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DE20005297U1 - Active ingredient combination against nicotine addiction - Google Patents

Active ingredient combination against nicotine addiction

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Publication number
DE20005297U1
DE20005297U1 DE20005297U DE20005297U DE20005297U1 DE 20005297 U1 DE20005297 U1 DE 20005297U1 DE 20005297 U DE20005297 U DE 20005297U DE 20005297 U DE20005297 U DE 20005297U DE 20005297 U1 DE20005297 U1 DE 20005297U1
Authority
DE
Germany
Prior art keywords
approx
choline
active ingredient
nicotine addiction
ingredient combination
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE20005297U
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German (de)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
FEHLING LUTZ
Original Assignee
FEHLING LUTZ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by FEHLING LUTZ filed Critical FEHLING LUTZ
Priority to DE20005297U priority Critical patent/DE20005297U1/en
Publication of DE20005297U1 publication Critical patent/DE20005297U1/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/14Quaternary ammonium compounds, e.g. edrophonium, choline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Description

Ludwig Wilhelm Fehling, Stückenberg 43,24226 HeikendorfLudwig Wilhelm Fehling, Stückenberg 43,24226 Heikendorf

-2--2-

Beschreibung
Wirkstofikombination gegen Nikotinabhängigkeit
Description
Combination of active ingredients against nicotine addiction

Die meisten "Designer-Foods" von Durk Pearson und Sandy Shaw basieren auf Erhöhung eines Neurotransmitterspiegels im Gehirn durch Vorläufermischung aus Aminosäure(n) oder Cholin, Vitamin(en), evtl. Mineralien sowie Fruchtzucker, der Insulinauschüttung bewirkt, dadurch Blut-Gehirnschranke öffnet, was den Vorläufern Zugang zum Gehirn verschafft. Quelle: Zeitschrift "Wiener" 5/1990, S. 108, 3. bis 4. SpalteMost of Durk Pearson and Sandy Shaw's "designer foods" are based on increasing neurotransmitter levels in the brain through a precursor mixture of amino acids or choline, vitamins, possibly minerals and fructose, which causes insulin to be released, thereby opening the blood-brain barrier, which gives the precursors access to the brain. Source: "Wiener" magazine 5/1990, p. 108, 3rd to 4th column

Auch Saccharose bewirkt Insulinausschüttung.Sucrose also causes insulin release.

"Life Extension" von Durk Pearson und Sandy Shaw bei Warner Books (C) 1987, Aufl. unauff., S. 372, 1. Abs."Life Extension" by Durk Pearson and Sandy Shaw at Warner Books (C) 1987, unpublished edition, p. 372, 1st paragraph.

Um Azetvlcholin herzustellen, braucht das Gehirn Cholin oder Lezithin sowie Pantothensäure, dto., S. 187,1. Abs.To produce acetylcholine, the brain needs choline or lecithin as well as pantothenic acid, dto., p. 187, 1st paragraph.

Auch Cholinbitartrat und Cholinchlorid sind geeignet,
dto., S. 164,1. Abs.
Choline bitartrate and choline chloride are also suitable,
ibid., p. 164,1. para.

Eine Mischung aus Cholin, Fruktose, Kupfer und den Vitaminen B3, B-5 und B-12 ist als "Gourmet Choline Cooler", ein "Designer-Food" zur Verbesserung von Intelligenz und Gedächtnis auf dem Markt in den USA, ob patentiert, ist mir unbekannt,
o. a. "Wiener", S. 110,1. Spalte, letzter Abs.
A mixture of choline, fructose, copper and vitamins B3, B-5 and B-12 is on the market in the USA as "Gourmet Choline Cooler", a "designer food" to improve intelligence and memory, whether patented or not, is unknown to me.
oa "Wiener", p. 110, 1st column, last paragraph.

3 g Cholin haben geistige Leistungen von Studenten verbessert, o. a. "Life Extension", S. 164 oben3 g of choline improved the mental performance of students, see "Life Extension", p. 164 above

Dimethylaminoäthanolbitartrat erhöht den Azetylcholinspiegel im Gehini. Der aktive Bestandteil ist das Dimethylaminoäthanol.Dimethylaminoethanol bitartrate increases the level of acetylcholine in the brain. The active ingredient is dimethylaminoethanol.

o. a. "Life Extension", S. 484 Mitteo.a. "Life Extension", p. 484 middle

Azetylcholinvorläufer verschlimmern depressive Phase bei manisch-depressiver Psychose, o. a. "Life Extension", S. 187 "Warning"Acetylcholine precursors worsen depressive phase in manic-depressive psychosis, o. a. "Life Extension", p. 187 "Warning"

Der tägliche Bedarf eines Erwachsenen an Pantothensäure liegt bei 8 mg. Z. B. "Die grosse Vitamin und Mineralstofftabelle" von Prof. Dr. I. Elmadfa, Dipl. oec troph D. Fritsche. Prof Dr. H.-D. Cremer, Gräfe und Unzer Verlag (Jahr und Aufl. unauff., aber später als 1986), S. 21, 2. Abs.The daily requirement of pantothenic acid for an adult is 8 mg. For example, "The large vitamin and mineral table" by Prof. Dr. I. Elmadfa, Dipl. oec troph D. Fritsche. Prof. Dr. H.-D. Cremer, Gräfe und Unzer Verlag (year and edition unpublished, but later than 1986), p. 21, 2nd paragraph.

Eine erhöhte Aufnahme wasserlöslicher Vitamine ausser B-12 ist unschädlich. Pantothensäure ist wasserlöslich.An increased intake of water-soluble vitamins other than B-12 is harmless. Pantothenic acid is water-soluble.

dto.. S. 4,2. u. 3. Abs.dto.. p. 4,2. and 3. para.

Die Blut-Gehirn-Schranke schliesst sich nach Einlass einer bestimmten Menge Aminosäuren. "Brain Food" von Dr. Arthur Winter u. Ruth Winter, Verlag Bruno Martin, (C) 1988, S. 35, 2. Abs.The blood-brain barrier closes after a certain amount of amino acids have entered. "Brain Food" by Dr. Arthur Winter and Ruth Winter, Bruno Martin Publishing, (C) 1988, p. 35, 2nd paragraph.

Bekanntlich können Cholinverbindungen zu Gefäßerweiterung fuhren. Erweiterte Gefäße im Gehirn können durch den "Steal-Effect" eine schwächere Durchblutung anderer Gefäße im Gehirn bewirken. Quellen nicht mehr auffindbarIt is known that choline compounds can cause vasodilation. Dilated vessels in the brain can cause weaker blood flow to other vessels in the brain through the "steal effect". Sources can no longer be found

Rosskastanienextrakte wirken gefaßadstringierend.Horse chestnut extracts have a vascular astringent effect.

"Der Gesundheits-Brockhaus" unter Mitarbeit von Prof. Dr. M. Alexander etc., begr. von Prof. Dr. H. Mommseo. Bearb. Dr. med E. Hilka, 3. Aufl., F. A. Brockhaus, Wiesbaden 1984, S. 323"The Health Brockhaus" with the collaboration of Prof. Dr. M. Alexander etc., founded by Prof. Dr. H. Mommseo. Edited by Dr. med. E. Hilka, 3rd edition, F. A. Brockhaus, Wiesbaden 1984, p. 323

Ludwig Wilhelm Fehling, Stückenberg 43, 24226 HeikendorfLudwig Wilhelm Fehling, Stückenberg 43, 24226 Heikendorf

-3--3-

Die Abhängigkeit des Rauchers kommt durch das Rauchen bewirkte vermehrte Bildung von Azetylcholinrezeptoren im Gehirn, an die sich das Nikotin heftet, die nach Aufgeben des Rauchens nicht sofort wieder verschwinden und Entzugserscheinungen bewirken, wenn sie unbesetzt sind, zustande. Das Rauchen kann nicht aufgegeben werden und hat gesundheitliche Beeinträchtigungen zur Folge.The smoker's addiction is caused by the increased formation of acetylcholine receptors in the brain, which nicotine attaches to, and which do not disappear immediately after quitting smoking and cause withdrawal symptoms if they are not occupied. Smoking cannot be stopped and results in health problems.

Prof Dr. Roman Ferstl zitiert in "Therapie gegen den Qualm", 1. Spalte unten bis 5. Spalte oben aus "Kieler Nachrichten11 vom 20.6.92 in Beilage "KN-Joumal", S. 4Prof. Dr. Roman Ferstl quotes in "Therapy against smoke", 1st column bottom to 5th column top from "Kieler Nachrichten 11 of 20.6.92 in the supplement "KN-Joumal", p. 4

Problemproblem

die unbesetzten Azetylcholinrezeptoren müssen ohne die Aufnahme schädlicher Substanzen und ohne Nebenwirkungen besetzt werden.the unoccupied acetylcholine receptors must be occupied without the intake of harmful substances and without side effects.

Erfindunginvention

Das Problem wird durch Einnahme der Wirkstoffkombination, bei Rauchverlangen oder vorbeugend, gelöst. Nach Gelangen der Substanzen aus dem Verdauungstrakt ins Blut passiert Folgendes: Wenn Zucker enthalten ist bewirkt er eine Abgabe von Insulin ins Blut. Dies öffnet die Blut-Gehirn-Schranke, falls geschlossen. Wenn keine Zucker enthalten sind, ist die Öffnung nicht gesichert Die Substanzen gelangen ins Gehirn. Dort wird unter Verwendung von dekm Azetylcholinvorläufer und der Pantothensäure vermehrt Azetylcholin hergestellt. Das Dimethylaminoäthanol (wenn enthalten) führt ebenfalls zur Erhöhung des Azetylcholinspiegels. Unbesetzte, durch Rauchen neugebildete Rezeptoren können besetzt werden. Die Nikotinabhängigkeit vermindert sich. Einer Mangeldurchblutung im Gehirn durch "Steal-Effect" durch das Cholin im Blut wird durch die gefäßspannungserhöhende Wirkung z. B. des Rosskastanienextraktes als gefäßadstringierender Substanz (wenn dieser oder andere Angiotonika enthalten sind), bei Retardwirkung für längere Zeit vorgebeugt. Eine zu grosse Menge Aminosäuren oder die Blut-Gehirn-Schranke schließender Substanzen im Blut kann die Aufnahme der Vorläufer verhindern oder verzögern. In depressiver Phase manisch-depressiver Erkrankung soll die Mischung nicht genommen werden.The problem is solved by taking the combination of active ingredients when you feel like smoking or as a preventative measure. After the substances have passed from the digestive tract into the blood, the following happens: If sugar is present, it causes insulin to be released into the blood. This opens the blood-brain barrier if it is closed. If no sugar is present, the opening is not guaranteed. The substances reach the brain. There, acetylcholine is produced in greater quantities using the acetylcholine precursor and pantothenic acid. Dimethylaminoethanol (if present) also increases the acetylcholine level. Unoccupied receptors newly formed by smoking can be occupied. Nicotine dependence is reduced. Insufficient blood flow in the brain due to the "steal effect" caused by the choline in the blood is prevented for a longer period of time by the vascular tension-increasing effect of, for example, horse chestnut extract as a vascular astringent substance (if this or other angiotonics are present), with a sustained release effect. Too much amino acids or substances that close the blood-brain barrier in the blood can prevent or delay the absorption of the precursors. The mixture should not be taken during the depressive phase of manic-depressive illness.

Claims (1)

1. Wirkstoffkombination gegen Nikotinabhängigkeit gekennzeichnet durch: Grundinhalt bestehend aus a) und/oder b), c), d), e) in Mischungsverhältnis: a) Cholinchlorid und/oder Cholinbitartrat und/oder Lezithin (evtl. mit hohem Phosphatidylcholinanteil) und/oder Phosphatidylcholin und/oder Cholin (ca. 1 mg bis 30 g) b) Dimethylaminoäthanol (ca. 0 mg bis 1000 mg) c) Angiotonikum (eins oder mehrere), evtl. mit Retardwirkung (z. B. Rosskastanienextrakt) (ca. 0 mg bis 1000 mg) bzw. nach empfohlenen Dosierungen d) Fruktose und/oder Saccharose und/oder Glukose (ca. 0 bis 20 g) e) Pantothensäure und/oder Panthenol und/oder Pantothenate (ca. 0,1 mg bis 1000 mg. 1. Active ingredient combination against nicotine addiction characterized by : Basic content consisting of a) and/or b), c), d), e) in mixing ratio: a) Choline chloride and/or choline bitartrate and/or lecithin (possibly with a high phosphatidylcholine content) and/or phosphatidylcholine and/or choline (approx. 1 mg to 30 g) b) Dimethylaminoethanol (approx. 0 mg to 1000 mg) c) Angiotonic (one or more), possibly with sustained release effect (e.g. horse chestnut extract) (approx. 0 mg to 1000 mg) or according to recommended dosages d) Fructose and/or sucrose and/or glucose (approx. 0 to 20 g) e) Pantothenic acid and/or panthenol and/or pantothenates (approx. 0.1 mg to 1000 mg.
DE20005297U 2000-03-21 2000-03-21 Active ingredient combination against nicotine addiction Expired - Lifetime DE20005297U1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
DE20005297U DE20005297U1 (en) 2000-03-21 2000-03-21 Active ingredient combination against nicotine addiction

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE20005297U DE20005297U1 (en) 2000-03-21 2000-03-21 Active ingredient combination against nicotine addiction

Publications (1)

Publication Number Publication Date
DE20005297U1 true DE20005297U1 (en) 2000-07-27

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DE20005297U Expired - Lifetime DE20005297U1 (en) 2000-03-21 2000-03-21 Active ingredient combination against nicotine addiction

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DE (1) DE20005297U1 (en)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003035092A1 (en) 2001-10-26 2003-05-01 Angiolab Inc. Composition containing horse chestnut extract for anti-angiogenic and matrix metalloproteinase inhibitory activity

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2003035092A1 (en) 2001-10-26 2003-05-01 Angiolab Inc. Composition containing horse chestnut extract for anti-angiogenic and matrix metalloproteinase inhibitory activity
EP1438059A4 (en) * 2001-10-26 2008-01-23 Angiolab Inc Composition containing horse chestnut extract for anti-angiogenic and matrix metalloproteinase inhibitory activity

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Legal Events

Date Code Title Description
R207 Utility model specification

Effective date: 20000831

R150 Utility model maintained after payment of first maintenance fee after three years

Effective date: 20030506

R157 Lapse of ip right after 6 years

Effective date: 20061003