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BRPI1010546B8 - processo para produzir composto, método para isolar e purificar cristais de solvato do composto, e, uso do composto - Google Patents

processo para produzir composto, método para isolar e purificar cristais de solvato do composto, e, uso do composto

Info

Publication number
BRPI1010546B8
BRPI1010546B8 BRPI1010546A BRPI1010546A BRPI1010546B8 BR PI1010546 B8 BRPI1010546 B8 BR PI1010546B8 BR PI1010546 A BRPI1010546 A BR PI1010546A BR PI1010546 A BRPI1010546 A BR PI1010546A BR PI1010546 B8 BRPI1010546 B8 BR PI1010546B8
Authority
BR
Brazil
Prior art keywords
compound
isolating
producing
solvate crystals
purifying
Prior art date
Application number
BRPI1010546A
Other languages
English (en)
Inventor
Fukuda Yoshimasa
Ando Takashi
Goto Kimihiko
Nakanishi Nozomu
Watanabe Takashi
Kurihara Kenichi
Minowa Nobuto
Mitomi Masaaki
Original Assignee
Meiji Seika Pharma Co Ltd
Mmag Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Meiji Seika Pharma Co Ltd, Mmag Co Ltd filed Critical Meiji Seika Pharma Co Ltd
Publication of BRPI1010546A2 publication Critical patent/BRPI1010546A2/pt
Publication of BRPI1010546B1 publication Critical patent/BRPI1010546B1/pt
Publication of BRPI1010546B8 publication Critical patent/BRPI1010546B8/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/04—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/04—Ortho-condensed systems
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)

Abstract

PROCESSO PARA PRODUZIR COMPOSTO, MÉTODO PARA ISOLAR E PURIFICAR CRISTAIS DE SOLVATO DO COMPOSTO, E, USO DO COMPOSTO. Um processo para produzir eficientemente um derivado de piripiropeno tendo grupos acilóxi nas posições 1 e 11 e um grupo hidróxi na posição 7. O processo compreende uma etapa na qual os grupos hidróxi nas posições 1 e 11 do composto representado pela fórmula (B1) são seletivamente acilados com um agente de acilação na presença ou ausência de uma base em um a três estágios.
BRPI1010546A 2009-05-13 2010-05-12 processo para produzir composto, método para isolar e purificar cristais de solvato do composto, e, uso do composto BRPI1010546B8 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2009116305 2009-05-13
JP2010044416 2010-03-01
PCT/JP2010/058040 WO2010131676A1 (ja) 2009-05-13 2010-05-12 ピリピロペン誘導体の製造法

Publications (3)

Publication Number Publication Date
BRPI1010546A2 BRPI1010546A2 (pt) 2015-08-25
BRPI1010546B1 BRPI1010546B1 (pt) 2017-04-11
BRPI1010546B8 true BRPI1010546B8 (pt) 2022-08-23

Family

ID=43085049

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI1010546A BRPI1010546B8 (pt) 2009-05-13 2010-05-12 processo para produzir composto, método para isolar e purificar cristais de solvato do composto, e, uso do composto

Country Status (21)

Country Link
US (1) US8853413B2 (pt)
EP (1) EP2426124B1 (pt)
JP (1) JP5781432B2 (pt)
KR (1) KR101589335B1 (pt)
CN (2) CN104370932A (pt)
AR (1) AR076867A1 (pt)
AU (1) AU2010248488B2 (pt)
BR (1) BRPI1010546B8 (pt)
CA (1) CA2760078C (pt)
CR (1) CR20110587A (pt)
DK (1) DK2426124T3 (pt)
EC (1) ECSP11011518A (pt)
ES (1) ES2433650T3 (pt)
IL (1) IL215904A (pt)
MX (1) MX2011011414A (pt)
NZ (1) NZ596159A (pt)
PL (1) PL2426124T3 (pt)
RU (1) RU2532441C2 (pt)
TW (1) TWI516492B (pt)
WO (1) WO2010131676A1 (pt)
ZA (1) ZA201107695B (pt)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN102144030B (zh) * 2008-07-24 2016-05-04 明治制果药业株式会社 啶南平a生物合成基因
CA2787829A1 (en) * 2010-01-26 2011-08-04 Meiji Seika Pharma Co., Ltd. Method for producing pyripyropene derivatives by the enzymatic method
UA111151C2 (uk) * 2010-03-01 2016-04-11 Мейдзі Сейка Фарма Ко., Лтд. Спосіб одержання похідних пірипіропену
AU2011303970B2 (en) * 2010-09-14 2015-08-13 Basf Se Composition containing a pyripyropene insecticide and an adjuvant
ES2566910T3 (es) 2012-03-12 2016-04-18 Basf Se Formulación de concentrado líquido que contiene un insecticida de piripiropeno II
CN104168769B (zh) * 2012-03-12 2016-12-14 巴斯夫欧洲公司 生产啶南平杀虫剂的含水悬浮液浓缩物配制剂的方法
AU2014206958B2 (en) * 2013-01-16 2017-08-10 Basf Se Method for preparing a pyripyropene compound
JP6465860B2 (ja) 2013-03-28 2019-02-06 ビーエーエスエフ ソシエタス・ヨーロピアＢａｓｆ Ｓｅ 乾燥バイオマスからのピリピロペンの生産

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP3233476B2 (ja) 1992-10-22 2001-11-26 社団法人北里研究所 Ｆｏ−１２８９物質およびその製造法
JPH08239385A (ja) 1995-03-03 1996-09-17 Kitasato Inst:The Ｆｏ−１２８９物質およびその製造法
JP3725198B2 (ja) * 1995-03-27 2005-12-07 社団法人北里研究所 ピリピロペン誘導体
JPH08269065A (ja) 1995-04-03 1996-10-15 Kitasato Inst:The ピリピロペン誘導体
KR100522446B1 (ko) 2003-01-07 2005-10-18 한국생명공학연구원 아실 코에이:콜레스테롤 아실 트란스퍼라제의 저해활성을갖는 화합물 또는 그 염을 유효성분으로 하는 살충제
DE602004021640D1 (de) * 2003-12-23 2009-07-30 Tibotec Pharm Ltd Verfahren zur herstellung von (1s,2r)-3-ää(4-aminophenyl)sulfonylü(isobutyl)aminoü-1-benzyl-2-hydroxypropylcarbamidsäure-(3r,3as,6ar)-hexahydrofuroä2,3-büfuran-3-ylester
TW200616623A (en) 2004-05-28 2006-06-01 Speedel Experimenta Ag Organic compounds
JP2006129714A (ja) 2004-11-02 2006-05-25 Koken:Kk カバノアナタケの細胞壁の破壊方法、破壊装置及びカバノアナタケの有効成分の抽出方法。
US7491738B2 (en) 2005-06-01 2009-02-17 Meiji Seika Kaisha, Ltd. Pest control agents
TWI388282B (zh) 2005-06-01 2013-03-11 Meiji Seika Pharma Co Ltd 害蟲控制劑
JP2008050997A (ja) 2006-08-24 2008-03-06 Matsushita Electric Ind Co Ltd 密閉型電動圧縮機
US8202890B2 (en) 2006-11-30 2012-06-19 Meiji Seika Pharma Co., Ltd. Pest control agent
JP4488033B2 (ja) 2007-02-06 2010-06-23 ソニー株式会社 偏光素子及び液晶プロジェクター
JP2009022702A (ja) 2007-07-18 2009-02-05 Katariki Shoji:Kk 口腔内保護手段を備えた舌圧排子
AU2008287799B2 (en) 2007-08-13 2013-10-31 Meiji Seika Pharma Co., Ltd. Method for producing pyripyropene derivative and production intermediate thereof
JP5206145B2 (ja) 2007-10-15 2013-06-12 株式会社リコー 廃トナー回収容器ユニットおよび画像形成装置
EP2223599A4 (en) 2007-12-21 2012-01-11 Meiji Seika Kaisha NEW SYSTEMIC PESTICIDE
UA111151C2 (uk) * 2010-03-01 2016-04-11 Мейдзі Сейка Фарма Ко., Лтд. Спосіб одержання похідних пірипіропену

Also Published As

Publication number Publication date
EP2426124B1 (en) 2013-08-07
CN104370932A (zh) 2015-02-25
ES2433650T3 (es) 2013-12-12
ECSP11011518A (es) 2012-06-29
DK2426124T3 (da) 2013-09-30
KR101589335B1 (ko) 2016-01-27
PL2426124T3 (pl) 2013-12-31
CA2760078C (en) 2016-01-19
RU2532441C2 (ru) 2014-11-10
ZA201107695B (en) 2013-03-27
US20120046470A1 (en) 2012-02-23
RU2011150505A (ru) 2013-06-20
AU2010248488B2 (en) 2016-01-07
JP5781432B2 (ja) 2015-09-24
MX2011011414A (es) 2011-12-06
CN102348706A (zh) 2012-02-08
TWI516492B (zh) 2016-01-11
CR20110587A (es) 2012-01-12
BRPI1010546A2 (pt) 2015-08-25
WO2010131676A1 (ja) 2010-11-18
EP2426124A1 (en) 2012-03-07
TW201105678A (en) 2011-02-16
WO2010131676A9 (ja) 2011-02-03
AR076867A1 (es) 2011-07-13
NZ596159A (en) 2014-03-28
IL215904A0 (en) 2012-01-31
BRPI1010546B1 (pt) 2017-04-11
US8853413B2 (en) 2014-10-07
KR20120111929A (ko) 2012-10-11
CN102348706B (zh) 2015-03-04
EP2426124A4 (en) 2012-03-07
CA2760078A1 (en) 2010-11-18
IL215904A (en) 2016-03-31
JPWO2010131676A1 (ja) 2012-11-01
AU2010248488A1 (en) 2011-11-17

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Legal Events

Date Code Title Description
B06F Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 12/05/2010, OBSERVADAS AS CONDICOES LEGAIS.

B16C Correction of notification of the grant [chapter 16.3 patent gazette]
B25A Requested transfer of rights approved
B25G Requested change of headquarter approved
B25A Requested transfer of rights approved
B25D Requested change of name of applicant approved