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CL2018001744A1 - Compuestos depsipeptídicos como anthelmínticos - Google Patents

Compuestos depsipeptídicos como anthelmínticos

Info

Publication number
CL2018001744A1
CL2018001744A1 CL2018001744A CL2018001744A CL2018001744A1 CL 2018001744 A1 CL2018001744 A1 CL 2018001744A1 CL 2018001744 A CL2018001744 A CL 2018001744A CL 2018001744 A CL2018001744 A CL 2018001744A CL 2018001744 A1 CL2018001744 A1 CL 2018001744A1
Authority
CL
Chile
Prior art keywords
compounds
animals
anthelmintics
parasites
depsipeptide compounds
Prior art date
Application number
CL2018001744A
Other languages
English (en)
Inventor
Fallois Loic Le Hir De
Gregory Pacofsky
Alan Long
Charles Meng
Hyoung Ik Lee
Original Assignee
Merial Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merial Inc filed Critical Merial Inc
Publication of CL2018001744A1 publication Critical patent/CL2018001744A1/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • A61K38/15—Depsipeptides; Derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/10—Anthelmintics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K11/00—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02—Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Engineering & Computer Science (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Epidemiology (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Dentistry (AREA)
  • Wood Science & Technology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Immunology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Peptides Or Proteins (AREA)

Abstract

COMPUESTOS DEPSIPEPTÍDICOS CÍCLICOS DE FÓRMULA (I) Y COMPOSICIONES QUE COMPRENDEN LOS COMPUESTOS QUE SON EFICACES CONTRA PARÁSITOS QUE DAÑAN A LOS ANIMALES, INCLUYENDO A LOS HUMANOS. LOS COMPUESTOS Y LAS COMPOSICIONES SE PUEDEN USAR PARA COMBATIR PARÁSITOS DENTRO O SOBRE LOS ANIMALES INCLUYENDO A MAMÍFEROS Y AVES. LA INVENCIÓN TAMBIÉN PROVEE UN MÉTODO MEJORADO PARA ERRADICAR, CONTROLAR Y PREVENIR UNA INFESTACIÓN POR PARÁSITOS EN ANIMALES, INCLUYENDO AVES Y MAMÍFEROS.
CL2018001744A 2015-12-28 2018-06-25 Compuestos depsipeptídicos como anthelmínticos CL2018001744A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US201562272040P 2015-12-28 2015-12-28

Publications (1)

Publication Number Publication Date
CL2018001744A1 true CL2018001744A1 (es) 2018-08-17

Family

ID=57868331

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2018001744A CL2018001744A1 (es) 2015-12-28 2018-06-25 Compuestos depsipeptídicos como anthelmínticos

Country Status (23)

Country Link
US (3) US10344056B2 (es)
EP (1) EP3397638B1 (es)
JP (1) JP6943859B2 (es)
KR (2) KR102427124B1 (es)
CN (1) CN108699052B (es)
AR (1) AR107249A1 (es)
AU (2) AU2016380868B2 (es)
BR (1) BR112018013369A2 (es)
CA (1) CA3009867C (es)
CL (1) CL2018001744A1 (es)
CO (1) CO2018006527A2 (es)
HK (1) HK1255391A1 (es)
HU (1) HUE065907T2 (es)
IL (1) IL260262B2 (es)
MX (1) MX2018007948A (es)
MY (1) MY194716A (es)
NZ (1) NZ743913A (es)
PH (1) PH12018501367B1 (es)
RU (2) RU2715556C2 (es)
SG (1) SG11201805368YA (es)
TW (1) TWI787165B (es)
UY (1) UY37050A (es)
WO (1) WO2017116702A1 (es)

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SG11201805368YA (en) 2015-12-28 2018-07-30 Merial Inc Anthelmintic depsipeptide compounds
WO2018039508A1 (en) 2016-08-25 2018-03-01 Merial, Inc. Method for reducing unwanted effects in parasiticidal treatments
WO2018093920A1 (en) 2016-11-16 2018-05-24 Merial, Inc. Anthelmintic depsipeptide compounds
HRP20230870T1 (hr) 2017-02-08 2023-11-10 Boehringer Ingelheim Animal Health USA Inc. Model in vivo za infekciju parazitnim crvima i postupak ocjenjivanja antiparazitnih spojeva, uključujući spojeve koji djeluju protiv pseće dirofilarioze
KR102795744B1 (ko) 2017-11-07 2025-04-11 엘랑코 애니멀 헬스 게엄베하 시클릭 뎁시펩티드의 합성 방법
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WO2020146338A1 (en) 2019-01-10 2020-07-16 Zoetis Services Llc Anthelmintic laboratory animal model for heartworm
US11560388B2 (en) 2019-03-19 2023-01-24 Boehringer Ingelheim Vetmedica Gmbh Anthelmintic aza-benzothiophene and aza-benzofuran compounds
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EP4185589A1 (en) 2020-05-29 2023-05-31 Boehringer Ingelheim Animal Health USA Inc. Anthelmintic heterocyclic compounds
EP4262789A1 (en) 2020-12-21 2023-10-25 Boehringer Ingelheim Vetmedica GmbH Parasiticidal collar comprising isoxazoline compounds
JP2025507585A (ja) 2022-02-17 2025-03-21 ベーリンガー インゲルハイム フェトメディカ ゲーエムベーハー 流体製品メーラーを提供する方法及びシステム
WO2025057117A1 (en) * 2023-09-15 2025-03-20 Animol Discovery, Inc. Antiparasitic cyclic depsipeptides

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Also Published As

Publication number Publication date
TW201726670A (zh) 2017-08-01
IL260262A (en) 2018-07-31
CN108699052A (zh) 2018-10-23
TWI787165B (zh) 2022-12-21
AU2020200854B2 (en) 2021-08-05
CA3009867A1 (en) 2017-07-06
MY194716A (en) 2022-12-15
NZ743913A (en) 2019-04-26
EP3397638B1 (en) 2023-08-23
KR20180100349A (ko) 2018-09-10
JP6943859B2 (ja) 2021-10-06
CA3009867C (en) 2022-05-31
US11230571B2 (en) 2022-01-25
US12018048B2 (en) 2024-06-25
RU2020107484A (ru) 2020-03-19
BR112018013369A2 (pt) 2019-02-19
KR20220003663A (ko) 2022-01-10
JP2019504050A (ja) 2019-02-14
HUE065907T2 (hu) 2024-06-28
PH12018501367A1 (en) 2019-02-27
AU2020200854A1 (en) 2020-02-27
SG11201805368YA (en) 2018-07-30
AU2016380868A1 (en) 2018-07-19
MX2018007948A (es) 2018-08-01
CO2018006527A2 (es) 2018-07-10
RU2018127195A3 (es) 2020-01-30
PH12018501367B1 (en) 2022-10-21
RU2715556C2 (ru) 2020-03-02
KR102427124B1 (ko) 2022-07-28
RU2018127195A (ru) 2020-01-30
EP3397638A1 (en) 2018-11-07
US20170233438A1 (en) 2017-08-17
AR107249A1 (es) 2018-04-11
AU2016380868B2 (en) 2019-11-28
HK1255391A1 (zh) 2019-08-16
UY37050A (es) 2017-07-31
US20190248840A1 (en) 2019-08-15
US10344056B2 (en) 2019-07-09
IL260262B2 (en) 2023-06-01
WO2017116702A1 (en) 2017-07-06
US20220098241A1 (en) 2022-03-31
CN108699052B (zh) 2022-04-29

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