CU23993B1 - NEW DERIVATIVES OF AZABICICLO [3.2.0] PET-3-ILO AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM - Google Patents
NEW DERIVATIVES OF AZABICICLO [3.2.0] PET-3-ILO AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEMInfo
- Publication number
- CU23993B1 CU23993B1 CU2010000236A CU20100236A CU23993B1 CU 23993 B1 CU23993 B1 CU 23993B1 CU 2010000236 A CU2010000236 A CU 2010000236A CU 20100236 A CU20100236 A CU 20100236A CU 23993 B1 CU23993 B1 CU 23993B1
- Authority
- CU
- Cuba
- Prior art keywords
- azabiciclo
- ilo
- pet
- pharmaceutical compositions
- compositions containing
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 125000002947 alkylene group Chemical group 0.000 abstract 1
- 229940079593 drug Drugs 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- -1 hept-3-yl compounds Chemical class 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/52—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring condensed with a ring other than six-membered
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/16—Central respiratory analeptics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Urology & Nephrology (AREA)
- Child & Adolescent Psychology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Anesthesiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
Abstract
Compuestos de azabiciclo [3.2.0] hept-3-ilo de fórmula (I): en la que: ALK representa una cadena alquileno, W representa un grupo ó en el que R y R' son tales como se han definido en la descripción. Medicamento.Azabicyclo [3.2.0] hept-3-yl compounds of formula (I): in which: ALK represents an alkylene chain, W represents a group or in which R and R 'are as defined in the description . Medicine.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR0905957A FR2953514B1 (en) | 2009-12-09 | 2009-12-09 | NOVEL AZABICYCLO [3.2.0] HEPT-3-YL DERIVATIVES, PROCESS FOR PREPARING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| CU20100236A7 CU20100236A7 (en) | 2011-11-15 |
| CU23993B1 true CU23993B1 (en) | 2014-04-24 |
Family
ID=42133738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CU2010000236A CU23993B1 (en) | 2009-12-09 | 2010-12-02 | NEW DERIVATIVES OF AZABICICLO [3.2.0] PET-3-ILO AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
Country Status (44)
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI9300625B (en) * | 1993-12-02 | 2002-02-28 | Basf Aktiengesellschaft | N-substituted azabicycloheptane derivatives, their preparation and use |
| DE4341402A1 (en) * | 1993-12-04 | 1995-06-08 | Basf Ag | N-substituted azabicycloheptane derivatives, their preparation and use |
| DE4427647A1 (en) * | 1994-08-04 | 1996-02-08 | Basf Ag | N-substituted azabicycloheptane derivatives, their preparation and use |
| FR2866647B1 (en) * | 2004-02-20 | 2006-10-27 | Servier Lab | NOVEL AZABICYCLIC DERIVATIVES, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM |
-
2009
- 2009-12-09 FR FR0905957A patent/FR2953514B1/en not_active Expired - Fee Related
-
2010
- 2010-11-19 MY MYPI2010005458 patent/MY150598A/en unknown
- 2010-11-21 IL IL209463A patent/IL209463A/en not_active IP Right Cessation
- 2010-11-22 UY UY0001033046A patent/UY33046A/en unknown
- 2010-11-22 JO JO2010408A patent/JO2880B1/en active
- 2010-11-23 SG SG2010085959A patent/SG172543A1/en unknown
- 2010-11-24 CR CR11811A patent/CR11811A/en not_active Application Discontinuation
- 2010-11-25 PE PE2010001083A patent/PE20110542A1/en not_active Application Discontinuation
- 2010-11-25 AU AU2010246426A patent/AU2010246426B2/en not_active Ceased
- 2010-11-26 TW TW099141093A patent/TWI419875B/en not_active IP Right Cessation
- 2010-11-26 CL CL2010001309A patent/CL2010001309A1/en unknown
- 2010-11-29 CO CO10150441A patent/CO6280059A1/en active IP Right Grant
- 2010-11-29 CN CN2010105733405A patent/CN102127004B/en not_active Expired - Fee Related
- 2010-11-30 MX MX2010013093A patent/MX2010013093A/en active IP Right Grant
- 2010-12-01 MA MA33380A patent/MA32444B1/en unknown
- 2010-12-01 ZA ZA2010/08651A patent/ZA201008651B/en unknown
- 2010-12-01 EC EC2010010649A patent/ECSP10010649A/en unknown
- 2010-12-01 AP AP2010005489A patent/AP2755A/en active
- 2010-12-02 NI NI201000206A patent/NI201000206A/en unknown
- 2010-12-02 CU CU2010000236A patent/CU23993B1/en not_active IP Right Cessation
- 2010-12-02 SV SV2010003746A patent/SV2010003746A/en unknown
- 2010-12-03 CA CA2724151A patent/CA2724151C/en not_active Expired - Fee Related
- 2010-12-06 UA UAA201014568A patent/UA106721C2/en unknown
- 2010-12-06 AR ARP100104487A patent/AR079268A1/en unknown
- 2010-12-07 KR KR1020100124116A patent/KR101292705B1/en not_active Expired - Fee Related
- 2010-12-07 SA SA110320007A patent/SA110320007B1/en unknown
- 2010-12-07 EA EA201001755A patent/EA018971B1/en not_active IP Right Cessation
- 2010-12-07 GE GEAP201012026A patent/GEP20135801B/en unknown
- 2010-12-07 NZ NZ589763A patent/NZ589763A/en not_active IP Right Cessation
- 2010-12-07 US US12/928,237 patent/US8008337B2/en not_active Expired - Fee Related
- 2010-12-08 HN HN2010002593A patent/HN2010002593A/en unknown
- 2010-12-08 PL PL10290642T patent/PL2332910T3/en unknown
- 2010-12-08 BR BRPI1005270-4A patent/BRPI1005270A2/en not_active IP Right Cessation
- 2010-12-08 EP EP10290642A patent/EP2332910B1/en active Active
- 2010-12-08 WO PCT/FR2010/000820 patent/WO2011070250A1/en not_active Ceased
- 2010-12-08 ME MEP-2013-42A patent/ME01504B/en unknown
- 2010-12-08 ES ES10290642T patent/ES2405206T3/en active Active
- 2010-12-08 SI SI201030183T patent/SI2332910T1/en unknown
- 2010-12-08 RS RS20130092A patent/RS52698B/en unknown
- 2010-12-08 PT PT102906427T patent/PT2332910E/en unknown
- 2010-12-08 DK DK10290642.7T patent/DK2332910T3/en active
- 2010-12-09 JP JP2010274280A patent/JP5511645B2/en not_active Expired - Fee Related
-
2013
- 2013-04-04 HR HRP20130307AT patent/HRP20130307T1/en unknown
- 2013-04-29 CY CY20131100354T patent/CY1113971T1/en unknown
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Grant of patent | ||
| FD | Lapse (for not paying fees) |