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CL2016001216A1 - Acrilamidas de pirrolo[2,3-d]pirimidinilo, pirrolo[2,3-b]pirazinilo y pirrolo[2,3-d]piridinilo. - Google Patents

Acrilamidas de pirrolo[2,3-d]pirimidinilo, pirrolo[2,3-b]pirazinilo y pirrolo[2,3-d]piridinilo.

Info

Publication number
CL2016001216A1
CL2016001216A1 CL2016001216A CL2016001216A CL2016001216A1 CL 2016001216 A1 CL2016001216 A1 CL 2016001216A1 CL 2016001216 A CL2016001216 A CL 2016001216A CL 2016001216 A CL2016001216 A CL 2016001216A CL 2016001216 A1 CL2016001216 A1 CL 2016001216A1
Authority
CL
Chile
Prior art keywords
pyrrolo
pyrazinyl
pyrimidinyl
pirrolo
acrylamides
Prior art date
Application number
CL2016001216A
Other languages
English (en)
Inventor
Ye Che
Justin Ian Montgomery
Matthew Merrill Hayward
Matthew Frank Brown
Agustin Casimiro-Garcia
Jothan Wadsworth Coe
Mark Edward Flanagan
Adam Matthew Gilbert
Jean Baptiste Telliez
Atli Thorarensen
Rayomand Jal Unwalla
John I Trujillo
Jonathan David Langille
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=52144776&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2016001216(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer filed Critical Pfizer
Publication of CL2016001216A1 publication Critical patent/CL2016001216A1/es

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    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/4375—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having nitrogen as a ring heteroatom, e.g. quinolizines, naphthyridines, berberine, vincamine
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Abstract

<p>ACRILAMIDAS DE PIRROLO[2,3-D]PIRIMIDINILO, PIRROLO[2,3-B]PIRAZINILO Y PIRROLO[2.3-D]PIRIDINILO; COMPOSICIÓN FARMACÉUTICA O VETERINARIA Y USO EN EL TRATAMIENTO DE ENFERMEDADES TALES COMO ARTRITIS REUMATOIDE, MIOSITIS, CROHN, ALZHEIMER, CANCER, ENTRE OTRAS.</p>
CL2016001216A 2013-12-05 2016-05-20 Acrilamidas de pirrolo[2,3-d]pirimidinilo, pirrolo[2,3-b]pirazinilo y pirrolo[2,3-d]piridinilo. CL2016001216A1 (es)

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