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BR9612750A - Preparado para o transporte de substância ativa através de barreiras - Google Patents

Preparado para o transporte de substância ativa através de barreiras

Info

Publication number
BR9612750A
BR9612750A BR9612750-3A BR9612750A BR9612750A BR 9612750 A BR9612750 A BR 9612750A BR 9612750 A BR9612750 A BR 9612750A BR 9612750 A BR9612750 A BR 9612750A
Authority
BR
Brazil
Prior art keywords
active substance
prepared
barriers
preparation
transport
Prior art date
Application number
BR9612750-3A
Other languages
English (en)
Inventor
Gregor Cevc
Original Assignee
Idea Innovat Dermale Appl Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27179110&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=BR9612750(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Idea Innovat Dermale Appl Gmbh filed Critical Idea Innovat Dermale Appl Gmbh
Priority to BR9612750-3A priority Critical patent/BR9612750A/pt
Publication of BR9612750A publication Critical patent/BR9612750A/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • A61K9/1271Non-conventional liposomes, e.g. PEGylated liposomes or liposomes coated or grafted with polymers
    • A61K9/1272Non-conventional liposomes, e.g. PEGylated liposomes or liposomes coated or grafted with polymers comprising non-phosphatidyl surfactants as bilayer-forming substances, e.g. cationic lipids or non-phosphatidyl liposomes coated or grafted with polymers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/10Dispersions; Emulsions
    • A61K9/127Synthetic bilayered vehicles, e.g. liposomes or liposomes with cholesterol as the only non-phosphatidyl surfactant
    • A61K9/1271Non-conventional liposomes, e.g. PEGylated liposomes or liposomes coated or grafted with polymers

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Dispersion Chemistry (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Patente de Invenção: <B>"PREPARADO PARA O TRANSPORTE DE SUBSTâNCIA ATIVA ATRAVéS DE BARREIRAS"<D>. Preparado para a plicação da substância ativa na forma das menores gotículas, especialmente com um invólucro membranoso de uma ou de menos camadas de moléculas anfifílicas ou com gotículas de líquido providas de uma substância de veículo anfifílica, especialmente para o transporte da substância ativa para e através de barreiras naturais e constrições, como peles e similares. O preparado não apresenta nenhum ponto de solubilização ou a composição do preparado é largamente afastada do ponto de solubilização com capacidade máxima de permeação. O preparado apresenta um teor de pelo menos dois componentes, que se diferenciam em sua solubilidade no meio de suspensão dos preparados, usualmente água, em pelo menos o fator 10.
BR9612750-3A 1994-12-30 1996-10-17 Preparado para o transporte de substância ativa através de barreiras BR9612750A (pt)

Priority Applications (1)

Application Number Priority Date Filing Date Title
BR9612750-3A BR9612750A (pt) 1994-12-30 1996-10-17 Preparado para o transporte de substância ativa através de barreiras

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE4447287A DE4447287C1 (de) 1994-12-30 1994-12-30 Präparat zum Wirkstofftransport durch Barrieren
PCT/EP1996/004526 WO1998017255A1 (de) 1994-12-30 1996-10-17 Präparat zum wirkstofftransport durch barrieren
BR9612750-3A BR9612750A (pt) 1994-12-30 1996-10-17 Preparado para o transporte de substância ativa através de barreiras
CNB961804734A CN1151777C (zh) 1994-12-30 1996-10-17 转运活性成分通过屏障的制剂

Publications (1)

Publication Number Publication Date
BR9612750A true BR9612750A (pt) 1999-12-28

Family

ID=27179110

Family Applications (1)

Application Number Title Priority Date Filing Date
BR9612750-3A BR9612750A (pt) 1994-12-30 1996-10-17 Preparado para o transporte de substância ativa através de barreiras

Country Status (13)

Country Link
EP (1) EP0935457B1 (pt)
JP (1) JP2001502676A (pt)
KR (1) KR100446832B1 (pt)
CN (1) CN1151777C (pt)
AT (1) ATE257373T1 (pt)
AU (1) AU724218B2 (pt)
BR (1) BR9612750A (pt)
CA (1) CA2268670A1 (pt)
DE (2) DE4447287C1 (pt)
ES (1) ES2211984T3 (pt)
HU (1) HUP9903363A3 (pt)
MX (1) MXPA97007996A (pt)
WO (1) WO1998017255A1 (pt)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE4447287C1 (de) * 1994-12-30 1996-11-07 Cevc Gregor Präparat zum Wirkstofftransport durch Barrieren
JP4838936B2 (ja) * 1998-10-23 2011-12-14 イデア アクチェンゲゼルシャフト 装荷量を改善しおよび脱/会合速度を制御可能とするための、巨大分子と複合凝集体との会合体を開発し、テストし、かつ利用する方法
AU1327000A (en) * 1998-10-28 2000-05-15 Invitrogen Corporation Compositions comprising plant cell growth regulating compounds and methods of use thereof
HRP20010309B1 (en) * 1998-12-23 2005-06-30 Idea Ag Improved formulation for topical non-invasive application in vivo
EP1031347B1 (en) * 1999-01-27 2002-04-17 Idea Ag Transnasal transport/immunisation with highly adaptable carriers
PT1031346E (pt) 1999-01-27 2002-09-30 Idea Ag Vacinacao nao invasiva atraves da pele
MXPA02000053A (es) * 1999-07-05 2003-07-21 Idea Ag Un metodo para mejorar el tratamiento a traves de barreras adaptables semipermeables.
WO2001041738A2 (en) * 1999-12-10 2001-06-14 Celator Technologies Inc. Lipid carrier compositions with protected surface reactive functions
US20040105881A1 (en) 2002-10-11 2004-06-03 Gregor Cevc Aggregates with increased deformability, comprising at least three amphipats, for improved transport through semi-permeable barriers and for the non-invasive drug application in vivo, especially through the skin
PT1551370E (pt) * 2002-10-11 2008-02-07 Idea Ag Agregado com capacidade de deformação aumentada, que compreende pelo menos três anfipáticos, para o transporte melhorado através de barreiras semi-permeáveis e para a aplicação de fármaco não invasiva in vivo, especialmente através da pele
EP1585548B1 (en) * 2002-12-09 2018-06-27 Abraxis BioScience, LLC Compositions and methods of delivery of pharmacological agents
DE102008034098A1 (de) 2008-07-21 2010-02-04 Lts Lohmann Therapie-Systeme Ag Zubereitung und lontophoretische Vorrichtung für die transdermale Anwendung von Wirkstoffen
CN105434353A (zh) 2009-06-03 2016-03-30 斯昆申技术控股有限责任公司 用于治疗深部组织疼痛的制剂
DE112010003355T5 (de) 2009-08-21 2012-07-12 Targeted Delivery Technologies Ltd. Veskuläre Formulierungen
WO2013057208A1 (en) 2011-10-18 2013-04-25 Targeted Delivery Technologies Limited Compositions and methods for reducing the proliferation and viability of microbial agents
CN102579350B (zh) * 2012-03-02 2013-04-24 海南灵康制药有限公司 右旋布洛芬脂质体固体制剂
GB201205642D0 (en) 2012-03-29 2012-05-16 Sequessome Technology Holdings Ltd Vesicular formulations
PT3316857T (pt) 2015-06-30 2021-11-03 Sequessome Tech Holdings Limited Composições multifásicas
CH713023A2 (de) * 2016-10-11 2018-04-13 Kuhs Bernd Verfahren zur Herstellung von dermatologischen und kosmetischen Präparaten mit ausgeprägten lamellaren Strukturen unter Verwendung von Phosphatidylcholin und biologischen Zellmaterialien, welche durch die Einwirkung von Ultraschallwellen aufgeschlossen werden und gleichzeitig zwischen den lamellaren Strukturen eingelagert werden.
WO2019023247A1 (en) 2017-07-25 2019-01-31 Immutics, Inc. TREATMENT OF CANCER BY BLOCKING THE INTERACTION OF TIM-3 AND ITS LIGAND
CN116063505B (zh) 2019-01-30 2024-05-03 真和制药有限公司 抗gal3抗体及其用途
CN110101591B (zh) * 2019-05-23 2022-01-18 广州科斯曼生物科技有限公司 一种长效保湿组合物及其制备方法和应用
EP4157338A4 (en) 2020-05-26 2024-11-13 TrueBinding, Inc. METHOD FOR TREATING INFLAMMATORY DISEASES BY GALECTIN-3 BLOCKING

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4921706A (en) * 1984-11-20 1990-05-01 Massachusetts Institute Of Technology Unilamellar lipid vesicles and method for their formation
DE3542773A1 (de) * 1985-12-04 1987-06-11 Roehm Pharma Gmbh Hautwirksame pharmaka mit liposomen als wirkstofftraeger
US5064655A (en) * 1989-02-24 1991-11-12 Liposome Technology, Inc. Liposome gel composition and method
FR2649155B1 (fr) * 1989-06-28 1991-09-13 Elf Aquitaine Dispositif de mesure dynamometrique pour tige de forage
JP2844756B2 (ja) * 1989-12-01 1999-01-06 日本新薬株式会社 脂肪乳剤
WO1992003122A1 (de) * 1990-08-24 1992-03-05 Gregor Cevc Präparat zur wirkstoffapplikation in kleinsttröpfchenform
SE9003100D0 (sv) * 1990-09-28 1990-09-28 Kabivitrum Ab Lipid formulation system
SE9200952D0 (sv) * 1992-03-27 1992-03-27 Kabi Pharmacia Ab Pharmaceutical carrier system containing defined lipids
SE9200951D0 (sv) * 1992-03-27 1992-03-27 Kabi Pharmacia Ab Pharmaceutical composition containing a defined lipid system
FR2714601B1 (fr) * 1993-12-30 1996-02-09 Oreal Composition dépigmentante pour le traitement simultané des couches superficielles et profondes, son utilisation.
JPH0881360A (ja) * 1994-07-13 1996-03-26 Wakamoto Pharmaceut Co Ltd 安定な脂肪乳剤
ATE223202T1 (de) * 1994-09-30 2002-09-15 Mika Pharma Ges Fuer Die Entwi Pharmazeutische zusammensetzung
IT1270678B (it) * 1994-10-20 1997-05-07 Bayer Ag Liposomi al chetoprofen
DE4447287C1 (de) * 1994-12-30 1996-11-07 Cevc Gregor Präparat zum Wirkstofftransport durch Barrieren

Also Published As

Publication number Publication date
KR100446832B1 (ko) 2004-09-04
CN1151777C (zh) 2004-06-02
AU724218B2 (en) 2000-09-14
HUP9903363A3 (en) 2008-04-28
DE59610889D1 (de) 2004-02-12
AU4510897A (en) 1998-05-15
ES2211984T3 (es) 2004-07-16
JP2001502676A (ja) 2001-02-27
DE4447287C1 (de) 1996-11-07
ATE257373T1 (de) 2004-01-15
CN1234736A (zh) 1999-11-10
HK1021622A1 (en) 2000-06-23
WO1998017255A1 (de) 1998-04-30
MXPA97007996A (es) 2004-03-15
CA2268670A1 (en) 1998-04-30
KR20000049266A (ko) 2000-07-25
EP0935457B1 (de) 2004-01-07
HUP9903363A2 (hu) 2000-03-28
EP0935457A1 (de) 1999-08-18

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Legal Events

Date Code Title Description
B25D Requested change of name of applicant approved
B07A Application suspended after technical examination (opinion) [chapter 7.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B06A Patent application procedure suspended [chapter 6.1 patent gazette]
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE AS 14A E 15A ANUIDADES.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: NAO APRESENTADA A GUIA DE CUMPRIMENTO DE EXIGENCIA. REFERENTE AS 14A E 15A ANUIDADES.