BR9603432A - Antagonistas de receptores de endotelina - Google Patents

Antagonistas de receptores de endotelina

Info

Publication number: BR9603432A
Authority: BR; Brazil
Prior art keywords: receptor antagonists; endothelin receptor; endothelin; antagonists; receptor
Prior art date: 1995-08-16

Application number

BR9603432A

Other languages

English (en)

Inventor

Dieter Dr Dorsch

Mathias Dr Oswald

Werner Dr Mederski

Claudia Dr Wilm

Claus Dr Schmitges

Maria Christadler

Original Assignee

Merck Patent Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1995-08-16

Filing date

1996-08-15

Publication date

1998-05-12

1996-08-15 Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh

1998-05-12 Publication of BR9603432A publication Critical patent/BR9603432A/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
- C07D307/77—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
- C07D307/78—Benzo [b] furans; Hydrogenated benzo [b] furans
- C07D307/79—Benzo [b] furans; Hydrogenated benzo [b] furans with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
- A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Pain & Pain Management (AREA)
Vascular Medicine (AREA)
Rheumatology (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pulmonology (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Compounds That Contain Two Or More Ring Oxygen Atoms (AREA)
Plural Heterocyclic Compounds (AREA)

BR9603432A 1995-08-16 1996-08-15 Antagonistas de receptores de endotelina BR9603432A (pt)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19530032A DE19530032A1 (de)	1995-08-16	1995-08-16	Endothelin-Rezeptor-Antagonisten

Publications (1)

Publication Number	Publication Date
BR9603432A true BR9603432A (pt)	1998-05-12

Family

ID=7769557

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BR9603432A BR9603432A (pt)	1995-08-16	1996-08-15	Antagonistas de receptores de endotelina

Country Status (17)

Country	Link
US (1)	US5821256A (pt)
EP (1)	EP0758650A1 (pt)
JP (1)	JPH0959273A (pt)
KR (1)	KR970010756A (pt)
CN (1)	CN1149583A (pt)
AR (1)	AR003286A1 (pt)
AU (1)	AU6200296A (pt)
BR (1)	BR9603432A (pt)
CA (1)	CA2183307A1 (pt)
CZ (1)	CZ240096A3 (pt)
DE (1)	DE19530032A1 (pt)
HU (1)	HUP9602253A3 (pt)
MX (1)	MX9603343A (pt)
NO (1)	NO963411L (pt)
PL (1)	PL315707A1 (pt)
SK (1)	SK100096A3 (pt)
ZA (1)	ZA966933B (pt)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9602029D0 (en) *	1996-02-01	1996-04-03	Fujisawa Pharmaceutical Co	New heterocyclic compounds
DE19710831A1 (de) *	1997-03-15	1998-09-17	Merck Patent Gmbh	Endothelin-Rezeptor-Antagonisten
AU2002251978B2 (en) *	2001-02-09	2007-07-19	Merck & Co., Inc.	2-aryloxy-2-arylalkanoic acids for diabetes and lipid disorders
DE10155076A1 (de) *	2001-11-09	2003-05-22	Merck Patent Gmbh	Verwendung von Endothelin-Rezeptor-Antagonisten zur Behandlung von Tumorerkrankungen
EP1926989A4 (en) *	2005-08-12	2008-12-24	Uop Llc	METHOD AND DEVICE FOR ACCELERATING SAMPLE ANALYSIS

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH07110833B2 (ja) *	1986-12-02	1995-11-29	株式会社トクヤマ	α−置換フエニル酢酸誘導体
RU2086544C1 (ru) *	1991-06-13	1997-08-10	Хоффманн-Ля Рош АГ	Бензолсульфонамидные производные пиримидина или их соли, фармацевтическая композиция для лечения заболеваний, связанных с активностью эндотелина
GB9115153D0 (en) *	1991-07-12	1991-08-28	Patel Bipin C M	Sol-gel composition for producing glassy coatings
DE69232072T2 (de) *	1991-11-05	2002-06-20	Smithkline Beecham Corp., Philadelphia	Endothelin-rezeptor-antagonisten
ZA939516B (en) *	1992-12-22	1994-06-06	Smithkline Beecham Corp	Endothelin receptor antagonists
DK0617001T3 (da) *	1993-03-19	2000-04-17	Merck & Co Inc	Phenoxyphenyleddikesyrederivater
AU3642795A (en) *	1994-09-27	1996-04-19	Merck & Co., Inc.	Endothelin receptor antagonists for the treatment of emesis

1995
- 1995-08-16 DE DE19530032A patent/DE19530032A1/de not_active Withdrawn
1996
- 1996-07-31 SK SK1000-96A patent/SK100096A3/sk unknown
- 1996-08-06 EP EP96112667A patent/EP0758650A1/de not_active Withdrawn
- 1996-08-09 AU AU62002/96A patent/AU6200296A/en not_active Abandoned
- 1996-08-13 MX MX9603343A patent/MX9603343A/es unknown
- 1996-08-14 CZ CZ962400A patent/CZ240096A3/cs unknown
- 1996-08-14 CN CN96111668A patent/CN1149583A/zh active Pending
- 1996-08-14 KR KR1019960033775A patent/KR970010756A/ko not_active Withdrawn
- 1996-08-14 CA CA002183307A patent/CA2183307A1/en not_active Abandoned
- 1996-08-14 PL PL96315707A patent/PL315707A1/xx unknown
- 1996-08-15 NO NO963411A patent/NO963411L/no unknown
- 1996-08-15 BR BR9603432A patent/BR9603432A/pt not_active Application Discontinuation
- 1996-08-15 ZA ZA9606933A patent/ZA966933B/xx unknown
- 1996-08-15 US US08/698,331 patent/US5821256A/en not_active Expired - Fee Related
- 1996-08-15 HU HU9602253A patent/HUP9602253A3/hu unknown
- 1996-08-16 JP JP8233711A patent/JPH0959273A/ja active Pending
- 1996-08-16 AR ARP960104020A patent/AR003286A1/es unknown

Also Published As

Publication number	Publication date
HU9602253D0 (en)	1996-10-28
CN1149583A (zh)	1997-05-14
DE19530032A1 (de)	1997-02-20
ZA966933B (en)	1997-02-19
US5821256A (en)	1998-10-13
JPH0959273A (ja)	1997-03-04
AR003286A1 (es)	1998-07-08
EP0758650A1 (de)	1997-02-19
HUP9602253A3 (en)	1999-06-28
AU6200296A (en)	1997-02-20
MX9603343A (es)	1997-03-29
NO963411L (no)	1997-02-17
NO963411D0 (no)	1996-08-15
SK100096A3 (en)	1997-03-05
CA2183307A1 (en)	1997-02-17
CZ240096A3 (en)	1997-03-12
HUP9602253A2 (en)	1997-12-29
KR970010756A (ko)	1997-03-27
PL315707A1 (en)	1997-02-17

Publication	Publication Date	Title
FI960953A0 (fi)	1996-02-29	Endoteliinireseptoriantagonisteja
BR9407933A (pt)	1996-11-26	Antagonistas de receptores de endotelina
NO972016D0 (no)	1997-04-30	Indolyl-Y-reseptorantagonister
BR9612327A (pt)	1999-07-13	Antagonistas receptores de vitronectina
BR9612378A (pt)	1999-07-13	Antagonistas receptores de vitronectina
EP0810994A4 (en)	1998-05-06	FIBRINOGEN RECEPTOR ANTAGONISTS
BR9612381A (pt)	1999-07-13	Antagonistas receptores vitronectina
DE69327720D1 (de)	2000-03-02	Endothelin rezeptor antagonisten
NO305559B1 (no)	1999-06-21	Substituerte bifenyl-sulfonamid-endotelin-antagonister
EP0866705A4 (en)	1999-03-03	FIBRINOGENIC RECEPTOR ANTAGONISTS
BR9406572A (pt)	1996-01-30	Antagonistas receptores do endotelin
DK0741133T3 (da)	2004-04-26	Adhæsionsreceptorantagonister
BR9507220A (pt)	1997-09-09	Antagonistas de receptores de endotelina
DE69636597D1 (de)	2006-11-16	Endothelin rezeptor antagonisten
NO972612D0 (no)	1997-06-06	Pyridazoner som endotelinreseptorantagonister
HU9602054D0 (en)	1996-09-30	Endothelin receptor antagonists
EP0854721A4 (en)	1998-12-02	ENDOTHELIN RECEPTOR ANTAGONISTS
EP0841926A4 (en)	1999-08-04	ENDOTHELIN RECEPTOR ANTAGONISTS
BR9603432A (pt)	1998-05-12	Antagonistas de receptores de endotelina
EP0841916A4 (en)	2001-04-11	ENDOTHELINE RECEPTOR ANTAGONISTS
EP0868180A4 (en)	1999-08-04	ENDOTHELINM RECEPTOR ANTOGONISTS
ZA966593B (en)	1997-03-24	Endothelin receptor antagonists
GB9510203D0 (en)	1995-07-12	Novel endothelin receptor antagonists

Legal Events

Date	Code	Title	Description
2001-09-18	FA10	Dismissal: dismissal - article 33 of industrial property law