BR9915965A - Benzilmaltosìdeos de acetal como inibidores da proliferação celular do músculo liso - Google Patents
Benzilmaltosìdeos de acetal como inibidores da proliferação celular do músculo lisoInfo
- Publication number
- BR9915965A BR9915965A BR9915965-1A BR9915965A BR9915965A BR 9915965 A BR9915965 A BR 9915965A BR 9915965 A BR9915965 A BR 9915965A BR 9915965 A BR9915965 A BR 9915965A
- Authority
- BR
- Brazil
- Prior art keywords
- smooth muscle
- acetal
- inhibitors
- cell proliferation
- muscle cell
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/203—Monocyclic carbocyclic rings other than cyclohexane rings; Bicyclic carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Urology & Nephrology (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Neurology (AREA)
- Biochemistry (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Heart & Thoracic Surgery (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Physical Education & Sports Medicine (AREA)
- Saccharide Compounds (AREA)
Abstract
Patente de Invenção: <B>"BENZILMALTOSìDEOS DE ACETAL COMO INIBIDORES DA PROLIFERAçãO CELULAR DO MúSCULO LISO"<D>. Esta invenção fornece inibidores da proliferação celular do músculo liso de fórmula (I), tendo a estrutura (I), em que X, R^ 1^, R^ 2^, R^ 3^, R^ 4^, R^ 5^, R^ 6^, R^ 7^, R^ 8^ e R^ 9^ têm os significados dados nas reivindicações e descrição.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19880398A | 1998-11-24 | 1998-11-24 | |
| PCT/US1999/027828 WO2000031096A1 (en) | 1998-11-24 | 1999-11-23 | Acetal benzylmaltosides as inhibitors of smooth muscle cell proliferation |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9915965A true BR9915965A (pt) | 2001-08-21 |
Family
ID=22734926
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9915965-1A BR9915965A (pt) | 1998-11-24 | 1999-11-23 | Benzilmaltosìdeos de acetal como inibidores da proliferação celular do músculo liso |
Country Status (7)
| Country | Link |
|---|---|
| EP (1) | EP1133509A1 (pt) |
| JP (1) | JP2002530421A (pt) |
| CN (1) | CN1328566A (pt) |
| AU (1) | AU1633000A (pt) |
| BR (1) | BR9915965A (pt) |
| CA (1) | CA2350066A1 (pt) |
| WO (1) | WO2000031096A1 (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2000034295A2 (en) * | 1998-11-24 | 2000-06-15 | American Home Products Corporation | Acylated benzylmaltosides as inhibitors of smooth muscle cell proliferation |
| CN103360437B (zh) * | 2013-04-27 | 2015-10-21 | 江苏教育学院 | 一种硫辛酸糖类衍生物及其制备方法和在制备抗肿瘤药物中的应用 |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL115745A (en) * | 1994-11-07 | 2000-11-21 | American Home Prod | Acylated benzylglycosides and pharmaceutical compositions containing them |
-
1999
- 1999-11-23 CN CN99813691A patent/CN1328566A/zh active Pending
- 1999-11-23 WO PCT/US1999/027828 patent/WO2000031096A1/en not_active Ceased
- 1999-11-23 EP EP99959083A patent/EP1133509A1/en not_active Withdrawn
- 1999-11-23 JP JP2000583924A patent/JP2002530421A/ja active Pending
- 1999-11-23 CA CA002350066A patent/CA2350066A1/en not_active Abandoned
- 1999-11-23 BR BR9915965-1A patent/BR9915965A/pt not_active Application Discontinuation
- 1999-11-23 AU AU16330/00A patent/AU1633000A/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| JP2002530421A (ja) | 2002-09-17 |
| CA2350066A1 (en) | 2000-06-02 |
| WO2000031096A1 (en) | 2000-06-02 |
| CN1328566A (zh) | 2001-12-26 |
| EP1133509A1 (en) | 2001-09-19 |
| AU1633000A (en) | 2000-06-13 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| BR0317822A (pt) | Composição fluoroquìmica | |
| PT1140944E (pt) | Derivados de epotilona e sua utilizacao como agentes antitumorais | |
| DK1268558T3 (da) | Derivater af delvist desulfaterede glycosaminoglycaner forsynet med antiangionisk aktivitet og uden antikoagulerende virkning | |
| MXPA03001511A (es) | Imidazol-5-il-2-amino-pirimidinas como agentes para la inhibicion de la proliferacion celular. | |
| BR9706934A (pt) | Novos compostos de imidazol substituìdo | |
| MY135732A (en) | 5,6-trimethylenepyrimidin - 4 - one compounds | |
| TR199801348T2 (xx) | Heterosikl-kondanse morfinoid t�revleri(II). | |
| BR9706973A (pt) | Novos compostos de imidazol substituídos | |
| IT1313625B1 (it) | Derivati benzimidazolonici aventi affinita' mista per i recettori diserotonina e dopamina. | |
| ES2124668B1 (es) | "nuevosl-arilpirazoles con propiedades plaguicidas. | |
| MA26771A1 (fr) | Benzoheterocycles et leur utilisation comme inhibiteurs de mek. | |
| BR9905873A (pt) | Revestimentos para dispositivos biomédicos | |
| UY25712A1 (es) | Benzamidas sustituidas y su aplicación en medicamentos | |
| TR200103216T2 (tr) | Pirimidinon bileşimleri | |
| DK0901522T3 (da) | Immortaliserede aviære celler | |
| BR0007864A (pt) | Composto, e, uso de um composto | |
| ES2172536T3 (es) | Liberacion y movilizacion de celulas hematopoyeticas. | |
| PT1086096E (pt) | Benzamidas com substituintes etra-hidrofuraniloxi como inibidores da fosfodiesterase 4 | |
| BR9915965A (pt) | Benzilmaltosìdeos de acetal como inibidores da proliferação celular do músculo liso | |
| BR9711273A (pt) | 1,2,3,4- Tetraidro-2-dibenzofuranaminas substituidas e 2- aminociclohepta b benzofuranos | |
| ATE299703T1 (de) | Mmp-hemmer bei bindegewebserweichung | |
| ATE248709T1 (de) | Verbundelemente | |
| ES2196802T3 (es) | Lactatos de citronelilo y/o de dihidrocitronelilo, su preparacion y su utilizacion. | |
| NO305234B1 (no) | Lasteslange-fort°yning | |
| EE04494B1 (et) | 1-oksa-, asa- ja tianaftaleen-2-oon biseetrid fosfolambaani inhibiitoritena |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal acc. article 33 of ipl - extension of time limit for request of examination expired |