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BR9917475B1 - processo para a manufatura de compostos, e, modificação do processo. - Google Patents

processo para a manufatura de compostos, e, modificação do processo.

Info

Publication number
BR9917475B1
BR9917475B1 BRPI9917475-8B1A BR9917475A BR9917475B1 BR 9917475 B1 BR9917475 B1 BR 9917475B1 BR 9917475 A BR9917475 A BR 9917475A BR 9917475 B1 BR9917475 B1 BR 9917475B1
Authority
BR
Brazil
Prior art keywords
compounds
manufacture
modification
process modification
Prior art date
Application number
BRPI9917475-8B1A
Other languages
English (en)
Other versions
BR9917475A (pt
Inventor
John A Robinson
Daniel Obrecht
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of BR9917475A publication Critical patent/BR9917475A/pt
Publication of BR9917475B1 publication Critical patent/BR9917475B1/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K1/00General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length
    • C07K1/04General methods for the preparation of peptides, i.e. processes for the organic chemical preparation of peptides or proteins of any length on carriers
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/02Linear peptides containing at least one abnormal peptide link
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/08Linear peptides containing only normal peptide links having 12 to 20 amino acids
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64Cyclic peptides containing only normal peptide links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Analytical Chemistry (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
BRPI9917475-8B1A 1999-08-30 1999-08-30 processo para a manufatura de compostos, e, modificação do processo. BR9917475B1 (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PCT/EP1999/006369 WO2001016161A1 (en) 1999-08-30 1999-08-30 SYNTHESIS OF TEMPLATE-FIXED β-HAIRPIN LOOP MIMETICS

Publications (2)

Publication Number Publication Date
BR9917475A BR9917475A (pt) 2002-05-14
BR9917475B1 true BR9917475B1 (pt) 2013-07-23

Family

ID=8167411

Family Applications (1)

Application Number Title Priority Date Filing Date
BRPI9917475-8B1A BR9917475B1 (pt) 1999-08-30 1999-08-30 processo para a manufatura de compostos, e, modificação do processo.

Country Status (8)

Country Link
US (2) US6878804B1 (pt)
EP (1) EP1214336A1 (pt)
JP (1) JP4625603B2 (pt)
CN (1) CN1367789B (pt)
AU (1) AU5856699A (pt)
BR (1) BR9917475B1 (pt)
CA (1) CA2382931C (pt)
WO (1) WO2001016161A1 (pt)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR0207502A (pt) 2001-02-23 2004-03-09 Polyphor Ltd Compostos, enanciÈmeros, composição farmacêutica, uso de compostos, e, processo para a fabricação de compostos
US6914123B2 (en) * 2001-04-17 2005-07-05 Genentech, Inc. Hairpin peptides with a novel structural motif and methods relating thereto
CN101157924A (zh) * 2001-12-11 2008-04-09 人体基因组科学有限公司 嗜中性白细胞因子α
EP1532164B1 (en) * 2002-08-20 2012-09-26 Polyphor Ltd. Template-fixed peptidomimetics with antibacterial activity
US7855179B2 (en) 2002-10-02 2010-12-21 Polyphor Ltd. Template-fixed peptidomimetics with antimicrobial activity
ES2305355T3 (es) * 2002-10-02 2008-11-01 Polyphor Ltd. Peptidomimeticos fijados a una matriz con actividad antimicrobiana.
ATE395355T1 (de) * 2003-05-02 2008-05-15 Polyphor Ag Matrizenfixierte peptidmimetika als medikamente gegen hiv und krebs
WO2004096839A1 (en) 2003-05-02 2004-11-11 Polyphor Ag Template-fixed beta-hairpin peptidomimetics with cxcr4 antagonizing activity
GB0323728D0 (en) * 2003-10-10 2003-11-12 Royal College Of Surgeons Ie Peptidomimetics and uses thereof
WO2005047503A1 (en) * 2003-11-15 2005-05-26 Polyphor Ltd. Template fixed βετα-hairpin loop mimetics and their use in phage display
JO2897B1 (en) * 2004-11-05 2015-09-15 نوفارتيس ايه جي Organic compounds
WO2007079597A1 (en) 2006-01-16 2007-07-19 Polyphor Ltd. Template - fixed peptidomimetics with antimicrobial activity
AU2007345497B2 (en) * 2007-01-29 2013-01-17 Polyphor Ltd. Template-fixed peptidomimetics
PL2132221T3 (pl) 2007-02-28 2011-04-29 Polyphor Ltd Przyłączone do matrycy peptydomimetyki
EP2237798A2 (en) 2007-12-12 2010-10-13 Imperial Innovations Limited Methods
AU2009290137A1 (en) * 2008-09-03 2010-03-11 Xenome Ltd Libraries of peptide conjugates and methods for making them
WO2011060832A1 (en) * 2009-11-20 2011-05-26 Polyphor Ag Template-fixed peptidomimetics with ccr10 antagonistic activity

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5475085A (en) 1991-02-07 1995-12-12 Molecumetics, Ltd. Conformationally restricted mimetics of beta turns and beta bulges and peptides containing the same
WO1992013878A2 (en) * 1991-02-07 1992-08-20 Board Of Trustees Of The University Of Illinois Conformationally restricted mimetics of beta turns and beta bulges and peptides containing the same
CA2101599A1 (en) * 1992-08-31 1994-03-01 Wilhelm Bannwarth Tri- and tetracyclic compounds

Also Published As

Publication number Publication date
US6878804B1 (en) 2005-04-12
US20050181454A1 (en) 2005-08-18
CA2382931C (en) 2011-01-25
CN1367789B (zh) 2012-06-06
JP2004511424A (ja) 2004-04-15
WO2001016161A1 (en) 2001-03-08
CN1367789A (zh) 2002-09-04
JP4625603B2 (ja) 2011-02-02
AU5856699A (en) 2001-03-26
CA2382931A1 (en) 2001-03-08
EP1214336A1 (en) 2002-06-19
US7091313B2 (en) 2006-08-15
BR9917475A (pt) 2002-05-14

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Legal Events

Date Code Title Description
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B09A Decision: intention to grant [chapter 9.1 patent gazette]
B16A Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]

Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 23/07/2013, OBSERVADAS AS CONDICOES LEGAIS.

B21F Lapse acc. art. 78, item iv - on non-payment of the annual fees in time

Free format text: REFERENTE A 21A ANUIDADE.

B24J Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)

Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2595 DE 29-09-2020 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.