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BRPI0811165A2 - Método para a preparação de um composto de éster, e, composição de branqueamento da pele - Google Patents

Método para a preparação de um composto de éster, e, composição de branqueamento da pele

Info

Publication number
BRPI0811165A2
BRPI0811165A2 BRPI0811165-0A2A BRPI0811165A BRPI0811165A2 BR PI0811165 A2 BRPI0811165 A2 BR PI0811165A2 BR PI0811165 A BRPI0811165 A BR PI0811165A BR PI0811165 A2 BRPI0811165 A2 BR PI0811165A2
Authority
BR
Brazil
Prior art keywords
preparing
ester compound
skin
composition
skin blanking
Prior art date
Application number
BRPI0811165-0A2A
Other languages
English (en)
Inventor
Stephanie Kay Clendennen
Neil Warren Boaz
Jeffrey Michael Clauson
Original Assignee
Eastman Chem Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Eastman Chem Co filed Critical Eastman Chem Co
Publication of BRPI0811165A2 publication Critical patent/BRPI0811165A2/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P7/00Preparation of oxygen-containing organic compounds
    • C12P7/62Carboxylic acid esters
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/21Esters, e.g. nitroglycerine, selenocyanates
    • A61K31/215Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids
    • A61K31/235Esters, e.g. nitroglycerine, selenocyanates of carboxylic acids having an aromatic ring attached to a carboxyl group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D309/00Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
    • C07D309/34Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D309/36Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C07D309/38Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms one oxygen atom in position 2 or 4, e.g. pyrones
    • CCHEMISTRY; METALLURGY
    • C12BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
    • C12PFERMENTATION OR ENZYME-USING PROCESSES TO SYNTHESISE A DESIRED CHEMICAL COMPOUND OR COMPOSITION OR TO SEPARATE OPTICAL ISOMERS FROM A RACEMIC MIXTURE
    • C12P17/00Preparation of heterocyclic carbon compounds with only O, N, S, Se or Te as ring hetero atoms
    • C12P17/02Oxygen as only ring hetero atoms
    • C12P17/06Oxygen as only ring hetero atoms containing a six-membered hetero ring, e.g. fluorescein

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Epidemiology (AREA)
  • General Engineering & Computer Science (AREA)
  • Biotechnology (AREA)
  • Microbiology (AREA)
  • Emergency Medicine (AREA)
  • Dermatology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Cosmetics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BRPI0811165-0A2A 2007-06-08 2008-05-27 Método para a preparação de um composto de éster, e, composição de branqueamento da pele BRPI0811165A2 (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US11/811,055 US20080306144A1 (en) 2007-06-08 2007-06-08 Hydroxybenzyl or hydroxypyranonemethyl esters as tyrosinase inhibitors
PCT/US2008/006699 WO2008153784A2 (en) 2007-06-08 2008-05-27 Hydroxybenzyl or hydroxypyranonemethyl esters as tyrosinase inhibitors

Publications (1)

Publication Number Publication Date
BRPI0811165A2 true BRPI0811165A2 (pt) 2014-12-23

Family

ID=40096459

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI0811165-0A2A BRPI0811165A2 (pt) 2007-06-08 2008-05-27 Método para a preparação de um composto de éster, e, composição de branqueamento da pele

Country Status (9)

Country Link
US (2) US20080306144A1 (pt)
EP (2) EP2155886B1 (pt)
JP (1) JP2010528654A (pt)
CN (1) CN101680008B (pt)
AT (1) ATE548084T1 (pt)
BR (1) BRPI0811165A2 (pt)
DK (1) DK2155886T3 (pt)
ES (1) ES2383385T3 (pt)
WO (1) WO2008153784A2 (pt)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP5618126B2 (ja) * 2010-01-21 2014-11-05 三菱レイヨン株式会社 エステル化合物の製造方法
EP2666460A4 (en) * 2011-01-20 2014-06-11 Nichirei Biosciences Inc SKIN HELLENDER WITH 3-HYDROXY-2-PYRONE
KR102777432B1 (ko) * 2019-02-19 2025-03-07 (주)애거슨바이오 모노메틸 푸마레이트 유도체 및 이들의 약학적 조성물
WO2022075787A1 (ko) * 2020-10-07 2022-04-14 주식회사 큐롬바이오사이언스 신규한 퀴논 유도체 화합물 및 이의 용도

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS567710A (en) * 1979-06-28 1981-01-27 Sansho Seiyaku Kk Whitening cosmetic
JP2565513B2 (ja) * 1987-09-25 1996-12-18 三省製薬株式会社 メラニン生成抑制外用薬剤
AU647603B2 (en) * 1991-04-02 1994-03-24 Hoechst Aktiengesellschaft An immobilized biocatalyst, its preparation and use for ester synthesis in a column reactor
JP2002257704A (ja) 2001-02-28 2002-09-11 Ricoh Co Ltd 近接場光プローブ及びその製造方法
JP4389101B2 (ja) * 2001-09-04 2009-12-24 独立行政法人産業技術総合研究所 コウジ酸エステルおよびその合成方法
KR20060031007A (ko) * 2004-10-07 2006-04-12 주식회사 바이오랜드 피부 미백 효과를 갖는 천마 추출물 및 이로부터 분리된화합물을 함유하는 화장료 조성물
KR101527739B1 (ko) * 2005-02-18 2015-06-12 아지노모토 가부시키가이샤 캡시노이드 조성물 및 이의 제조방법

Also Published As

Publication number Publication date
CN101680008A (zh) 2010-03-24
CN101680008B (zh) 2013-06-26
EP2155886A2 (en) 2010-02-24
JP2010528654A (ja) 2010-08-26
ES2383385T3 (es) 2012-06-20
EP2155886B1 (en) 2012-03-07
US20080306144A1 (en) 2008-12-11
ATE548084T1 (de) 2012-03-15
US20110129430A1 (en) 2011-06-02
DK2155886T3 (da) 2012-05-29
WO2008153784A3 (en) 2009-04-02
WO2008153784A2 (en) 2008-12-18
EP2428577A1 (en) 2012-03-14
EP2428577B1 (en) 2014-01-22

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]
B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]