BRPI0509211A - uso de compostos de peptìdeo para o tratamento de dor em neuropatia diabética - Google Patents
uso de compostos de peptìdeo para o tratamento de dor em neuropatia diabéticaInfo
- Publication number
- BRPI0509211A BRPI0509211A BRPI0509211-6A BRPI0509211A BRPI0509211A BR PI0509211 A BRPI0509211 A BR PI0509211A BR PI0509211 A BRPI0509211 A BR PI0509211A BR PI0509211 A BRPI0509211 A BR PI0509211A
- Authority
- BR
- Brazil
- Prior art keywords
- pain
- treatment
- diabetic neuropathy
- peptide compounds
- compounds
- Prior art date
Links
- 208000032131 Diabetic Neuropathies Diseases 0.000 title abstract 3
- 150000001875 compounds Chemical class 0.000 title abstract 3
- 108090000765 processed proteins & peptides Proteins 0.000 title abstract 2
- 206010036105 Polyneuropathy Diseases 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 230000007824 polyneuropathy Effects 0.000 abstract 1
- 230000001953 sensory effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
- A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/16—Amides, e.g. hydroxamic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/05—Dipeptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Gastroenterology & Hepatology (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Diabetes (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
Abstract
USO DE COMPOSTOS DE PEPTìDEO PARA O TRATAMENTO DE DOR EM NEUROPATIA DIABéTICA. A presente invenção refere-se ao uso de compostos para o tratamento de dor em neuropatia diabética dolorosa, de preferência em polineuropatia sensória distal diabética.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US55649904P | 2004-03-26 | 2004-03-26 | |
| EP04007360A EP1579858A1 (en) | 2004-03-26 | 2004-03-26 | Novel use of peptide compounds for treating pain in painful diabetic neuropathy |
| PCT/EP2005/003176 WO2005092313A1 (en) | 2004-03-26 | 2005-03-24 | Novel use of peptide compounds for treating pain in painful diabetic neuropathy |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0509211A true BRPI0509211A (pt) | 2007-08-28 |
Family
ID=34854637
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0509211-6A BRPI0509211A (pt) | 2004-03-26 | 2005-03-24 | uso de compostos de peptìdeo para o tratamento de dor em neuropatia diabética |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20060100157A1 (pt) |
| EP (2) | EP1579858A1 (pt) |
| JP (1) | JP2007530493A (pt) |
| CN (1) | CN1938010B (pt) |
| AU (1) | AU2005226928B2 (pt) |
| BR (1) | BRPI0509211A (pt) |
| CA (1) | CA2558311A1 (pt) |
| EA (1) | EA012176B1 (pt) |
| MX (1) | MXPA06010995A (pt) |
| NZ (1) | NZ549668A (pt) |
| SG (1) | SG151309A1 (pt) |
| TW (1) | TW200701977A (pt) |
| UA (1) | UA90467C2 (pt) |
| WO (1) | WO2005092313A1 (pt) |
| ZA (1) | ZA200607269B (pt) |
Families Citing this family (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP1243262B1 (en) | 2001-03-20 | 2006-05-31 | Schwarz Pharma Ag | Novel use of a peptide class of compound for treating non-neuropathic inflammatory pain |
| EP1243263B1 (en) * | 2001-03-21 | 2002-11-27 | Schwarz Pharma Ag | Novel use of a peptide class of compound for treating allodynia or other different types of chronic or phantom pain |
| EP1689378B1 (en) | 2003-12-02 | 2009-04-15 | Schwarz Pharma Ag | Novel use of peptide compounds for treating central neuropathic pain |
| US20100256179A1 (en) * | 2004-03-26 | 2010-10-07 | Ucb Pharma Gmbh | Combination therapy for pain in painful diabetic neuropathy |
| US20070042969A1 (en) * | 2004-03-26 | 2007-02-22 | Srz Properties, Inc. | Combination therapy for pain in painful diabetic neuropathy |
| EA013591B1 (ru) | 2004-04-16 | 2010-06-30 | Шварц Фарма Аг | Применение пептидных соединений для профилактики, облегчения и лечения головной боли и болезненных состояний, связанных с или вызванных распространяющейся кортикальной депрессией (csd) |
| EP1604655A1 (en) | 2004-06-09 | 2005-12-14 | Schwarz Pharma Ag | Novel use of peptide compounds for treating pain in trigeminal neuralgia |
| PL1781276T3 (pl) | 2004-08-27 | 2010-11-30 | Ucb Pharma Gmbh | Zastosowanie związków peptydowych do leczenia bólu związanego z rakiem kości, bólu indukowanego przez chemioterapię oraz nukleozydy |
| EP1642889A1 (en) * | 2004-10-02 | 2006-04-05 | Schwarz Pharma Ag | Improved synthesis scheme for lacosamide |
| US20060252749A1 (en) * | 2005-01-28 | 2006-11-09 | Srz Properties, Inc. | Lacosamide for add-on therapy of psychosis |
| EP1754476A1 (en) * | 2005-08-18 | 2007-02-21 | Schwarz Pharma Ag | Lacosamide (SPM 927) for treating myalgia, e.g. fibromyalgia |
| US20070043120A1 (en) * | 2005-08-18 | 2007-02-22 | Bettina Beyreuther | Therapeutic combination for painful medical conditions |
| US7902401B2 (en) * | 2006-12-14 | 2011-03-08 | Nps Pharmaceuticals, Inc. | Fluorinated compounds |
| GB0603008D0 (en) * | 2006-02-14 | 2006-03-29 | Portela & Ca Sa | Method |
| AR061250A1 (es) * | 2006-06-08 | 2008-08-13 | Sanol Arznei Schwarz Gmbh | Combinacion terapeutica para condiciones medicas dolorosas |
| EP1873527A1 (en) * | 2006-06-30 | 2008-01-02 | Schwarz Pharma Ag | Method for identifying CRMP modulators |
| AU2007260207B2 (en) | 2006-06-15 | 2012-11-08 | Ucb Pharma Gmbh | Pharmaceutical composition with synergistic anticonvulsant effect |
| CN101466390B (zh) | 2006-06-15 | 2014-03-12 | 优时比制药有限公司 | 用于治疗难治性癫痫持续状态的肽类化合物 |
| EP2099444A4 (en) * | 2006-12-14 | 2012-11-07 | Nps Pharma Inc | USE OF D-SERIN DERIVATIVES FOR THE TREATMENT OF ANTIBODIES |
| EP2509939A4 (en) | 2009-09-23 | 2013-09-18 | Univ North Carolina | NOVEL N-BENZYLAMIDE SUBSTITUTED DERIVATIVES OF 2- (ACYLAMIDO) ACETIC ACID AND 2- (ACYLAMIDO) PROPIONIC ACIDS: POWERFUL NEUROLOGIC AGENTS |
| MX350056B (es) * | 2009-11-03 | 2017-08-25 | Lupin Ltd | Formulacion de liberacion modificada de lacosamida. |
| EP2468261A1 (en) | 2010-12-02 | 2012-06-27 | UCB Pharma GmbH | Formulation of lacosamide |
| EP2645997B1 (en) | 2010-12-02 | 2022-08-10 | UCB Pharma GmbH | Once daily formulation of lacosamide |
| AU2016381366A1 (en) | 2015-12-30 | 2018-06-28 | Adamas Pharmaceuticals, Inc. | Methods and compositions for the treatment of seizure-related disorders |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5378729A (en) * | 1985-02-15 | 1995-01-03 | Research Corporation Technologies, Inc. | Amino acid derivative anticonvulsant |
| US5585358A (en) * | 1993-07-06 | 1996-12-17 | Yissum Research Development Corporation Of The Hebrew University Of Jerusalem | Derivatives of valproic acid amides and 2-valproenoic acid amides, method of making and use thereof as anticonvulsant agents |
| US6589994B1 (en) * | 1996-08-30 | 2003-07-08 | Nps Pharmaceuticals, Inc. | Treating a variety of pathological conditions, including spasticity and convulsions, by effecting a modulation of CNS activity with isovaleramide, isovaleric acid, or a related compound |
| ATE301995T1 (de) * | 2000-08-17 | 2005-09-15 | Teva Pharma | Verwendung von derivaten der valproinsäureamide und 2-valproinsäureamid zur behandlung und prävention von schmerzen und/oder kopfschmerzen |
| DK1695703T3 (da) * | 2000-08-25 | 2010-10-25 | Res Corp Technologies Inc | Nye anvendelser for aminosyrekrampestillende midler |
| EP1243262B1 (en) * | 2001-03-20 | 2006-05-31 | Schwarz Pharma Ag | Novel use of a peptide class of compound for treating non-neuropathic inflammatory pain |
| EP1243263B1 (en) * | 2001-03-21 | 2002-11-27 | Schwarz Pharma Ag | Novel use of a peptide class of compound for treating allodynia or other different types of chronic or phantom pain |
| EP1689378B1 (en) * | 2003-12-02 | 2009-04-15 | Schwarz Pharma Ag | Novel use of peptide compounds for treating central neuropathic pain |
| US20060009384A1 (en) * | 2003-12-05 | 2006-01-12 | David Rudd | Novel use of peptide compounds for treating status epilepticus or related conditions |
| US20070042969A1 (en) * | 2004-03-26 | 2007-02-22 | Srz Properties, Inc. | Combination therapy for pain in painful diabetic neuropathy |
| EA013591B1 (ru) * | 2004-04-16 | 2010-06-30 | Шварц Фарма Аг | Применение пептидных соединений для профилактики, облегчения и лечения головной боли и болезненных состояний, связанных с или вызванных распространяющейся кортикальной депрессией (csd) |
| EP1604654A1 (en) * | 2004-05-18 | 2005-12-14 | Schwarz Pharma Ag | Novel use of peptide compounds for treating dyskinesia |
| EP1604656A1 (en) * | 2004-06-09 | 2005-12-14 | Schwarz Pharma Ag | Novel use of peptide compounds for treating amyotrophic lateral sclerosis (ALS) |
| US7427601B2 (en) * | 2004-06-24 | 2008-09-23 | Schwarz Pharma Ag | Method for treating tremor |
| EP1642889A1 (en) * | 2004-10-02 | 2006-04-05 | Schwarz Pharma Ag | Improved synthesis scheme for lacosamide |
| US20060252749A1 (en) * | 2005-01-28 | 2006-11-09 | Srz Properties, Inc. | Lacosamide for add-on therapy of psychosis |
| US20070043120A1 (en) * | 2005-08-18 | 2007-02-22 | Bettina Beyreuther | Therapeutic combination for painful medical conditions |
| EP1754476A1 (en) * | 2005-08-18 | 2007-02-21 | Schwarz Pharma Ag | Lacosamide (SPM 927) for treating myalgia, e.g. fibromyalgia |
| US20070048372A1 (en) * | 2005-08-18 | 2007-03-01 | Srz Properties, Inc. | Method for treating non-inflammatory osteoarthritic pain |
-
2004
- 2004-03-26 EP EP04007360A patent/EP1579858A1/en not_active Withdrawn
-
2005
- 2005-03-24 SG SG200902059-5A patent/SG151309A1/en unknown
- 2005-03-24 WO PCT/EP2005/003176 patent/WO2005092313A1/en not_active Ceased
- 2005-03-24 CA CA002558311A patent/CA2558311A1/en not_active Abandoned
- 2005-03-24 MX MXPA06010995A patent/MXPA06010995A/es active IP Right Grant
- 2005-03-24 AU AU2005226928A patent/AU2005226928B2/en not_active Ceased
- 2005-03-24 UA UAA200610139A patent/UA90467C2/ru unknown
- 2005-03-24 CN CN2005800097824A patent/CN1938010B/zh not_active Expired - Fee Related
- 2005-03-24 EP EP05716372A patent/EP1737437A1/en not_active Withdrawn
- 2005-03-24 BR BRPI0509211-6A patent/BRPI0509211A/pt not_active IP Right Cessation
- 2005-03-24 EA EA200601777A patent/EA012176B1/ru not_active IP Right Cessation
- 2005-03-24 JP JP2007504367A patent/JP2007530493A/ja active Pending
- 2005-03-24 NZ NZ549668A patent/NZ549668A/en unknown
- 2005-03-25 US US11/089,441 patent/US20060100157A1/en not_active Abandoned
- 2005-07-11 TW TW094123447A patent/TW200701977A/zh unknown
-
2006
- 2006-08-31 ZA ZA200607269A patent/ZA200607269B/xx unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UA90467C2 (ru) | 2010-05-11 |
| EA200601777A1 (ru) | 2007-02-27 |
| MXPA06010995A (es) | 2007-04-16 |
| ZA200607269B (en) | 2008-04-30 |
| CN1938010B (zh) | 2011-01-19 |
| EP1737437A1 (en) | 2007-01-03 |
| NZ549668A (en) | 2010-07-30 |
| SG151309A1 (en) | 2009-04-30 |
| EP1579858A1 (en) | 2005-09-28 |
| AU2005226928A1 (en) | 2005-10-06 |
| EA012176B1 (ru) | 2009-08-28 |
| AU2005226928B2 (en) | 2010-05-13 |
| JP2007530493A (ja) | 2007-11-01 |
| CA2558311A1 (en) | 2005-10-06 |
| TW200701977A (en) | 2007-01-16 |
| US20060100157A1 (en) | 2006-05-11 |
| CN1938010A (zh) | 2007-03-28 |
| WO2005092313A1 (en) | 2005-10-06 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B25D | Requested change of name of applicant approved |
Owner name: UCB PHARMA GMBH (DE) Free format text: NOME ALTERADO DE: SCHWARZ PHARMA AG |
|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 8A ANUIDADE |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2204 DE 02/04/2013. |