CH423799A - Verfahren zur Herstellung von 3,8-Diazabicyclo-(3,2,1)-oktanen - Google Patents
Verfahren zur Herstellung von 3,8-Diazabicyclo-(3,2,1)-oktanenInfo
- Publication number
- CH423799A CH423799A CH727862A CH727862A CH423799A CH 423799 A CH423799 A CH 423799A CH 727862 A CH727862 A CH 727862A CH 727862 A CH727862 A CH 727862A CH 423799 A CH423799 A CH 423799A
- Authority
- CH
- Switzerland
- Prior art keywords
- octanes
- diazabicyclo
- preparation
- Prior art date
Links
- LKDJYZBKCVSODK-UHFFFAOYSA-N 3,8-diazabicyclo[3.2.1]octane Chemical class C1NCC2CCC1N2 LKDJYZBKCVSODK-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/08—Bridged systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/5545—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having eight-membered rings not containing additional condensed or non-condensed nitrogen-containing 3-7 membered rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB23076/61A GB949088A (en) | 1961-06-26 | 1961-06-26 | Diazabicyclo-octane derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH423799A true CH423799A (de) | 1966-11-15 |
Family
ID=10189738
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH727862A CH423799A (de) | 1961-06-26 | 1962-06-18 | Verfahren zur Herstellung von 3,8-Diazabicyclo-(3,2,1)-oktanen |
Country Status (6)
| Country | Link |
|---|---|
| BE (1) | BE618813A (de) |
| BR (1) | BR6240334D0 (de) |
| CH (1) | CH423799A (de) |
| DK (1) | DK105414C (de) |
| FI (1) | FI40096C (de) |
| GB (1) | GB949088A (de) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1274018B (it) * | 1994-02-23 | 1997-07-14 | Riace Ets | Derivati del 3,8-diazabiciclo(3.2.1.)ottano ad attivita' analgesica |
| SE0003795D0 (sv) | 2000-10-20 | 2000-10-20 | Astrazeneca Ab | Pharmaceutically useful compounds |
| AU2005311311A1 (en) | 2004-11-30 | 2006-06-08 | Neurosearch A/S | Novel diazabicyclic aryl derivatives as cholinergy ligands |
| US8673920B2 (en) * | 2009-05-06 | 2014-03-18 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| WO2012058116A1 (en) | 2010-10-27 | 2012-05-03 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| WO2012058134A1 (en) | 2010-10-29 | 2012-05-03 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| JP2014521751A (ja) | 2011-08-19 | 2014-08-28 | メルク・シャープ・アンド・ドーム・コーポレーション | 腎髄質外層カリウムチャンネルの阻害薬 |
| US9527830B2 (en) | 2011-09-16 | 2016-12-27 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| US8999990B2 (en) | 2011-10-25 | 2015-04-07 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| WO2013062900A1 (en) | 2011-10-25 | 2013-05-02 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| US9108947B2 (en) | 2011-10-31 | 2015-08-18 | Merck Sharp & Dohme Corp. | Inhibitors of the Renal Outer Medullary Potassium channel |
| WO2013066718A2 (en) | 2011-10-31 | 2013-05-10 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| US9139585B2 (en) | 2011-10-31 | 2015-09-22 | Merck Sharp & Dohme Corp. | Inhibitors of the Renal Outer Medullary Potassium channel |
| EP2790511B1 (de) | 2011-12-16 | 2016-09-14 | Merck Sharp & Dohme Corp. | Inhibitoren des renalen kaliumkanals der äusseren medulla |
| AR092031A1 (es) | 2012-07-26 | 2015-03-18 | Merck Sharp & Dohme | Inhibidores del canal de potasio medular externo renal |
| WO2014085210A1 (en) | 2012-11-29 | 2014-06-05 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| EP2934533B1 (de) | 2012-12-19 | 2017-11-15 | Merck Sharp & Dohme Corp. | Inhibitoren des kaliumkanals des äusseren nierenmarks |
| WO2014126944A2 (en) | 2013-02-18 | 2014-08-21 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| US9765074B2 (en) | 2013-03-15 | 2017-09-19 | Merck Sharp & Dohme Corp. | Inhibitors of the renal outer medullary potassium channel |
| EP3027625B1 (de) | 2013-07-31 | 2018-05-30 | Merck Sharp & Dohme Corp. | Zur behandlung von unter anderem bluthochdruck und akuter oder chronischer herzinsuffizienz geeignete spirokondensierte derivate von piperidin |
| WO2016127358A1 (en) | 2015-02-12 | 2016-08-18 | Merck Sharp & Dohme Corp. | Inhibitors of renal outer medullary potassium channel |
-
1961
- 1961-06-26 GB GB23076/61A patent/GB949088A/en not_active Expired
-
1962
- 1962-06-12 BE BE618813A patent/BE618813A/fr unknown
- 1962-06-18 CH CH727862A patent/CH423799A/de unknown
- 1962-06-25 FI FI122162A patent/FI40096C/fi active
- 1962-06-25 DK DK282462AA patent/DK105414C/da active
- 1962-06-25 BR BR140334/62A patent/BR6240334D0/pt unknown
Also Published As
| Publication number | Publication date |
|---|---|
| BE618813A (fr) | 1962-10-01 |
| DK105414C (da) | 1966-09-26 |
| GB949088A (en) | 1964-02-12 |
| FI40096B (de) | 1968-06-28 |
| BR6240334D0 (pt) | 1973-05-24 |
| FI40096C (fi) | 1968-10-10 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CH412918A (de) | Verfahren zur Herstellung von 1,8-Naphthyridinen | |
| CH423799A (de) | Verfahren zur Herstellung von 3,8-Diazabicyclo-(3,2,1)-oktanen | |
| CH457473A (de) | Verfahren zur Herstellung von 9,10-Dihydroergovalin | |
| CH448128A (de) | Verfahren zur Herstellung von 2,3-Epithio-steroiden | |
| AT255031B (de) | Verfahren zur Herstellung von 1-Glykosyl-6-azauracilen | |
| CH403735A (de) | Verfahren zur Herstellung von 3-Brom-3-chlor-1,1,2,2-tetrafluor-propan | |
| CH405326A (de) | Verfahren zur Herstellung von 1,3-Diaryl-pyrazolinen | |
| CH398622A (de) | Verfahren zur Herstellung von 2,4-Bis-amino-6-trichlormethyl-s-triazinen | |
| CH416638A (de) | Verfahren zur Herstellung von Spirobiphenylphenazametalloverbindungen | |
| CH433236A (de) | Verfahren zur Herstellung von 2,6-Dichlorbenzonitril | |
| CH415664A (de) | Verfahren zur Herstellung von substituierten 1-Halogenphenyl-2-amino-alkanonen-(1) | |
| AT239438B (de) | Verfahren zur Herstellung von α-Aminobenzylpenicillin | |
| AT241687B (de) | Verfahren zur Herstellung von α-Aminobenzylpenicillin | |
| CH404678A (de) | Verfahren zur Herstellung von neuen 3,8-Diazabicyclo-(3,2,1)-octanen | |
| CH424758A (de) | Verfahren zur Herstellung von 2,6-Dichlorbenzaldoxim | |
| CH442323A (de) | Verfahren zur Herstellung von O,S-Dialkoxycarbonylthiaminen | |
| CH442352A (de) | Verfahren zur Herstellung von 2-Alkoxy-3,4-dihydroxy-5-hydroxymethyl-tetrahydrofuranderivaten | |
| CH397715A (de) | Verfahren zur Herstellung von 2,5-Diarylaminoterephthalsäuren | |
| CH432487A (de) | Verfahren zur Herstellung von Mononitro-1,3,5-trialkylbenzol | |
| CH435260A (de) | Verfahren zur Herstellung von 19-Hydroxy-4,5-dehydro-3-oxo-steroiden | |
| CH409933A (de) | Verfahren zur Herstellung von O,O-Dimethyldithiophosphoryl-essigsäure-monomethylamid | |
| CH408934A (de) | Verfahren zur Herstellung von 1,4,5-trisubstituierten Pyridazonen-(6) | |
| CH396021A (de) | Verfahren zur Herstellung von Derivaten des 2-Methylothio-4,6-bis-amino-s-triazins | |
| CH407086A (de) | Verfahren zur Herstellung von 1,2,3,4-Tetraalkyl-anthrachinon-8-carbonsäuren | |
| CH415675A (de) | Verfahren zur Herstellung von 4-Methyl-6-isobutenyl-pyron-(2) |