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CN112209819A - Preparation method of D-pantoic acid calcium - Google Patents

Preparation method of D-pantoic acid calcium Download PDF

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Publication number
CN112209819A
CN112209819A CN202011034914.1A CN202011034914A CN112209819A CN 112209819 A CN112209819 A CN 112209819A CN 202011034914 A CN202011034914 A CN 202011034914A CN 112209819 A CN112209819 A CN 112209819A
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Prior art keywords
calcium
pantoic acid
pantoate
preparation
solution containing
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CN202011034914.1A
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Inventor
陈修
王浩
杜斌
段小瑞
汪洪湖
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Anhui Tiger Biotechnology Co ltd
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Anhui Tiger Biotechnology Co ltd
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C51/00Preparation of carboxylic acids or their salts, halides or anhydrides
    • C07C51/41Preparation of salts of carboxylic acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07BGENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07Optical isomers

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Oil, Petroleum & Natural Gas (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

The invention provides a preparation method of D-pantoic acid calcium, which comprises the following steps: reacting D-pantoic acid lactone with calcium hydroxide to obtain a mixed solution containing D-pantoic acid calcium. The preparation method provided by the invention is simple and feasible, the solvent is safe and pollution-free, stable crystals can be formed at low temperature, and the obtained D-calcium pantoate crystals are not sticky to the wall and are not agglomerated, and have few impurities and high purity.

Description

Preparation method of D-pantoic acid calcium
Technical Field
The invention belongs to the technical field of chemical production, and relates to a preparation method of D-pantoic acid calcium.
Background
The D-pantoic acid lactone is derived from chiral resolution of DL-pantoic acid lactone, the DL-pantoic acid lactone is an organic chemical, and the D-pantoic acid lactone obtained by chiral resolution can be used for synthesizing D-panthenol or D-panthenyl ethyl ether and the like used for cosmetics. The greatest application of D-pantoic acid lactone is to synthesize D-calcium pantothenate, which is also called pantothenic acid and is also called vitamin B5, and the D-calcium pantothenate is a water-soluble B-group vitamin which is widely used in food, medicine, feed additives and the like.
In the synthesis of calcium D-pantothenate, the presence of calcium D-pantoate is found in both the mother liquor and the product, but since the content thereof is too low, studies on the presence of calcium D-pantoate cannot be made, and the application direction of the calcium D-pantoate cannot be judged, it is necessary to provide a production method capable of obtaining high-quality calcium D-pantoate.
Disclosure of Invention
The invention aims to provide a preparation method of D-calcium pantoate, which is simple and easy to implement, has safe and pollution-free solvent, can form stable crystals at low temperature, and the obtained D-calcium pantoate crystals are not sticky to walls, are not agglomerated, have few impurities and have high purity.
In order to achieve the purpose, the invention adopts the following technical scheme:
in a first aspect, the present invention provides a method for preparing D-pantoic acid calcium, the method comprising: reacting D-pantoic acid lactone with calcium hydroxide to obtain a mixed solution containing D-pantoic acid calcium.
In the present invention, the molar ratio of D-pantolactone to calcium hydroxide is 1 (1-1.2), for example, 1: 1.1.
In the present invention, the reaction is carried out in a solvent, and the solvent in the present invention is water.
The invention preferably selects water as solvent, and has the advantages of safety and environmental protection.
In order to avoid waste of the solvent and ensure easy handling of the D-pantoic acid calcium, the mass ratio of the solvent to the D-pantoic acid lactone is (2-5: 1), such as 2.5:1, 3:1, 3.5:1, 4:1, 4.5:1 and the like.
The calcium hydroxide is dropwise added into a reaction system in the form of a calcium hydroxide aqueous solution.
If the calcium hydroxide (or the calcium hydroxide aqueous solution) is directly added into a reaction system, implosion can be caused, rapid crystallization and precipitation can be carried out during the reaction, and the crystals are stirred and instantly locked, so that the impurities of the crystals are more, the purity is lower, and the separation is difficult.
In a preferred embodiment of the present invention, the concentration of the aqueous calcium hydroxide solution is 15 to 30 wt%, such as 16 wt%, 18 wt%, 20 wt%, 22 wt%, 25 wt%, 28 wt%, etc.
The concentration of the calcium hydroxide aqueous solution is preferably 15-30 wt%, within the range, the reaction rate is moderate, and the reaction time is suitable.
The dropping rate of the invention is 5-10mL/min, such as 6mL/min, 7mL/min, 8mL/min, 9mL/min and the like.
In order to ensure the yield and purity of the final product, the reaction temperature is 60-80 deg.C, such as 62 deg.C, 65 deg.C, 68 deg.C, 70 deg.C, 72 deg.C, 75 deg.C, 78 deg.C, etc.
The reaction temperature of 60-80 ℃ is optimized in the invention, the reaction rate is moderate within the reaction temperature range, and the finally obtained D-calcium pantoate has few impurities and high purity.
The reaction time of the invention is 1-3h, such as 1.2h, 1.5h, 1.8h, 2.0h, 2.2h, 2.5h, 2.8h and the like.
As a preferable technical solution of the present invention, the preparation method further comprises: and cooling the mixed solution containing the D-calcium pantoate for crystallization, and then filtering and drying to obtain the D-calcium pantoate.
The temperature reduction is carried out under the condition of stirring.
As a preferred technical scheme, the preparation method provided by the invention comprises the following steps:
(1) dropwise adding a calcium hydroxide aqueous solution into a D-pantoic acid lactone aqueous solution for reaction to obtain a mixed solution containing D-pantoic acid calcium;
(2) and cooling the mixed solution containing the D-calcium pantoate under the stirring condition for crystallization, filtering and drying to obtain the D-calcium pantoate.
Compared with the prior art, the invention has the following beneficial effects:
(1) the preparation method provided by the invention is simple and feasible, and the raw materials are easy to obtain;
(2) by controlling the concentration, the dropping speed, the reaction temperature and other conditions of the calcium hydroxide aqueous solution, the finally obtained D-calcium pantoate has less impurities, high purity and higher yield.
Detailed Description
The technical solution of the present invention is further explained by the following embodiments. It should be understood by those skilled in the art that the examples are only for the understanding of the present invention and should not be construed as the specific limitations of the present invention.
Example 1
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) sequentially adding 100g of deionized water and 50g of D-pantoic acid lactone with the specific rotation degree of +46 degrees into a clean 500mL single-mouth bottle, stirring and dissolving, then dropwise adding 114g of 25 wt% calcium hydroxide aqueous solution, and reacting for 1h at 60 ℃ to obtain mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing, filtering and drying to obtain the D-calcium pantoate.
Example 2
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) sequentially adding 100g of deionized water and 50g of D-pantoic acid lactone with the specific rotation degree of +46 degrees into a clean 500mL single-mouth bottle, stirring and dissolving, then dropwise adding 114g of 25 wt% calcium hydroxide aqueous solution, and reacting for 1h at 80 ℃ to obtain mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing, filtering and drying to obtain the D-calcium pantoate.
Example 3
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) sequentially adding 100g of deionized water and 50g of D-pantoic acid lactone with the specific rotation degree of +46 degrees into a clean 500mL single-mouth bottle, stirring and dissolving, then dropwise adding 190g of 15 wt% calcium hydroxide aqueous solution, and reacting for 3h at 80 ℃ to obtain mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing for 6 hours, filtering and drying to obtain the D-calcium pantoate.
Example 4
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) sequentially adding 100g of deionized water and 50g of D-pantoic acid lactone with the specific rotation degree of +46 degrees into a clean 500mL single-mouth bottle, stirring and dissolving, then dropwise adding 142.5g of 20 wt% calcium hydroxide aqueous solution, and reacting for 1h at 60 ℃ to obtain mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing, filtering and drying to obtain the D-calcium pantoate.
Comparative example 1
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) sequentially adding 100g of deionized water and 50g of D-pantoic acid lactone with the specific rotation degree of +46 degrees into a clean 500mL single-mouth bottle, stirring and dissolving, then dropwise adding 95g of 40 wt% calcium hydroxide aqueous solution, and reacting for 1h at 80 ℃ to obtain mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing, filtering and drying to obtain the D-calcium pantoate.
Comparative example 2
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) sequentially adding 100g of methanol and 50g of D-pantoic acid lactone with the specific rotation degree of +46 degrees into a clean 500mL single-mouth bottle, stirring and dissolving, then dropwise adding 142.5g of 20 wt% calcium hydroxide aqueous solution, and reacting for 1h at 60 ℃ to obtain mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing, filtering and drying to obtain the D-calcium pantoate.
Comparative example 3
A preparation method of D-pantoic acid calcium comprises the following steps:
(1) adding 100g of methanol into a clean 500mL single-mouth bottle, adding 50g of D-pantoic acid lactone with the specific rotation degree of +46 ℃ and 142.5g of 20 wt% calcium hydroxide aqueous solution under stirring, and reacting for 1h at 60 ℃ to obtain a mixed solution containing D-pantoic acid calcium;
(2) and (3) cooling the mixed solution containing the D-calcium pantoate to-5 ℃ under stirring, preserving heat, crystallizing, filtering and drying to obtain the D-calcium pantoate.
Performance testing
The samples provided in examples 1 to 4 and comparative examples 1 to 3 were weighed and the yield thereof was calculated, and the results are shown in table 1:
TABLE 1
Figure BDA0002704892260000041
Figure BDA0002704892260000051
Note: comparative example 1 suddenly agglomerates and adheres to the reaction vessel in the process of temperature reduction, loose particles cannot be formed, impurities are more, and separation is difficult, so that the particles are not recovered; comparative example 3 was already imploded in the reaction vessel at the beginning of the reaction and no subsequent steps could be performed.
The embodiment and the performance test show that the preparation method provided by the invention is simple and feasible, the prepared D-calcium pantoate is a stable crystal, does not stick to the wall, is easy to carry out subsequent treatment, and has high purity and high yield of the product.
As can be seen from the comparison of examples 2-3 with comparative example 1, the concentration of the aqueous calcium hydroxide solution provided by the present invention needs to be in the range of 15-30 wt% to obtain D-pantoic acid calcium which is not sticky to the wall and is easy for subsequent treatment; as can be seen from the comparison between example 4 and comparative example 2, the method can adopt water as a solvent to prepare the D-pantoic acid calcium, and the water as the solvent is safe and environment-friendly; as can be seen from a comparison of example 4 and comparative example 3, the calcium hydroxide solvent of the present invention is required to react with D-pantoic acid lactone in the form of a dropwise addition.
The applicant states that the present invention is illustrated by the above examples to the preparation of the calcium D-pantoate of the present invention, but the present invention is not limited to the above detailed methods, i.e. it is not meant that the present invention must rely on the above detailed methods to be practiced. It should be understood by those skilled in the art that any modification of the present invention, equivalent substitutions of the raw materials of the product of the present invention, addition of auxiliary components, selection of specific modes, etc., are within the scope and disclosure of the present invention.

Claims (10)

1. A preparation method of D-pantoic acid calcium, characterized in that, the preparation method comprises: reacting D-pantoic acid lactone with calcium hydroxide to obtain a mixed solution containing D-pantoic acid calcium.
2. The method according to claim 1, wherein the molar ratio of D-pantolactone to calcium hydroxide is 1 (1-1.2).
3. The method of claim 1 or 2, wherein the reaction is carried out in a solvent.
4. The method according to claim 3, wherein the solvent is water.
5. The production method according to claim 3 or 4, characterized in that the mass ratio of the solvent to the D-pantoic acid lactone is (2-5): 1.
6. The production method according to any one of claims 1 to 5, wherein the calcium hydroxide is added dropwise to the reaction system in the form of an aqueous calcium hydroxide solution.
7. The method according to claim 6, wherein the concentration of the aqueous calcium hydroxide solution is 15 to 30 wt%;
and/or the dropping rate is 5-10 mL/min.
8. The method for preparing according to any one of claims 1 to 7, wherein the temperature of the reaction is 60 to 80 ℃;
and/or the reaction time is 1-3 h.
9. The production method according to any one of claims 1 to 8, further comprising: cooling the mixed solution containing the D-calcium pantoate for crystallization, and then filtering and drying to obtain the D-calcium pantoate;
preferably, the temperature reduction is performed under stirring.
10. The production method according to any one of claims 1 to 8, characterized by comprising:
(1) dropwise adding a calcium hydroxide aqueous solution into a D-pantoic acid lactone aqueous solution for reaction to obtain a mixed solution containing D-pantoic acid calcium;
(2) and cooling the mixed solution containing the D-calcium pantoate under the stirring condition for crystallization, filtering and drying to obtain the D-calcium pantoate.
CN202011034914.1A 2020-09-27 2020-09-27 Preparation method of D-pantoic acid calcium Pending CN112209819A (en)

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Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114394948A (en) * 2021-12-29 2022-04-26 安徽泰格生物科技有限公司 Recycling method of panthenol mother liquor
CN116217428A (en) * 2022-12-22 2023-06-06 黑龙江新和成生物科技有限公司 Methanol hydrate crystal of D-calcium pantothenate and process for producing D-calcium pantothenate
CN116589437A (en) * 2023-04-07 2023-08-15 天津大学 Continuous crystallization method of D-pantolactone

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110835185A (en) * 2019-12-02 2020-02-25 安徽华恒生物科技股份有限公司 Method for separating acid and ester from mixed solution

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN110835185A (en) * 2019-12-02 2020-02-25 安徽华恒生物科技股份有限公司 Method for separating acid and ester from mixed solution

Cited By (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN114394948A (en) * 2021-12-29 2022-04-26 安徽泰格生物科技有限公司 Recycling method of panthenol mother liquor
CN116217428A (en) * 2022-12-22 2023-06-06 黑龙江新和成生物科技有限公司 Methanol hydrate crystal of D-calcium pantothenate and process for producing D-calcium pantothenate
CN116217428B (en) * 2022-12-22 2024-04-02 黑龙江新和成生物科技有限公司 Methanol hydrate crystal of D-calcium pantothenate and process for producing D-calcium pantothenate
CN116589437A (en) * 2023-04-07 2023-08-15 天津大学 Continuous crystallization method of D-pantolactone
CN116589437B (en) * 2023-04-07 2024-11-15 天津大学 A continuous crystallization method for D-pantolactone

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