BR9703384A - Análogos de vitamina d3 - Google Patents
Análogos de vitamina d3Info
- Publication number
- BR9703384A BR9703384A BR9703384A BR9703384A BR9703384A BR 9703384 A BR9703384 A BR 9703384A BR 9703384 A BR9703384 A BR 9703384A BR 9703384 A BR9703384 A BR 9703384A BR 9703384 A BR9703384 A BR 9703384A
- Authority
- BR
- Brazil
- Prior art keywords
- analogues
- vitamin
- Prior art date
Links
- QYSXJUFSXHHAJI-YRZJJWOYSA-N vitamin D3 Chemical class C1(/[C@@H]2CC[C@@H]([C@]2(CCC1)C)[C@H](C)CCCC(C)C)=C\C=C1\C[C@@H](O)CCC1=C QYSXJUFSXHHAJI-YRZJJWOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C401/00—Irradiation products of cholesterol or its derivatives; Vitamin D derivatives, 9,10-seco cyclopenta[a]phenanthrene or analogues obtained by chemical preparation without irradiation
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/02—Nutrients, e.g. vitamins, minerals
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Nutrition Science (AREA)
- Diabetes (AREA)
- Obesity (AREA)
- Hematology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US1818696P | 1996-05-23 | 1996-05-23 | |
| US1815396P | 1996-05-23 | 1996-05-23 | |
| US3990097P | 1997-03-19 | 1997-03-19 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9703384A true BR9703384A (pt) | 1998-09-15 |
Family
ID=27360973
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9703384A BR9703384A (pt) | 1996-05-23 | 1997-05-23 | Análogos de vitamina d3 |
Country Status (29)
| Country | Link |
|---|---|
| EP (2) | EP1464640A3 (pt) |
| JP (1) | JP2859247B2 (pt) |
| KR (1) | KR100783856B1 (pt) |
| CN (1) | CN1176072C (pt) |
| AR (1) | AR007241A1 (pt) |
| AT (1) | ATE277008T1 (pt) |
| AU (1) | AU723929B2 (pt) |
| BR (1) | BR9703384A (pt) |
| CA (1) | CA2205275C (pt) |
| CO (1) | CO4950531A1 (pt) |
| CZ (1) | CZ157897A3 (pt) |
| DE (1) | DE69730774T2 (pt) |
| DK (1) | DK0808833T3 (pt) |
| ES (1) | ES2227635T3 (pt) |
| HR (1) | HRP970273A2 (pt) |
| HU (1) | HUP9700926A3 (pt) |
| IL (1) | IL120843A0 (pt) |
| MA (1) | MA24251A1 (pt) |
| NO (1) | NO972304L (pt) |
| NZ (1) | NZ314839A (pt) |
| PE (1) | PE70198A1 (pt) |
| PL (1) | PL320132A1 (pt) |
| PT (1) | PT808833E (pt) |
| SG (1) | SG70009A1 (pt) |
| TR (1) | TR199700415A2 (pt) |
| TW (1) | TW445252B (pt) |
| UY (1) | UY24561A1 (pt) |
| YU (1) | YU20197A (pt) |
| ZA (1) | ZA974336B (pt) |
Families Citing this family (26)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5939408A (en) | 1996-05-23 | 1999-08-17 | Hoffman-La Roche Inc. | Vitamin D3 analogs |
| CN100360121C (zh) * | 1997-02-25 | 2008-01-09 | 密执安州立大学董事会 | 防护和处理人皮肤经时性衰老的方法和组合物 |
| AU743514B2 (en) * | 1997-05-16 | 2002-01-24 | Women & Infants Hospital | Cyclic ether vitamin D3 compounds, 1alpha (OH) 3-EPI-vitamin D3 compounds and uses thereof |
| DE69834109T2 (de) * | 1997-05-16 | 2007-04-19 | Woman & Infants Hospital | 3-epi-vitamin d2 verbindungen und ihre anwendungen |
| EP0957098A1 (en) * | 1998-05-14 | 1999-11-17 | F. Hoffmann-La Roche Ag | Intermediates for the synthesis of 3-epi vitamin D3 metabolites and analogs |
| US6603030B1 (en) * | 1999-04-22 | 2003-08-05 | Hoffman-La Roche Inc. | Process for producing phosphineoxide vitamin D precursors |
| SK287653B6 (sk) * | 1999-04-23 | 2011-05-06 | Leo Pharmaceutical Products Ltd. A/S (Lovens Kemiske Fabrik | Nevodná farmaceutická kompozícia na dermálne použitie |
| US6255501B1 (en) | 1999-04-26 | 2001-07-03 | Hoffman-La Roche Inc. | Process for preparing antiosteoporotic agents |
| AU2058701A (en) * | 1999-12-02 | 2001-06-12 | F. Hoffmann-La Roche Ag | Esters of vitamin D3 and uses thereof |
| SG110107A1 (en) | 2003-09-24 | 2005-04-28 | Bioxell Spa | Compound and use in treatment |
| GB2407499B (en) * | 2003-11-03 | 2008-02-27 | Bioxell Spa | Vitamin D3 analogue for use in the treatment of BPH |
| CH698144B1 (fr) * | 2003-09-24 | 2009-05-29 | Bioxell Spa | Analogue de la vitamine D3 |
| CA2557809A1 (en) | 2004-03-01 | 2005-09-09 | Bioxell Spa | Treatment of interstitial cystitis with vitamin d compounds |
| JP2008519808A (ja) | 2004-11-12 | 2008-06-12 | ビオエクセル エスピーエー | 膀胱癌治療のためのビタミンd誘導体及び抗増殖薬の併用 |
| US8906888B2 (en) * | 2005-04-25 | 2014-12-09 | Cytochroma Inc. | Low-calcemic 16,23-diene 25-oxime analogs of 1α,25-dihydroxy vitamin D3 |
| AU2006279331A1 (en) * | 2005-08-18 | 2007-02-22 | Bioxell S.P.A. | Synthesis of 1alpha-fluoro-25-hydroxy-16-23e-diene-26,27-bishomo-20-epi-cholecalciferol |
| TW200838544A (en) * | 2007-01-25 | 2008-10-01 | Bioxell Spa | Synthesis of 1 α-fluoro-25-hydroxy-16-23E-diene-26, 27-bishomo-20-epi-cholecalciferol |
| ES2544819T3 (es) | 2007-05-30 | 2015-09-04 | Opko IP Holdings II, Inc. | Proceso para la producción de precursores de la vitamina D de óxido de fosfina |
| ES2366077B2 (es) * | 2010-03-30 | 2012-06-25 | Universidade De Vigo | Compuestos quirales, procedimientos de obtención y uso. |
| DK2634171T3 (en) * | 2010-10-25 | 2015-07-13 | Teijin Pharma Ltd | 23-yne-vitamin D 3 DERIVATIVE |
| JP2016503613A (ja) * | 2012-11-07 | 2016-02-04 | ヴィド スケール インコーポレイテッド | 高ダイナミックレンジビデオをノイズ除去するための時間フィルタ |
| CN105348164B (zh) * | 2015-10-29 | 2017-03-29 | 无锡福祈制药有限公司 | 一种1α‑羟基维生素D2的制备方法 |
| CN106748942B (zh) * | 2016-11-28 | 2018-06-29 | 无锡福祈制药有限公司 | 度骨化醇类似物wxfq-65及其合成方法 |
| ES2731558B2 (es) * | 2018-05-15 | 2020-03-18 | Univ Santiago Compostela | Compuestos de interés farmacéutico |
| CN109738252B (zh) * | 2019-01-23 | 2021-03-09 | 深圳天辰医疗科技有限公司 | 25-羟基-维生素d解离液 |
| CN109696435B (zh) * | 2019-01-25 | 2021-03-09 | 深圳天辰医疗科技有限公司 | 维生素d的测定方法 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ZA8923B (en) * | 1988-01-20 | 1989-09-27 | Hoffmann La Roche | 16-dehydro-vitamin d3-derivatives |
| GB8914963D0 (en) * | 1989-06-29 | 1989-08-23 | Leo Pharm Prod Ltd | Chemical compounds |
| GB9017890D0 (en) * | 1990-08-15 | 1990-09-26 | Leo Pharm Prod Ltd | Chemical compounds i |
| GB9206648D0 (en) * | 1992-03-26 | 1992-05-06 | Leo Pharm Prod Ltd | Chemical compounds |
| DK0580968T3 (da) * | 1992-05-20 | 1996-10-14 | Hoffmann La Roche | Fluorerede analoger af vitamin D3 |
| US5428029A (en) * | 1993-11-24 | 1995-06-27 | Hoffmann-La Roche Inc. | Vitamin D3 fluorinated analogs |
| JP3228488B2 (ja) * | 1993-12-24 | 2001-11-12 | 株式会社クラレ | 20−エピステロイド誘導体およびその製造方法 |
-
1997
- 1997-05-09 SG SG1997001439A patent/SG70009A1/en unknown
- 1997-05-13 CA CA002205275A patent/CA2205275C/en not_active Expired - Fee Related
- 1997-05-16 IL IL12084397A patent/IL120843A0/xx unknown
- 1997-05-16 NZ NZ314839A patent/NZ314839A/xx unknown
- 1997-05-19 ZA ZA9704336A patent/ZA974336B/xx unknown
- 1997-05-20 DE DE69730774T patent/DE69730774T2/de not_active Expired - Lifetime
- 1997-05-20 PT PT97108134T patent/PT808833E/pt unknown
- 1997-05-20 EP EP04014488A patent/EP1464640A3/en not_active Withdrawn
- 1997-05-20 PE PE1997000398A patent/PE70198A1/es not_active Application Discontinuation
- 1997-05-20 HR HR60/039,900A patent/HRP970273A2/xx not_active Application Discontinuation
- 1997-05-20 ES ES97108134T patent/ES2227635T3/es not_active Expired - Lifetime
- 1997-05-20 EP EP97108134A patent/EP0808833B1/en not_active Expired - Lifetime
- 1997-05-20 DK DK97108134T patent/DK0808833T3/da active
- 1997-05-20 TW TW086106731A patent/TW445252B/zh not_active IP Right Cessation
- 1997-05-20 YU YU20197A patent/YU20197A/sh unknown
- 1997-05-20 AT AT97108134T patent/ATE277008T1/de not_active IP Right Cessation
- 1997-05-21 HU HU9700926A patent/HUP9700926A3/hu unknown
- 1997-05-21 NO NO972304A patent/NO972304L/no not_active Application Discontinuation
- 1997-05-21 AR ARP970102158A patent/AR007241A1/es unknown
- 1997-05-22 UY UY24561A patent/UY24561A1/es unknown
- 1997-05-22 CZ CZ971578A patent/CZ157897A3/cs unknown
- 1997-05-22 CN CNB971134316A patent/CN1176072C/zh not_active Expired - Fee Related
- 1997-05-22 AU AU23577/97A patent/AU723929B2/en not_active Ceased
- 1997-05-22 CO CO97028098A patent/CO4950531A1/es unknown
- 1997-05-22 PL PL97320132A patent/PL320132A1/xx unknown
- 1997-05-22 KR KR1019970020030A patent/KR100783856B1/ko not_active Expired - Fee Related
- 1997-05-22 JP JP9131794A patent/JP2859247B2/ja not_active Expired - Fee Related
- 1997-05-22 MA MA24635A patent/MA24251A1/fr unknown
- 1997-05-23 BR BR9703384A patent/BR9703384A/pt not_active Application Discontinuation
- 1997-05-23 TR TR97/00415A patent/TR199700415A2/xx unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB34 | Technical and formal requirements: requirement - article 34 of industrial property law | ||
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: INDEFERIMENTO DO PRESENTE PEDIDO, TENDO EM VISTA O DESACORDO COM OS ARTS. 8O, 11, 13, 24 E 25 DA LPI 9279/96 |
|
| B12B | Appeal against refusal [chapter 12.2 patent gazette] |