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BR9911574A - Ciclooctadepsipeptìdeos substituìdos - Google Patents

Ciclooctadepsipeptìdeos substituìdos

Info

Publication number
BR9911574A
BR9911574A BR9911574-3A BR9911574A BR9911574A BR 9911574 A BR9911574 A BR 9911574A BR 9911574 A BR9911574 A BR 9911574A BR 9911574 A BR9911574 A BR 9911574A
Authority
BR
Brazil
Prior art keywords
cyclooctadepsipeptides
replaced
substituted
cycleoctocopsype
formula
Prior art date
Application number
BR9911574-3A
Other languages
English (en)
Inventor
Juergen Scherkenbeck
Hubert Dyker
Andrew Plant
Achim Harder
Georg Von Samson Himmelstjerna
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of BR9911574A publication Critical patent/BR9911574A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K11/00Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K11/02Depsipeptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof cyclic, e.g. valinomycins ; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Veterinary Medicine (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Hydrogenated Pyridines (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Patente de Invenção: <B>''CICLOOCTADEPSIPEPTìDEOS SUBSTITUìDOS''<D>. A invenção refere-se a novos ciclooctadepsipeptídeos substituídos da fórmula (I), na qual R¹, R², m, n têm o significado indicado na descrição, processo para sua preparação, e seu emprego para o combate de endoparasitas, e agentes contendo essas substâncias ativas.
BR9911574-3A 1998-06-24 1999-06-11 Ciclooctadepsipeptìdeos substituìdos BR9911574A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19828047A DE19828047A1 (de) 1998-06-24 1998-06-24 Substituierte Cyclooctadepsipeptide
PCT/EP1999/004028 WO1999067281A1 (de) 1998-06-24 1999-06-11 Substituierte cyclooctadepsipeptide

Publications (1)

Publication Number Publication Date
BR9911574A true BR9911574A (pt) 2001-03-20

Family

ID=7871814

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9911574-3A BR9911574A (pt) 1998-06-24 1999-06-11 Ciclooctadepsipeptìdeos substituìdos

Country Status (11)

Country Link
EP (1) EP1090031A1 (pt)
JP (1) JP2002518520A (pt)
KR (1) KR20010043957A (pt)
CN (1) CN1307586A (pt)
AU (1) AU4511499A (pt)
BR (1) BR9911574A (pt)
CA (1) CA2332122A1 (pt)
DE (1) DE19828047A1 (pt)
HU (1) HUP0102476A3 (pt)
PL (1) PL345866A1 (pt)
WO (1) WO1999067281A1 (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE102008030764A1 (de) 2008-06-28 2009-12-31 Bayer Animal Health Gmbh Kombination von Amidin-Derivaten mit cyclischen Depsipeptiden
DE102008031284A1 (de) * 2008-07-02 2010-01-07 Bayer Schering Pharma Aktiengesellschaft Neue Bekämpfungsmöglichkeit der Giardiose
DE102009012423A1 (de) 2009-03-10 2010-09-16 Bayer Animal Health Gmbh Zubereitung auf Ölbasis
DE102010064245A1 (de) 2010-12-28 2012-06-28 Bayer Animal Health Gmbh Makrocylischen Lactone und deren Verwendung und deren Kombinationen mit anderen Wirkstoffen
WO2012028556A1 (en) 2010-08-31 2012-03-08 Bayer Animal Health Gmbh Macrocyclic lactones and their use and their combinations with other active substances

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0685469A4 (en) * 1993-02-19 1996-04-03 Meiji Seika Kaisha DERIVATIVE OF PF 1022 USED AS A CYCLIC DEPSIPEPTIDE.
DE4317457A1 (de) * 1993-05-26 1994-12-01 Bayer Ag Octacyclodepsipeptide mit endoparasitizider Wirkung
DE19713626A1 (de) * 1997-04-02 1998-10-08 Bayer Ag Neue Thiodepsipeptide zur Bekämpfung von Endoparasiten und ein einfaches Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
AU4511499A (en) 2000-01-10
HUP0102476A3 (en) 2003-08-28
CN1307586A (zh) 2001-08-08
PL345866A1 (en) 2002-01-14
DE19828047A1 (de) 1999-12-30
KR20010043957A (ko) 2001-05-25
EP1090031A1 (de) 2001-04-11
HUP0102476A2 (hu) 2001-10-28
CA2332122A1 (en) 1999-12-29
WO1999067281A1 (de) 1999-12-29
JP2002518520A (ja) 2002-06-25

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 5,6,7 E 8A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1911 DE 21/08/2007.