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CA3019145C - Composes de pyrrolotriazine en tant qu'inhibiteurs de tam - Google Patents

Composes de pyrrolotriazine en tant qu'inhibiteurs de tam

Info

Publication number
CA3019145C
CA3019145C CA3019145A CA3019145A CA3019145C CA 3019145 C CA3019145 C CA 3019145C CA 3019145 A CA3019145 A CA 3019145A CA 3019145 A CA3019145 A CA 3019145A CA 3019145 C CA3019145 C CA 3019145C
Authority
CA
Canada
Prior art keywords
phenyl
amino
triazin
carboxamide
pyrrolo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Active
Application number
CA3019145A
Other languages
English (en)
Other versions
CA3019145A1 (fr
Inventor
Yun-Long Li
Xiaozhao Wang
Joseph Barbosa
David M. Burns
Hao Feng
Joseph Glenn
Chunhong He
Taisheng Huang
Song Mei
Jincong Zhuo
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Incyte Corp filed Critical Incyte Corp
Priority claimed from PCT/US2017/024270 external-priority patent/WO2017172596A1/fr
Publication of CA3019145A1 publication Critical patent/CA3019145A1/fr
Application granted granted Critical
Publication of CA3019145C publication Critical patent/CA3019145C/fr
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

Abstract

Cette application décrit des composés de Formule I : et des sels acceptables sur le plan pharmaceutique, qui sont des inhibiteurs de kinases TAM et peuvent ainsi être utiles dans le traitement de maladies comme le cancer. Dans certaines réalisations, il est décrit des composés de Formule (IIb1) ou (IIb2) : et des sels acceptables sur le plan pharmaceutique.
CA3019145A 2016-03-28 2017-03-27 Composes de pyrrolotriazine en tant qu'inhibiteurs de tam Active CA3019145C (fr)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201662314066P 2016-03-28 2016-03-28
US62/314,066 2016-03-28
US201662362934P 2016-07-15 2016-07-15
US62/362,934 2016-07-15
US201662438750P 2016-12-23 2016-12-23
US62/438,750 2016-12-23
PCT/US2017/024270 WO2017172596A1 (fr) 2016-03-28 2017-03-27 Composés de pyrrolotriazine en tant qu'inhibiteurs de tam

Publications (2)

Publication Number Publication Date
CA3019145A1 CA3019145A1 (fr) 2017-10-05
CA3019145C true CA3019145C (fr) 2025-11-18

Family

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