CU23338A3 - XA FACTOR INHIBITORS AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION WATERFALL - Google Patents
XA FACTOR INHIBITORS AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION WATERFALLInfo
- Publication number
- CU23338A3 CU23338A3 CU20040116A CU20040116A CU23338A3 CU 23338 A3 CU23338 A3 CU 23338A3 CU 20040116 A CU20040116 A CU 20040116A CU 20040116 A CU20040116 A CU 20040116A CU 23338 A3 CU23338 A3 CU 23338A3
- Authority
- CU
- Cuba
- Prior art keywords
- formula
- serine proteases
- factor inhibitors
- proteases involved
- compounds
- Prior art date
Links
- 102000012479 Serine Proteases Human genes 0.000 title 1
- 108010022999 Serine Proteases Proteins 0.000 title 1
- 230000015271 coagulation Effects 0.000 title 1
- 238000005345 coagulation Methods 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 4
- 208000007536 Thrombosis Diseases 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención proporciona compuestos de fórmula ESPACIO PARA FÓRMULA en la que A,B,C,G y W a la1 tienen cualquiera de los valores definidos en la memoria descriptiva, y sales farmacéuticamente aceptables de los mismos, que son útiles para tratar trastornos trombóticos. También se describen composiciones farmacéuticas que comprenden uno o más compuestos de fórmula I, procedimientos para la preparación de compuestos de fórmula I e intermedios útiles para la preparación de compuestos de fórmula I.The present invention provides compounds of the formula SPACE FOR FORMULA in which A, B, C, G and W at 1 have any of the values defined in the specification, and pharmaceutically acceptable salts thereof, which are useful for treating thrombotic disorders. . Also described are pharmaceutical compositions comprising one or more compounds of formula I, processes for the preparation of compounds of formula I and intermediates useful for the preparation of compounds of formula I.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20040116A CU23338A3 (en) | 2004-05-31 | 2004-05-31 | XA FACTOR INHIBITORS AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION WATERFALL |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CU20040116A CU23338A3 (en) | 2004-05-31 | 2004-05-31 | XA FACTOR INHIBITORS AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION WATERFALL |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU23338A3 true CU23338A3 (en) | 2009-01-20 |
Family
ID=40348308
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU20040116A CU23338A3 (en) | 2004-05-31 | 2004-05-31 | XA FACTOR INHIBITORS AND OTHER SERINE PROTEASES INVOLVED IN THE COAGULATION WATERFALL |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU23338A3 (en) |
-
2004
- 2004-05-31 CU CU20040116A patent/CU23338A3/en not_active IP Right Cessation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FD | Lapse (for not paying fees) |