BR9612000A - Naphthyl glyoxamides as spla inhibitors; ' - Google Patents
Naphthyl glyoxamides as spla inhibitors; 'Info
- Publication number
- BR9612000A BR9612000A BR9612000-2A BR9612000A BR9612000A BR 9612000 A BR9612000 A BR 9612000A BR 9612000 A BR9612000 A BR 9612000A BR 9612000 A BR9612000 A BR 9612000A
- Authority
- BR
- Brazil
- Prior art keywords
- spla
- inhibitors
- compounds
- glyoxamides
- naphthyl
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title abstract 2
- 125000001624 naphthyl group Chemical group 0.000 title 1
- -1 naphthyl glyoxamide compounds Chemical class 0.000 abstract 2
- 206010040070 Septic Shock Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 235000014113 dietary fatty acids Nutrition 0.000 abstract 1
- 229930195729 fatty acid Natural products 0.000 abstract 1
- 239000000194 fatty acid Substances 0.000 abstract 1
- 150000004665 fatty acids Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 230000036303 septic shock Effects 0.000 abstract 1
Landscapes
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Patente de Invenção: <B>"NAFTIL GLIOXAMIDAS COMO INIBIDORES DE sPLA~ 2~"<D>. Uma classe de novos compostos de glioxamida naftil é divulgado juntamente com o processo de fabricação de novos compostos de glioxamidas de naftil e o uso de tais compostos para inibição da liberação de ácidos graxos mediada pelo sPLA~ 2~, para o tratamento de condições tal como o choque séptico.Invention Patent: <B> "NAFTYL GLIOXAMIDES AS INHIBITORS OF sPLA ~ 2 ~" <D>. A class of new naphthyl glyoxamide compounds is disclosed along with the manufacturing process of new naphthyl glyoxamide compounds and the use of such compounds to inhibit sPLA ~ 2 ~ -mediated fatty acid release for the treatment of conditions such as septic shock.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US855795P | 1995-12-13 | 1995-12-13 | |
| PCT/US1996/019529 WO1997021716A1 (en) | 1995-12-13 | 1996-12-09 | NAPHTHYL GLYOXAMIDES AS sPLA2 INHIBITORS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9612000A true BR9612000A (en) | 2000-03-28 |
Family
ID=21732283
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9612000-2A BR9612000A (en) | 1995-12-13 | 1996-12-09 | Naphthyl glyoxamides as spla inhibitors; ' |
Country Status (1)
| Country | Link |
|---|---|
| BR (1) | BR9612000A (en) |
-
1996
- 1996-12-09 BR BR9612000-2A patent/BR9612000A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FB36 | Technical and formal requirements: requirement - article 36 of industrial property law | ||
| B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements | ||
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |