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CA1094061A - 5(6)-benzene ring substituted benzimidazole-2- carbamate derivatives having anthelmintic activity - Google Patents

5(6)-benzene ring substituted benzimidazole-2- carbamate derivatives having anthelmintic activity

Info

Publication number
CA1094061A
CA1094061A CA273,928A CA273928A CA1094061A CA 1094061 A CA1094061 A CA 1094061A CA 273928 A CA273928 A CA 273928A CA 1094061 A CA1094061 A CA 1094061A
Authority
CA
Canada
Prior art keywords
compound
prepared
process according
steps
heterocyclic ring
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA273,928A
Other languages
English (en)
French (fr)
Inventor
Colin C. Beard
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Syntex USA LLC
Original Assignee
Syntex USA LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US05/758,112 external-priority patent/US4139626A/en
Application filed by Syntex USA LLC filed Critical Syntex USA LLC
Application granted granted Critical
Publication of CA1094061A publication Critical patent/CA1094061A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
    • C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
    • C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
    • C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • C07D235/30—Nitrogen atoms not forming part of a nitro radical
    • C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C335/00—Thioureas, i.e. compounds containing any of the groups, the nitrogen atoms not being part of nitro or nitroso groups
    • C07C335/30—Isothioureas
    • C07C335/38—Isothioureas containing any of the groups, X being a hetero atom, Y being any atom

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CA273,928A 1976-03-19 1977-03-14 5(6)-benzene ring substituted benzimidazole-2- carbamate derivatives having anthelmintic activity Expired CA1094061A (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US66877876A 1976-03-19 1976-03-19
US05/758,112 US4139626A (en) 1976-03-19 1977-01-10 Anthelmintic 5(6)-benzene ring substituted benzimidazole-2-carbamates
US758,112 1977-01-10
US668,778 1991-03-13

Publications (1)

Publication Number Publication Date
CA1094061A true CA1094061A (en) 1981-01-20

Family

ID=27099988

Family Applications (1)

Application Number Title Priority Date Filing Date
CA273,928A Expired CA1094061A (en) 1976-03-19 1977-03-14 5(6)-benzene ring substituted benzimidazole-2- carbamate derivatives having anthelmintic activity

Country Status (14)

Country Link
AR (1) AR219071A1 (es)
AU (1) AU509378B2 (es)
CA (1) CA1094061A (es)
DE (1) DE2711945A1 (es)
ES (2) ES456912A1 (es)
FR (1) FR2344543A1 (es)
GB (1) GB1542203A (es)
IE (1) IE44789B1 (es)
IL (1) IL51659A0 (es)
NL (1) NL7702820A (es)
NZ (1) NZ183615A (es)
PH (1) PH14078A (es)
PL (1) PL107159B1 (es)
SE (1) SE7702986L (es)

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6825219B2 (en) 2001-11-09 2004-11-30 Boehringer Ingelheim Pharmaceuticals, Inc. Substituted benzimidazole compounds
US7138420B2 (en) 2002-08-08 2006-11-21 Boehringer Ingelheim Pharmaceuticals Inc. Substituted benzimidazole compounds

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4297365A (en) 1978-08-04 1981-10-27 Ciba-Geigy Corporation Benzimidazoles and pharmaceutical preparations containing such compounds
DE2845537A1 (de) * 1978-10-19 1980-04-30 Bayer Ag Benzimidazolylcarbamidsaeureester, verfahren zu ihrer herstellung sowie ihre verwendung als arzneimittel

Cited By (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6825219B2 (en) 2001-11-09 2004-11-30 Boehringer Ingelheim Pharmaceuticals, Inc. Substituted benzimidazole compounds
US7138420B2 (en) 2002-08-08 2006-11-21 Boehringer Ingelheim Pharmaceuticals Inc. Substituted benzimidazole compounds

Also Published As

Publication number Publication date
IE44789B1 (en) 1982-04-07
IE44789L (en) 1977-09-19
PL196734A1 (pl) 1978-01-16
AU509378B2 (en) 1980-05-08
PH14078A (en) 1981-01-30
ES467267A1 (es) 1979-10-16
FR2344543A1 (fr) 1977-10-14
ES456912A1 (es) 1978-07-16
AU2333477A (en) 1978-09-21
DE2711945A1 (de) 1977-09-29
AR219071A1 (es) 1980-07-31
PL107159B1 (pl) 1980-01-31
NZ183615A (en) 1979-10-25
FR2344543B1 (es) 1981-01-09
SE7702986L (sv) 1977-09-20
IL51659A0 (en) 1977-05-31
NL7702820A (nl) 1977-09-21
GB1542203A (en) 1979-03-14

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Legal Events

Date Code Title Description
MKEX Expiry