BRPI1012859A2 - composto, composição, uso de um compostos, e, método para tratar um mamífero - Google Patents
composto, composição, uso de um compostos, e, método para tratar um mamíferoInfo
- Publication number
- BRPI1012859A2 BRPI1012859A2 BRPI1012859A BRPI1012859A BRPI1012859A2 BR PI1012859 A2 BRPI1012859 A2 BR PI1012859A2 BR PI1012859 A BRPI1012859 A BR PI1012859A BR PI1012859 A BRPI1012859 A BR PI1012859A BR PI1012859 A2 BRPI1012859 A2 BR PI1012859A2
- Authority
- BR
- Brazil
- Prior art keywords
- compound
- mammal
- treating
- composition
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 2
- 241000124008 Mammalia Species 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/472—Non-condensed isoquinolines, e.g. papaverine
- A61K31/4725—Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/10—Antioedematous agents; Diuretics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Urology & Nephrology (AREA)
- Biomedical Technology (AREA)
- Endocrinology (AREA)
- Vascular Medicine (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Obesity (AREA)
- Rheumatology (AREA)
- Ophthalmology & Optometry (AREA)
- Emergency Medicine (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP09160829 | 2009-05-20 | ||
| PCT/EP2010/056968 WO2010133669A1 (en) | 2009-05-20 | 2010-05-20 | Substituted quinolines for use as vegf inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI1012859A2 true BRPI1012859A2 (pt) | 2016-04-05 |
Family
ID=41152142
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI1012859A BRPI1012859A2 (pt) | 2009-05-20 | 2010-05-20 | composto, composição, uso de um compostos, e, método para tratar um mamífero |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US20120065199A1 (pt) |
| EP (1) | EP2432764A1 (pt) |
| JP (1) | JP2012527431A (pt) |
| KR (1) | KR20120023807A (pt) |
| CN (1) | CN102625798A (pt) |
| AU (1) | AU2010251134A1 (pt) |
| BR (1) | BRPI1012859A2 (pt) |
| CA (1) | CA2762232A1 (pt) |
| EA (1) | EA201101658A1 (pt) |
| IL (1) | IL216408A0 (pt) |
| MX (1) | MX2011012340A (pt) |
| SG (1) | SG176167A1 (pt) |
| WO (1) | WO2010133669A1 (pt) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2013103317A1 (en) * | 2012-01-05 | 2013-07-11 | Clanotech Ab | Quinoline compounds which are anti-angiogenic integrin alpha5 betal inhibitors for use in the treatment of fibrosis or fibrosis-related diseases |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SE0400284D0 (sv) * | 2004-02-10 | 2004-02-10 | Astrazeneca Ab | Novel compounds |
| WO2008119771A2 (en) | 2007-03-30 | 2008-10-09 | Clanotech Ab | Quinoline-s-carboxylic acid derivatives as tyrosine kinase inhibitors |
-
2010
- 2010-05-20 MX MX2011012340A patent/MX2011012340A/es not_active Application Discontinuation
- 2010-05-20 CA CA2762232A patent/CA2762232A1/en not_active Abandoned
- 2010-05-20 AU AU2010251134A patent/AU2010251134A1/en not_active Abandoned
- 2010-05-20 WO PCT/EP2010/056968 patent/WO2010133669A1/en not_active Ceased
- 2010-05-20 US US13/321,602 patent/US20120065199A1/en not_active Abandoned
- 2010-05-20 EA EA201101658A patent/EA201101658A1/ru unknown
- 2010-05-20 JP JP2012511290A patent/JP2012527431A/ja not_active Withdrawn
- 2010-05-20 SG SG2011085461A patent/SG176167A1/en unknown
- 2010-05-20 KR KR1020117030328A patent/KR20120023807A/ko not_active Withdrawn
- 2010-05-20 CN CN201080033815XA patent/CN102625798A/zh active Pending
- 2010-05-20 BR BRPI1012859A patent/BRPI1012859A2/pt not_active IP Right Cessation
- 2010-05-20 EP EP10723066A patent/EP2432764A1/en not_active Withdrawn
-
2011
- 2011-11-17 IL IL216408A patent/IL216408A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2432764A1 (en) | 2012-03-28 |
| US20120065199A1 (en) | 2012-03-15 |
| SG176167A1 (en) | 2011-12-29 |
| KR20120023807A (ko) | 2012-03-13 |
| JP2012527431A (ja) | 2012-11-08 |
| EA201101658A1 (ru) | 2012-05-30 |
| MX2011012340A (es) | 2011-12-14 |
| CA2762232A1 (en) | 2010-11-25 |
| WO2010133669A1 (en) | 2010-11-25 |
| AU2010251134A1 (en) | 2011-12-08 |
| IL216408A0 (en) | 2012-02-29 |
| CN102625798A (zh) | 2012-08-01 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 5A E 6A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |