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BRPI0811956A2 - Solução tópica não aquosa de diclofenaco e processo para sua preparação - Google Patents

Solução tópica não aquosa de diclofenaco e processo para sua preparação

Info

Publication number
BRPI0811956A2
BRPI0811956A2 BRPI0811956-2A2A BRPI0811956A BRPI0811956A2 BR PI0811956 A2 BRPI0811956 A2 BR PI0811956A2 BR PI0811956 A BRPI0811956 A BR PI0811956A BR PI0811956 A2 BRPI0811956 A2 BR PI0811956A2
Authority
BR
Brazil
Prior art keywords
dichlophenac
aqueous
preparation
topical solution
topical
Prior art date
Application number
BRPI0811956-2A2A
Other languages
English (en)
Inventor
Ketan R Patel
Original Assignee
Ketan R Patel
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ketan R Patel filed Critical Ketan R Patel
Publication of BRPI0811956A2 publication Critical patent/BRPI0811956A2/pt
Publication of BRPI0811956A8 publication Critical patent/BRPI0811956A8/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/0014Skin, i.e. galenical aspects of topical compositions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/196Carboxylic acids, e.g. valproic acid having an amino group the amino group being directly attached to a ring, e.g. anthranilic acid, mefenamic acid, diclofenac, chlorambucil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/08Solutions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Dermatology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
BRPI0811956A 2007-06-08 2008-06-09 Solução tópica não aquosa de diclofenaco e processo para sua preparação BRPI0811956A8 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN1092MU2007 2007-06-08
PCT/IN2008/000363 WO2009047785A2 (en) 2007-06-08 2008-06-09 A non-aqueous topical solution of diclofenac and process for preparing the same

Publications (2)

Publication Number Publication Date
BRPI0811956A2 true BRPI0811956A2 (pt) 2014-11-11
BRPI0811956A8 BRPI0811956A8 (pt) 2015-09-22

Family

ID=40524886

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0811956A BRPI0811956A8 (pt) 2007-06-08 2008-06-09 Solução tópica não aquosa de diclofenaco e processo para sua preparação

Country Status (22)

Country Link
US (1) US10702469B2 (pt)
EP (1) EP2211837B1 (pt)
JP (2) JP5535066B2 (pt)
KR (1) KR101517494B1 (pt)
CN (1) CN101790370B (pt)
AP (1) AP3643A (pt)
AU (1) AU2008309170B2 (pt)
BR (1) BRPI0811956A8 (pt)
CA (1) CA2697458C (pt)
CO (1) CO6270203A2 (pt)
CU (1) CU23999B1 (pt)
DK (1) DK2211837T3 (pt)
EA (1) EA018119B1 (pt)
ES (1) ES2445443T3 (pt)
IL (1) IL202009A (pt)
MX (1) MX2009013352A (pt)
MY (1) MY151437A (pt)
PL (1) PL2211837T3 (pt)
PT (1) PT2211837E (pt)
UA (1) UA97529C2 (pt)
WO (1) WO2009047785A2 (pt)
ZA (1) ZA200908705B (pt)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100099766A1 (en) * 2008-10-16 2010-04-22 Novartis Ag Topical NSAID compositions having sensate component
EP2416816B1 (en) * 2009-04-10 2014-10-15 Spiracur Inc. Methods and devices for applying closed incision negative pressure wound therapy
US10695431B2 (en) 2010-10-29 2020-06-30 Infirst Healthcare Limited Solid solution compositions and use in cardiovascular disease
US9744132B2 (en) 2010-10-29 2017-08-29 Infirst Healthcare Limited Solid solution compositions and use in chronic inflammation
US8895537B2 (en) 2010-10-29 2014-11-25 Infirst Healthcare Ltd. Compositions and methods for treating cardiovascular diseases
US9308213B2 (en) 2010-10-29 2016-04-12 Infirst Healthcare Limited Solid solution compositions and use in chronic inflammation
US11202831B2 (en) 2010-10-29 2021-12-21 Infirst Healthcare Limited Solid solution compositions and use in cardiovascular disease
US11730709B2 (en) 2010-10-29 2023-08-22 Infirst Healthcare Limited Compositions and methods for treating severe pain
US9504664B2 (en) 2010-10-29 2016-11-29 Infirst Healthcare Limited Compositions and methods for treating severe pain
US11224659B2 (en) 2010-10-29 2022-01-18 Infirst Healthcare Limited Solid solution compositions and use in severe pain
US9271950B2 (en) 2010-10-29 2016-03-01 Infirst Healthcare Limited Compositions for treating chronic inflammation and inflammatory diseases
US10695432B2 (en) 2010-10-29 2020-06-30 Infirst Healthcare Limited Solid solution compositions and use in severe pain
US9737500B2 (en) 2010-10-29 2017-08-22 Infirst Healthcare Limited Compositions and methods for treating severe pain
ITMI20121205A1 (it) * 2012-07-11 2014-01-12 Glycores 2000 Srl Composizione con attivita' antinfiammatoria ed analgesica da somministrare per uso esterno mediante vaporizzazione
JP2014152172A (ja) * 2013-02-08 2014-08-25 Daiya Seiyaku Kk 清涼感付与外用組成物、清涼感付与貼付剤、清涼感付与方法、清涼感付与外用組成物の製造方法、及び、清涼感付与貼付剤の製造方法
CA3186350A1 (en) * 2013-02-27 2014-09-04 Argenta Innovation Limited Transdermal formulations
JP6738120B2 (ja) * 2013-03-29 2020-08-12 小林製薬株式会社 外用医薬組成物
JP6580305B2 (ja) * 2014-03-30 2019-09-25 小林製薬株式会社 外用医薬組成物
JP6580306B2 (ja) * 2014-03-30 2019-09-25 小林製薬株式会社 外用医薬組成物
JP6599083B2 (ja) * 2014-03-30 2019-10-30 小林製薬株式会社 外用医薬組成物
SG11201808231VA (en) * 2016-03-31 2018-10-30 Smartech Topical Inc Delivery system
US20210137829A1 (en) * 2017-03-07 2021-05-13 Yissum Research Development Company Of The Hebrew University Of Jerusalem Ltd. Topical delivery systems for active compounds
JP2018030893A (ja) * 2017-11-14 2018-03-01 ダイヤ製薬株式会社 清涼感付与外用組成物の製造方法及び清涼感付与貼付剤の製造方法
JP7515582B2 (ja) * 2019-11-06 2024-07-12 スマーテック トピカル,インコーポレイテッド シクロオキシゲナーゼ阻害剤の局所配合剤およびその使用
JP7706235B2 (ja) * 2020-12-18 2025-07-11 小林製薬株式会社 外用医薬組成物
WO2023180792A1 (en) 2022-03-25 2023-09-28 Glycores 2000 Srl Topical pharmaceutical composition with anti-inflammatory and analgesic activity and uses thereof

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4353896A (en) * 1981-06-08 1982-10-12 Levy Michael A Penetrating topical medicament
US4933184A (en) 1983-12-22 1990-06-12 American Home Products Corp. (Del) Menthol enhancement of transdermal drug delivery
CA1236029A (en) 1984-05-14 1988-05-03 Edmund Sandborn Pharmaceutical solutions comprising dimethyl sulfoxide
DE3522550A1 (de) 1985-06-24 1987-01-02 Klinge Co Chem Pharm Fab Aufspruehbare pharmazeutische zubereitung fuer die topische anwendung
US5093133A (en) * 1990-01-24 1992-03-03 Mcneil-Ppc, Inc. Method for percutaneous delivery of ibuprofen using hydroalcoholic gel
US5318960A (en) * 1992-06-03 1994-06-07 Frank Toppo System for transdermal delivery of pain relieving substances
US5985860A (en) 1992-06-03 1999-11-16 Toppo; Frank System for transdermal delivery of pain relieving substances
US5665378A (en) 1994-09-30 1997-09-09 Davis; Roosevelt Transdermal therapeutic formulation
US5654337A (en) 1995-03-24 1997-08-05 II William Scott Snyder Topical formulation for local delivery of a pharmaceutically active agent
US7833543B2 (en) * 1995-06-07 2010-11-16 Durect Corporation High viscosity liquid controlled delivery system and medical or surgical device
US5968542A (en) * 1995-06-07 1999-10-19 Southern Biosystems, Inc. High viscosity liquid controlled delivery system as a device
WO1997028794A1 (fr) * 1996-02-07 1997-08-14 Tsumura & Co. Solution aqueuse transparente de diclofenac sodique, compositions medicinales, et utilisations
DE19725615A1 (de) 1997-06-17 1998-12-24 Permamed Ag Zur topischen Applikation bestimmte Diclofenac-Lösung
US5976566A (en) * 1997-08-29 1999-11-02 Macrochem Corporation Non-steroidal antiinflammtory drug formulations for topical application to the skin
US6193996B1 (en) 1998-04-02 2001-02-27 3M Innovative Properties Company Device for the transdermal delivery of diclofenac
CH693625A5 (it) 1999-02-18 2003-11-28 Inpharma Sa Composizioni farmaceutiche contenenti composti ad attività promotrice di assorbimento di principi attivi.
DE60236084D1 (de) * 2001-05-31 2010-06-02 Hisamitsu Pharmaceutical Co Perkutan resorbierbare pflaster
US20070196453A1 (en) * 2004-06-07 2007-08-23 Jie Zhang Two or more non-volatile solvent-containing compositions and methods for dermal delivery of drugs
US20080319092A1 (en) * 2005-08-05 2008-12-25 Nuvo Research Inc. Transdermal Drug Delivery Formulation

Also Published As

Publication number Publication date
JP5535066B2 (ja) 2014-07-02
UA97529C2 (ru) 2012-02-27
WO2009047785A9 (en) 2010-03-11
IL202009A (en) 2015-10-29
BRPI0811956A8 (pt) 2015-09-22
WO2009047785A3 (en) 2009-07-02
JP2010529110A (ja) 2010-08-26
US10702469B2 (en) 2020-07-07
CO6270203A2 (es) 2011-04-20
MY151437A (en) 2014-05-30
CN101790370B (zh) 2013-06-12
PT2211837E (pt) 2014-02-17
ES2445443T3 (es) 2014-03-03
CU23999B1 (es) 2014-06-27
ZA200908705B (en) 2010-08-25
DK2211837T3 (da) 2014-02-10
EA018119B1 (ru) 2013-05-30
KR101517494B1 (ko) 2015-05-04
EA200971099A1 (ru) 2010-06-30
KR20100047840A (ko) 2010-05-10
CA2697458A1 (en) 2009-04-16
CN101790370A (zh) 2010-07-28
AP3643A (en) 2016-03-16
US20100120918A1 (en) 2010-05-13
IL202009A0 (en) 2010-06-16
AU2008309170B2 (en) 2013-03-14
PL2211837T3 (pl) 2014-05-30
CU20090206A7 (es) 2011-09-21
AU2008309170A1 (en) 2009-04-16
HK1147066A1 (en) 2011-07-29
EP2211837B1 (en) 2013-11-13
MX2009013352A (es) 2010-05-21
JP5734479B2 (ja) 2015-06-17
EP2211837A2 (en) 2010-08-04
WO2009047785A2 (en) 2009-04-16
AP2010005169A0 (en) 2010-02-28
JP2014098046A (ja) 2014-05-29
CA2697458C (en) 2016-02-09

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Legal Events

Date Code Title Description
B25A Requested transfer of rights approved

Owner name: TROIKAA PHARMACEUTICALS LTD (IN)

B07D Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]
B07E Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]

Free format text: NOTIFICACAO DE ANUENCIA RELACIONADA COM O ART 229 DA LPI

B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B09B Patent application refused [chapter 9.2 patent gazette]
B12B Appeal against refusal [chapter 12.2 patent gazette]
B350 Update of information on the portal [chapter 15.35 patent gazette]