BRPI1005147A2 - processo de preparação de sais de rosuvastatina - Google Patents
processo de preparação de sais de rosuvastatinaInfo
- Publication number
- BRPI1005147A2 BRPI1005147A2 BRPI1005147A BRPI1005147A BRPI1005147A2 BR PI1005147 A2 BRPI1005147 A2 BR PI1005147A2 BR PI1005147 A BRPI1005147 A BR PI1005147A BR PI1005147 A BRPI1005147 A BR PI1005147A BR PI1005147 A2 BRPI1005147 A2 BR PI1005147A2
- Authority
- BR
- Brazil
- Prior art keywords
- preparation process
- salt preparation
- rosuvastatin salt
- rosuvastatin
- salt
- Prior art date
Links
- 238000002360 preparation method Methods 0.000 title 1
- BPRHUIZQVSMCRT-VEUZHWNKSA-N rosuvastatin Chemical class CC(C)C1=NC(N(C)S(C)(=O)=O)=NC(C=2C=CC(F)=CC=2)=C1\C=C\[C@@H](O)C[C@@H](O)CC(O)=O BPRHUIZQVSMCRT-VEUZHWNKSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Medicinal Chemistry (AREA)
- Hematology (AREA)
- Engineering & Computer Science (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| HU0900019A HU0900019D0 (en) | 2009-01-15 | 2009-01-15 | Process for producing rosuvastatin |
| HU0900019 | 2009-01-15 | ||
| HU0900460 | 2009-07-24 | ||
| HU0900460A HU230848B1 (en) | 2009-07-24 | 2009-07-24 | Process for producing rosuvastatin salts |
| PCT/HU2010/000007 WO2010082072A1 (en) | 2009-01-15 | 2010-01-15 | Process for the preparation of rosuvastatin salts |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI1005147A2 true BRPI1005147A2 (pt) | 2019-09-24 |
Family
ID=89989132
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI1005147A BRPI1005147A2 (pt) | 2009-01-15 | 2010-01-15 | processo de preparação de sais de rosuvastatina |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US8507513B2 (pt) |
| EP (1) | EP2389365A1 (pt) |
| CN (1) | CN102317267A (pt) |
| AU (1) | AU2010205464A1 (pt) |
| BR (1) | BRPI1005147A2 (pt) |
| CA (1) | CA2749727A1 (pt) |
| EA (1) | EA021942B1 (pt) |
| MX (1) | MX2011007478A (pt) |
| WO (1) | WO2010082072A1 (pt) |
| ZA (1) | ZA201105124B (pt) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU227696B1 (en) * | 2006-04-13 | 2011-12-28 | Egyt Gyogyszervegyeszeti Gyar | Zinc salt of rosuvastatin, process for its preparation and pharmaceutical compositions containing it |
| JP5702778B2 (ja) * | 2009-07-24 | 2015-04-15 | エギシュ ヂョヂセルヂャール ザートケルエン ミケデ レースヴェーニタールササーグ | 結晶型ｉのロスバスタチン亜鉛塩 |
| HU230737B1 (hu) | 2010-11-16 | 2018-01-29 | EGIS Gyógyszergyár Nyrt | Eljárás rosuvastatin só előállítására |
| HU230987B1 (hu) * | 2010-11-29 | 2019-08-28 | Egis Gyógyszergyár Nyrt. | Eljárás nagy tisztaságú gyógyszeripari intermedierek előállítására |
| HU229260B1 (en) | 2010-11-29 | 2013-10-28 | Egis Gyogyszergyar Nyrt | Process for preparation of rosuvastatin salts |
Family Cites Families (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2648897B2 (ja) | 1991-07-01 | 1997-09-03 | 塩野義製薬株式会社 | ピリミジン誘導体 |
| GB0003305D0 (en) | 2000-02-15 | 2000-04-05 | Zeneca Ltd | Pyrimidine derivatives |
| AU2003228010A1 (en) | 2002-05-21 | 2003-12-02 | Ranbaxy Laboratories Limited | Process for the preparation of rosuvastatin |
| GB0218781D0 (en) | 2002-08-13 | 2002-09-18 | Astrazeneca Ab | Chemical process |
| EP1562912A2 (en) | 2003-08-28 | 2005-08-17 | Teva Pharmaceutical Industries Limited | Process for preparation of rosuvastatin calcium |
| UY28501A1 (es) * | 2003-09-10 | 2005-04-29 | Astrazeneca Uk Ltd | Compuestos químicos |
| GB0321827D0 (en) * | 2003-09-18 | 2003-10-15 | Astrazeneca Uk Ltd | Chemical compounds |
| CN1886383A (zh) | 2003-10-22 | 2006-12-27 | 兰贝克赛实验室有限公司 | 无定形罗苏伐他汀钙的制备方法 |
| GB0324791D0 (en) | 2003-10-24 | 2003-11-26 | Astrazeneca Ab | Chemical process |
| CA2546701C (en) * | 2003-11-24 | 2010-07-27 | Teva Pharmaceutical Industries Ltd. | Crystalline ammonium salts of rosuvastatin |
| EP1709008A1 (en) | 2004-01-19 | 2006-10-11 | Ranbaxy Laboratories Limited | Salts of hmg-coa reductase inhibitors and use thereof |
| HU227120B1 (hu) | 2005-05-26 | 2010-07-28 | Richter Gedeon Nyrt | Eljárás rosuvastatin kalciumsójának elõállítására új intermediereken keresztül |
| JP5146965B2 (ja) * | 2005-06-24 | 2013-02-20 | レツク・フアーマシユーテイカルズ・デー・デー | 不純物を含まない非晶質ロスバスタチンカルシウムの調製方法 |
| CN101203496B (zh) * | 2005-06-24 | 2011-04-20 | 力奇制药公司 | 纯的无定形瑞舒伐他汀钙的制备方法 |
| HU227696B1 (en) * | 2006-04-13 | 2011-12-28 | Egyt Gyogyszervegyeszeti Gyar | Zinc salt of rosuvastatin, process for its preparation and pharmaceutical compositions containing it |
| EP2024341B1 (en) | 2006-05-03 | 2015-12-02 | MSN Laboratories Private Limited | Novel process for statins and its pharmaceutically acceptable salts thereof |
| EP2066644A2 (en) * | 2006-08-04 | 2009-06-10 | Glenmark Pharmaceuticals Limited | Salts of rosuvastatin and processes for their preparation |
| ES2567171T3 (es) * | 2006-10-09 | 2016-04-20 | Msn Laboratories Private Limited | Nuevo procedimiento para la preparación de estatinas y sus sales farmacéuticamente aceptables |
| US20080249120A1 (en) * | 2006-11-22 | 2008-10-09 | Glenmark Pharmaceuticals Limited | Pharmaceutical compositions |
| US20100069635A1 (en) | 2006-11-29 | 2010-03-18 | Dr. Reddy's Laboratories Ltd. | Rosuvastatin dehydroabietylamine salt |
| PL2387566T3 (pl) * | 2009-01-14 | 2014-10-31 | Krka Tovarna Zdravil D D Novo Mesto | Sposób przygotowania rosuwastatyny |
-
2010
- 2010-01-15 AU AU2010205464A patent/AU2010205464A1/en not_active Abandoned
- 2010-01-15 MX MX2011007478A patent/MX2011007478A/es active IP Right Grant
- 2010-01-15 US US13/143,943 patent/US8507513B2/en not_active Expired - Fee Related
- 2010-01-15 WO PCT/HU2010/000007 patent/WO2010082072A1/en not_active Ceased
- 2010-01-15 CA CA2749727A patent/CA2749727A1/en not_active Abandoned
- 2010-01-15 CN CN2010800078203A patent/CN102317267A/zh active Pending
- 2010-01-15 EP EP10707657A patent/EP2389365A1/en not_active Withdrawn
- 2010-01-15 BR BRPI1005147A patent/BRPI1005147A2/pt not_active IP Right Cessation
- 2010-01-15 EA EA201190093A patent/EA021942B1/ru not_active IP Right Cessation
-
2011
- 2011-07-12 ZA ZA2011/05124A patent/ZA201105124B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| US20120116082A1 (en) | 2012-05-10 |
| EA021942B1 (ru) | 2015-10-30 |
| WO2010082072A8 (en) | 2010-10-14 |
| EP2389365A1 (en) | 2011-11-30 |
| WO2010082072A1 (en) | 2010-07-22 |
| CA2749727A1 (en) | 2010-07-22 |
| ZA201105124B (en) | 2012-09-26 |
| US8507513B2 (en) | 2013-08-13 |
| AU2010205464A1 (en) | 2011-08-18 |
| CN102317267A (zh) | 2012-01-11 |
| MX2011007478A (es) | 2011-09-15 |
| EA201190093A1 (ru) | 2012-02-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] | ||
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |