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CL2016003283A1 - Formulación compuesta para administración oral que comprende ezetimiba y rosuvastatina y un procedimiento para su preparación - Google Patents

Formulación compuesta para administración oral que comprende ezetimiba y rosuvastatina y un procedimiento para su preparación

Info

Publication number
CL2016003283A1
CL2016003283A1 CL2016003283A CL2016003283A CL2016003283A1 CL 2016003283 A1 CL2016003283 A1 CL 2016003283A1 CL 2016003283 A CL2016003283 A CL 2016003283A CL 2016003283 A CL2016003283 A CL 2016003283A CL 2016003283 A1 CL2016003283 A1 CL 2016003283A1
Authority
CL
Chile
Prior art keywords
ezetimibe
rosuvastatin
oral administration
procedure
preparation
Prior art date
Application number
CL2016003283A
Other languages
English (en)
Spanish (es)
Inventor
Yong Ii Kim
Jae Hyun Park
Jong Soo Woo
Seung Jun Lee
Ha Young Jeong
Kyong Soo Kim
Original Assignee
Hanmi Pharm Ind Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=54938391&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2016003283(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Hanmi Pharm Ind Co Ltd filed Critical Hanmi Pharm Ind Co Ltd
Publication of CL2016003283A1 publication Critical patent/CL2016003283A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2072Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2077Tablets comprising drug-containing microparticles in a substantial amount of supporting matrix; Multiparticulate tablets
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/397Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having four-membered rings, e.g. azetidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1682Processes
    • A61K9/1694Processes resulting in granules or microspheres of the matrix type containing more than 5% of excipient

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Obesity (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
CL2016003283A 2014-06-25 2016-12-21 Formulación compuesta para administración oral que comprende ezetimiba y rosuvastatina y un procedimiento para su preparación CL2016003283A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
KR1020140078388A KR101977785B1 (ko) 2014-06-25 2014-06-25 에제티미브 및 로수바스타틴을 포함하는 경구용 복합제제 및 그 제조방법

Publications (1)

Publication Number Publication Date
CL2016003283A1 true CL2016003283A1 (es) 2017-07-28

Family

ID=54938391

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2016003283A CL2016003283A1 (es) 2014-06-25 2016-12-21 Formulación compuesta para administración oral que comprende ezetimiba y rosuvastatina y un procedimiento para su preparación

Country Status (10)

Country Link
KR (1) KR101977785B1 (fr)
AR (1) AR100977A1 (fr)
BR (1) BR112016030111A2 (fr)
CL (1) CL2016003283A1 (fr)
EC (1) ECSP16096477A (fr)
JO (1) JOP20150154B1 (fr)
SG (2) SG11201610748RA (fr)
TW (1) TWI700100B (fr)
UY (1) UY36190A (fr)
WO (1) WO2015199356A1 (fr)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CZ2016539A3 (cs) 2016-09-05 2018-03-14 Zentiva, K.S. Farmaceutická kompozice obsahující dvě rozdílné účinné látky a způsob její přípravy
CZ2016538A3 (cs) 2016-09-05 2018-03-14 Zentiva, K.S. Farmaceutická kompozice obsahující dvě rozdílné účinné látky
KR102206535B1 (ko) * 2016-11-29 2021-01-22 한미약품 주식회사 에제티미브 및 로수바스타틴을 포함하는 경구용 복합정제
EP3437636A1 (fr) * 2017-08-02 2019-02-06 Adamed sp. z o.o. Composition pharmaceutique comprenant de l'ézétimibe
KR102500643B1 (ko) * 2019-04-18 2023-02-16 한미약품 주식회사 에제티미브 및 로사르탄을 포함하는 약제학적 복합제제
KR20200137243A (ko) 2019-05-29 2020-12-09 콜마파마(주) 로수바스타틴 및 에제티미브를 포함하는 복합제의 제조방법
WO2021019499A1 (fr) 2019-07-31 2021-02-04 TECNIMEDE - Sociedade Técnico-medicinal, SA Compositions solides orales à libération immédiate à unités multiples, procédés et utilisations de celles-ci
MX2023002403A (es) * 2020-08-25 2023-03-22 Daewoong Pharmaceutical Co Ltd Composicion farmaceutica en forma de dosificacion individual para tratar o prevenir hipertension e hipercolesterolemia.
KR20250096941A (ko) 2023-12-20 2025-06-30 안국약품 주식회사 피타바스타틴 및 에제티미브를 포함하는 단일 정제 형태의 약학 조성물 및 이의 제조방법

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100907144B1 (ko) * 2007-09-05 2009-07-09 박재섭 이동부재를 이용한 골프 클럽
WO2009024889A2 (fr) * 2007-08-21 2009-02-26 Ranbaxy Laboratories Limited Composition pharmaceutique comprenant un inhibiteur de réductase hmg-coa et un ézétimibe
WO2011019326A2 (fr) * 2009-07-02 2011-02-17 Mahmut Bilgic Formulation pharmaceutique permettant d'augmenter la solubilité et la stabilité
WO2011012912A2 (fr) * 2009-07-28 2011-02-03 Egis Gyógyszergyár Nyilvánosan Működő Részvénytársaság Nouveau procédé de granulation et granulé ainsi préparé
EP2468258A1 (fr) * 2010-12-22 2012-06-27 LEK Pharmaceuticals d.d. Procédé de préparation d'une composition pharmaceutique comportant un ingrédient actif pharmaceutiquement faiblement soluble
WO2013166117A1 (fr) * 2012-05-01 2013-11-07 Althera Life Sciences, Llc Formulation de comprimé oral constituée d'une combinaison fixe de rosuvastatine et d'ézétimibe pour le traitement de l'hyperlipidémie et de maladies cardiovasculaires

Also Published As

Publication number Publication date
TWI700100B (zh) 2020-08-01
WO2015199356A1 (fr) 2015-12-30
TW201625223A (zh) 2016-07-16
JOP20150154B1 (ar) 2021-08-17
KR101977785B1 (ko) 2019-05-14
SG11201610748RA (en) 2017-01-27
AR100977A1 (es) 2016-11-16
KR20160000762A (ko) 2016-01-05
ECSP16096477A (es) 2017-01-31
SG10201811586YA (en) 2019-02-27
BR112016030111A2 (pt) 2017-08-22
UY36190A (es) 2015-10-30

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