CL2008000474A1 - Compuestos derivados de azonia-biciclo-[2.2.2]octano, moduladores del receptor m3; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como epoc, asma, sindrome del intestino irritable, entre otras. - Google Patents
Compuestos derivados de azonia-biciclo-[2.2.2]octano, moduladores del receptor m3; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como epoc, asma, sindrome del intestino irritable, entre otras.Info
- Publication number
- CL2008000474A1 CL2008000474A1 CL200800474A CL2008000474A CL2008000474A1 CL 2008000474 A1 CL2008000474 A1 CL 2008000474A1 CL 200800474 A CL200800474 A CL 200800474A CL 2008000474 A CL2008000474 A CL 2008000474A CL 2008000474 A1 CL2008000474 A1 CL 2008000474A1
- Authority
- CL
- Chile
- Prior art keywords
- biciclo
- octano
- azonia
- copd
- asthma
- Prior art date
Links
- 208000006673 asthma Diseases 0.000 title 1
- 150000001875 compounds Chemical class 0.000 title 1
- 201000010099 disease Diseases 0.000 title 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 title 1
- 210000000936 intestine Anatomy 0.000 title 1
- TVMXDCGIABBOFY-UHFFFAOYSA-N octane Chemical compound CCCCCCCC TVMXDCGIABBOFY-UHFFFAOYSA-N 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 208000011580 syndromic disease Diseases 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/04—Drugs for disorders of the respiratory system for throat disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pulmonology (AREA)
- Urology & Nephrology (AREA)
- Otolaryngology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Medicinal Preparation (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0702994A GB0702994D0 (en) | 2007-02-15 | 2007-02-15 | Compound and thier use |
| GB0722678A GB0722678D0 (en) | 2007-11-19 | 2007-11-19 | Compounds and their use II |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CL2008000474A1 true CL2008000474A1 (es) | 2008-08-22 |
Family
ID=39323641
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CL200800474A CL2008000474A1 (es) | 2007-02-15 | 2008-02-14 | Compuestos derivados de azonia-biciclo-[2.2.2]octano, moduladores del receptor m3; composicion farmaceutica; y uso en el tratamiento de enfermedades tales como epoc, asma, sindrome del intestino irritable, entre otras. |
Country Status (21)
| Country | Link |
|---|---|
| US (1) | US20100056565A1 (es) |
| EP (1) | EP2121688A1 (es) |
| JP (1) | JP2010519193A (es) |
| KR (1) | KR20090110353A (es) |
| CN (1) | CN101657452A (es) |
| AR (1) | AR065344A1 (es) |
| AU (1) | AU2008215924B2 (es) |
| BR (1) | BRPI0807913A2 (es) |
| CA (1) | CA2676581A1 (es) |
| CL (1) | CL2008000474A1 (es) |
| CO (1) | CO6190612A2 (es) |
| EC (1) | ECSP099573A (es) |
| IL (1) | IL199971A0 (es) |
| MX (1) | MX2009008323A (es) |
| NZ (1) | NZ578489A (es) |
| PE (1) | PE20090357A1 (es) |
| RU (1) | RU2009133258A (es) |
| SA (1) | SA08290066B1 (es) |
| TW (1) | TW200843759A (es) |
| UY (1) | UY30916A1 (es) |
| WO (1) | WO2008099186A1 (es) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TW200825084A (en) | 2006-11-14 | 2008-06-16 | Astrazeneca Ab | New compounds 521 |
| WO2009098453A1 (en) * | 2008-02-06 | 2009-08-13 | Astrazeneca Ab | Azonia bicycloalkanes as m3 muscarinic acetylcholin receptor antagonists |
| WO2009138707A1 (en) | 2008-05-13 | 2009-11-19 | Astrazeneca Ab | Quinuclidine derivatives as muscarinic m3 receptor antagonists |
| GB0814728D0 (en) * | 2008-08-12 | 2008-09-17 | Argenta Discovery Ltd | New combination |
| WO2010018352A1 (en) * | 2008-08-12 | 2010-02-18 | Argenta Discovery Limited | Heterocyclic compounds used in the treatment of diseases where enhanced m3 receptor activation is implicated |
| WO2010019099A1 (en) * | 2008-08-12 | 2010-02-18 | Astrazeneca Ab | 2-hydroxy-ethanesulfonate salt |
| GB0814729D0 (en) * | 2008-08-12 | 2008-09-17 | Argenta Discovery Ltd | New combination |
| TW201036957A (en) | 2009-02-20 | 2010-10-16 | Astrazeneca Ab | Novel salt 628 |
| CN104418851A (zh) * | 2013-09-02 | 2015-03-18 | 上海龙翔生物医药开发有限公司 | 奎宁环衍生物的制备方法及纯化方法 |
| CN106573928B (zh) * | 2014-08-26 | 2020-04-14 | 安斯泰来制药株式会社 | 2-氨基噻唑衍生物或其盐 |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8334494D0 (en) * | 1983-12-24 | 1984-02-01 | Tanabe Seiyaku Co | Carbostyril derivatives |
| NZ225999A (en) * | 1987-09-10 | 1992-04-28 | Merck Sharp & Dohme | Azacyclic- or azabicyclic-substituted thiadiazole derivatives and pharmaceutical compositions |
| IL88846A0 (en) * | 1988-01-08 | 1989-07-31 | Merck Sharp & Dohme | Lipophilic oxadiazoles,their preparation and pharmaceutical compositions containing them |
| GB9603755D0 (en) * | 1996-02-22 | 1996-04-24 | Pfizer Ltd | Therapeutic agents |
| DE19856475A1 (de) * | 1998-11-27 | 2000-05-31 | Schering Ag | Nichtsteroidale Entzündungshemmer |
| US20020052312A1 (en) * | 2000-05-30 | 2002-05-02 | Reiss Theodore F. | Combination therapy of chronic obstructive pulmonary disease using muscarinic receptor antagonists |
| UA75626C2 (en) * | 2000-12-28 | 2006-05-15 | Almirall Prodesfarma Ag | Quinuclidine derivatives and medicinal compositions containing the same |
| DE60326894D1 (de) * | 2002-09-30 | 2009-05-07 | Neurosearch As | 1,4-Diazabicycloalkanderivate, deren Herstellung und Verwendung |
| BR0314183A (pt) * | 2002-09-30 | 2005-08-09 | Neurosearch As | Derivados de 1,4-diazabicicloalcano, quaisquer de seus enanciÈmeros ou qualquer mistura de seus enaciÈmeros, ou um seu sal de adição farmaceuticamente aceitável ou um seu n-óxido, composição farmacêutica, uso do dito composto, de qualquer um de seus enanciÈmeros ou de qualquer mistura de seus enanciÈmeros, ou de um seu sal de adição farmaceuticamente aceitável, e, método de tratamento, prevenção ou alìvio de uma doença ou um distúrbio ou condição de um corpo animal vivo |
| US7056916B2 (en) * | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| ES2239546B1 (es) * | 2004-03-15 | 2006-12-01 | Almirall Prodesfarma, S.A. | Nuevos esteres de quinuclidina cuaternizados. |
| GB0516313D0 (en) * | 2005-08-08 | 2005-09-14 | Argenta Discovery Ltd | Azole derivatives and their uses |
-
2008
- 2008-02-14 CN CN200880012083A patent/CN101657452A/zh active Pending
- 2008-02-14 AR ARP080100627A patent/AR065344A1/es unknown
- 2008-02-14 CA CA002676581A patent/CA2676581A1/en not_active Abandoned
- 2008-02-14 MX MX2009008323A patent/MX2009008323A/es active IP Right Grant
- 2008-02-14 BR BRPI0807913-7A2A patent/BRPI0807913A2/pt not_active IP Right Cessation
- 2008-02-14 CL CL200800474A patent/CL2008000474A1/es unknown
- 2008-02-14 WO PCT/GB2008/000519 patent/WO2008099186A1/en not_active Ceased
- 2008-02-14 TW TW097105181A patent/TW200843759A/zh unknown
- 2008-02-14 RU RU2009133258/04A patent/RU2009133258A/ru not_active Application Discontinuation
- 2008-02-14 JP JP2009549470A patent/JP2010519193A/ja active Pending
- 2008-02-14 NZ NZ578489A patent/NZ578489A/en not_active IP Right Cessation
- 2008-02-14 EP EP08709410A patent/EP2121688A1/en not_active Withdrawn
- 2008-02-14 US US12/523,609 patent/US20100056565A1/en not_active Abandoned
- 2008-02-14 AU AU2008215924A patent/AU2008215924B2/en not_active Ceased
- 2008-02-14 PE PE2008000323A patent/PE20090357A1/es not_active Application Discontinuation
- 2008-02-14 KR KR1020097017018A patent/KR20090110353A/ko not_active Withdrawn
- 2008-02-14 UY UY30916A patent/UY30916A1/es not_active Application Discontinuation
- 2008-02-16 SA SA08290066A patent/SA08290066B1/ar unknown
-
2009
- 2009-07-20 IL IL199971A patent/IL199971A0/en unknown
- 2009-07-28 CO CO09078490A patent/CO6190612A2/es not_active Application Discontinuation
- 2009-08-12 EC EC2009009573A patent/ECSP099573A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| IL199971A0 (en) | 2010-04-15 |
| JP2010519193A (ja) | 2010-06-03 |
| WO2008099186A8 (en) | 2008-11-13 |
| SA08290066B1 (ar) | 2011-05-14 |
| EP2121688A1 (en) | 2009-11-25 |
| BRPI0807913A2 (pt) | 2014-06-17 |
| RU2009133258A (ru) | 2011-03-20 |
| KR20090110353A (ko) | 2009-10-21 |
| AR065344A1 (es) | 2009-06-03 |
| NZ578489A (en) | 2011-05-27 |
| MX2009008323A (es) | 2009-08-13 |
| ECSP099573A (es) | 2009-12-28 |
| CN101657452A (zh) | 2010-02-24 |
| US20100056565A1 (en) | 2010-03-04 |
| CA2676581A1 (en) | 2008-08-21 |
| WO2008099186A1 (en) | 2008-08-21 |
| CO6190612A2 (es) | 2010-08-19 |
| UY30916A1 (es) | 2008-09-30 |
| PE20090357A1 (es) | 2009-04-01 |
| AU2008215924B2 (en) | 2011-04-21 |
| TW200843759A (en) | 2008-11-16 |
| AU2008215924A1 (en) | 2008-08-21 |
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