201A1 (en)	2004-08-09
WO2001085725A1 (en)	2001-11-15
HK1055952A1 (en)	2004-01-30
NZ522116A (en)	2004-04-30
DE60101386T2 (en)	2004-05-27
CN1429226A (en)	2003-07-09
AU6392701A (en)	2001-11-20
UA72337C2 (en)	2005-02-15
TR200302294T4 (en)	2004-02-23
SK286778B6 (en)	2009-05-07
NO323778B1 (en)	2007-07-02
EP1283838A1 (en)	2003-02-19
IL152177A (en)	2009-08-03
ATE255578T1 (en)	2003-12-15
EP1283838B1 (en)	2003-12-03
DK1283838T3 (en)	2004-03-22
ES2211809T3 (en)	2004-07-16
MXPA02011084A (en)	2003-03-10
AR028443A1 (en)	2003-05-07
ZA200208537B (en)	2004-01-22
CA2405971A1 (en)	2001-11-15
HUP0302016A2 (en)	2003-09-29
PL198857B1 (en)	2008-07-31
NO20025365L (en)	2002-11-08
BR0110592A (en)	2003-04-01
JP2003532729A (en)	2003-11-05
CN1174979C (en)	2004-11-10
CZ301464B6 (en)	2010-03-10
US20030119849A1 (en)	2003-06-26
IL152177A0 (en)	2003-05-29
DZ3370A1 (en)	2001-11-15

Publication	Publication Date	Title
NO20023787D0 (en)	2002-08-09	Piperazine and piperidine derivatives
DK1325008T3 (en)	2006-02-13	piperazine
ATE397595T1 (en)	2008-06-15	PIPERAZINE DERIVATIVES
IS6546A (en)	2002-09-10	New piperazine derivatives
AR028343A1 (en)	2003-05-07	PIRROLIDINE AND PIPERIDINE DERIVATIVES
DE60103472D1 (en)	2004-07-01	Rohrschneider
DE50105915D1 (en)	2005-05-19	CASES
NO20032585L (en)	2003-07-21	ABCA-1 raising compounds
NO20026125D0 (en)	2002-12-19	Tetrahydropyridine or piperidine heterocyclic derivatives
ATE255578T1 (en)	2003-12-15	PIPERAZINE AND PIPERIDINE COMPOUNDS
NO20043079L (en)	2004-09-21	piperazine
DK1131308T3 (en)	2004-06-28	Piperazine and piperidine derivatives
NO20030276D0 (en)	2003-01-20	Approach
ITMI20000901A0 (en)	2000-04-21	FLUOROELASTOMERS
NO20031572D0 (en)	2003-04-08	Bridged piperazine derivatives
NO20023954L (en)	2002-09-30	Substituted Piperazine Compounds
DE50113112D1 (en)	2007-11-22	circuitry
DE60109953D1 (en)	2005-05-12	CAPACITIVE TRANSFORMER
DK1202966T3 (en)	2004-09-27	Piperidine alcohols
FR2805803B1 (en)	2002-05-17	MONTE MATERIALS
DE60139781D1 (en)	2009-10-15	4-SUBSTITUTED PIPERIDINE COMPOUND
PT1131308E (en)	2004-10-29	NEW PIPERAZINE AND PIPERIDINE COMPOUNDS
FR2814381B1 (en)	2004-06-04	SHREDDER
FI20001114L (en)	2001-11-11	Corner protector
DK1037892T3 (en)	2005-02-07	piperidine

Legal Events

Date	Code	Title	Description
2004-12-30	8364	No opposition during term of opposition