BR9509888A - Composto formulação farmacéutica uso do composto e processos para a inibição de secreção de ácido gástrico para o tratamento das doenças inflamatórias gastrointestinais e para o tratamento ou profilaxia das condições envolvendo a infecção por helicobacter pylori da mucosa gástrica humana - Google Patents
Composto formulação farmacéutica uso do composto e processos para a inibição de secreção de ácido gástrico para o tratamento das doenças inflamatórias gastrointestinais e para o tratamento ou profilaxia das condições envolvendo a infecção por helicobacter pylori da mucosa gástrica humanaInfo
- Publication number
- BR9509888A BR9509888A BR9509888A BR9509888A BR9509888A BR 9509888 A BR9509888 A BR 9509888A BR 9509888 A BR9509888 A BR 9509888A BR 9509888 A BR9509888 A BR 9509888A BR 9509888 A BR9509888 A BR 9509888A
- Authority
- BR
- Brazil
- Prior art keywords
- treatment
- compound
- prophylaxis
- inhibition
- processes
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 2
- 238000011282 treatment Methods 0.000 title 2
- 208000018522 Gastrointestinal disease Diseases 0.000 title 1
- 206010019375 Helicobacter infections Diseases 0.000 title 1
- 230000027119 gastric acid secretion Effects 0.000 title 1
- 210000001156 gastric mucosa Anatomy 0.000 title 1
- 230000002757 inflammatory effect Effects 0.000 title 1
- 230000005764 inhibitory process Effects 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 238000011321 prophylaxis Methods 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/20—Oxygen atoms
- C07D215/24—Oxygen atoms attached in position 8
- C07D215/26—Alcohols; Ethers thereof
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/42—Nitrogen atoms attached in position 4
- C07D215/44—Nitrogen atoms attached in position 4 with aryl radicals attached to said nitrogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Quinoline Compounds (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US08/351,852 US5556863A (en) | 1993-06-11 | 1994-12-08 | Compound for gastric acid secretion inhibition |
| PCT/SE1995/001369 WO1996017830A1 (en) | 1994-12-08 | 1995-11-17 | Compounds for inhibition of gastric acid secretion |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9509888A true BR9509888A (pt) | 1997-10-21 |
Family
ID=23382690
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR9509888A BR9509888A (pt) | 1994-12-08 | 1995-11-17 | Composto formulação farmacéutica uso do composto e processos para a inibição de secreção de ácido gástrico para o tratamento das doenças inflamatórias gastrointestinais e para o tratamento ou profilaxia das condições envolvendo a infecção por helicobacter pylori da mucosa gástrica humana |
Country Status (20)
| Country | Link |
|---|---|
| US (1) | US5556863A (pt) |
| EP (1) | EP0796249A1 (pt) |
| JP (1) | JPH10510259A (pt) |
| CN (1) | CN1169142A (pt) |
| AR (1) | AR001996A1 (pt) |
| BR (1) | BR9509888A (pt) |
| CA (1) | CA2205896A1 (pt) |
| EE (1) | EE9700131A (pt) |
| FI (1) | FI972410L (pt) |
| HU (1) | HUT77949A (pt) |
| IL (1) | IL116285A0 (pt) |
| IS (1) | IS4485A (pt) |
| MX (1) | MX9704136A (pt) |
| NO (1) | NO972529L (pt) |
| NZ (1) | NZ297566A (pt) |
| PL (1) | PL320754A1 (pt) |
| SK (1) | SK63797A3 (pt) |
| TR (1) | TR199501536A2 (pt) |
| WO (1) | WO1996017830A1 (pt) |
| ZA (1) | ZA9510066B (pt) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| UA80393C2 (uk) | 2000-12-07 | 2007-09-25 | Алтана Фарма Аг | Фармацевтична композиція, яка містить інгібітор фде 4, диспергований в матриці |
| MY140561A (en) | 2002-02-20 | 2009-12-31 | Nycomed Gmbh | Dosage form containing pde 4 inhibitor as active ingredient |
Family Cites Families (38)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4042702A (en) * | 1973-08-16 | 1977-08-16 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Halogen pyrazole derivatives, a method for producing these halogen pyrazole derivatives, medicaments containing and methods of using them |
| LU69428A1 (pt) * | 1974-02-20 | 1975-12-09 | ||
| US4120972A (en) * | 1975-02-03 | 1978-10-17 | Smith Kline & French Laboratories Limited | Imidazolylmethylthio-ethyl isothiourea compounds |
| NO760996L (pt) * | 1975-03-25 | 1976-09-28 | Byk Gulden Lomberg Chem Fab | |
| AT364354B (de) * | 1976-10-14 | 1981-10-12 | Byk Gulden Lomberg Chem Fab | Verfahren zur herstellung von neuen pyrazol-1yl-phenylessigsaeuren, deren salzen und optischen isomeren |
| LU78804A1 (de) * | 1977-12-30 | 1979-07-20 | Byk Gulden Lomberg Chem Fab | N-substituierte w-aminoalkanoyl-w-aminoalkansaeuren,ihre verwendung und verfahren zu ihrer herstellung sowie diese verbindungen enthaltende arzneimittel |
| US4243678A (en) * | 1977-12-30 | 1981-01-06 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Acylhydrocarbylaminoalkanoic acids, compositions and uses |
| YU118379A (en) * | 1978-05-24 | 1983-02-28 | Byk Gulden Lomberg Chemischefa | Process for preparing phenylaminothiophene acetic acid |
| US4343804A (en) * | 1979-03-26 | 1982-08-10 | A. H. Robins Company, Inc. | 4-Amino-3-quinolinecarboxylic acids and esters-antisecretory anti-ulcer compounds |
| AU529934B2 (en) * | 1979-08-03 | 1983-06-23 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituted tetraazatricyclic compounds |
| EP0024638A1 (en) * | 1979-08-30 | 1981-03-11 | Byk Gulden Lomberg Chemische Fabrik GmbH | Substituted quinolinone-alkanecarboxylic acids, their preparation, and medicaments containing them |
| DE3063144D1 (en) * | 1979-09-07 | 1983-06-16 | Byk Gulden Lomberg Chem Fab | Substituted oxirane carboxylic acids, process for their preparation, their use and medicines containing them |
| ES496382A0 (es) * | 1979-10-31 | 1982-03-01 | Byk Gulden Lomberg Chem Fab | Procedimiento para la preparacion de acidos oxocarboxilicos sustituidos |
| US4381301A (en) * | 1980-05-07 | 1983-04-26 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Substituted tricyclic thieno compounds, their synthesis, their use, their compositions and their medicaments |
| US4337267A (en) * | 1980-08-25 | 1982-06-29 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Phenalkoxyalkyl- and phenoxyalkyl-substituted oxiranecarboxylic acids, their use and medicaments containing them |
| EP0046961B1 (de) * | 1980-08-29 | 1985-02-13 | Byk Gulden Lomberg Chemische Fabrik GmbH | Epoxi-cycloalkylalkancarbonsäuren, Verfahren zu ihrer Herstellung, ihre Verwendung sowie sie enthaltende Arzneimittel |
| DE3262922D1 (en) * | 1981-02-02 | 1985-05-15 | Byk Gulden Lomberg Chem Fab | Tricyclic pyrrols, process for their preparation, their use and compositions containing them |
| FI80022C (fi) * | 1982-07-05 | 1990-04-10 | Otsuka Pharma Co Ltd | Foerfarande foer framstaellning av ett nytt, terapeutiskt anvaendbart karbostyrilderivat. |
| DK585485A (da) * | 1984-12-18 | 1986-08-08 | Utsuka Pharm Co Ltd | Tetrahydroquinolinderivat, imidazopyridinderivat, fremgangsmaade til fremstilling deraf og farmaceutisk praeparat med mindst en saadan forbindelse |
| US5250527A (en) * | 1985-10-24 | 1993-10-05 | Smithkline & French Laboratories Limited | Pyridyl containing benzimidazoles, compositions and use |
| GB8621425D0 (en) * | 1986-09-05 | 1986-10-15 | Smith Kline French Lab | Compounds |
| GB8717644D0 (en) * | 1987-07-24 | 1987-09-03 | Smithkline Beckman Intercredit | Compounds |
| GB8804444D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
| GB8804443D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
| GB8804448D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
| GB8804446D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
| GB8804447D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
| US5049567A (en) * | 1988-02-25 | 1991-09-17 | Smithkline Beckman Intercredit B.V. | Substituted 4-aminoquinazoline derivatives and method of use |
| GB8804445D0 (en) * | 1988-02-25 | 1988-03-23 | Smithkline Beckman Intercredit | Compounds |
| CA2011086A1 (en) * | 1989-03-17 | 1990-09-17 | Karl-Heinz Geiss | 2-alkyl-4-arylmethylaminoquinolines, the use thereof and drugs prepared therefrom |
| GB8908229D0 (en) * | 1989-04-12 | 1989-05-24 | Smithkline Beckman Intercredit | Compounds |
| GB8910722D0 (en) * | 1989-05-10 | 1989-06-28 | Smithkline Beckman Intercredit | Compounds |
| DE3917233A1 (de) * | 1989-05-26 | 1990-11-29 | Basf Ag | 8-substituierte 4-(heterocyclylmethylamino)-chinoline, ihre verwendung und daraus hergestellte arzneimittel |
| GB8918265D0 (en) * | 1989-08-10 | 1989-09-20 | Smithkline Beckman Intercredit | Compounds |
| DK0480052T3 (da) * | 1990-03-28 | 1998-05-11 | Otsuka Pharma Co Ltd | Quinolinderivat, antiulcus-lægemiddel indeholdende derivatet og fremstilling af derivatet |
| MA22401A1 (fr) * | 1991-01-29 | 1992-10-01 | Smithkline Beecham Intercredit | Procede de preparation de sels de guinoleine |
| GB9126438D0 (en) * | 1991-12-12 | 1992-02-12 | Smithkline Beecham Intercredit | New quinoline derivatives |
| IS4164A (is) * | 1993-06-11 | 1994-12-12 | Ab Astra | Efnasambönd sem hindra flæði magasýru |
-
1994
- 1994-12-08 US US08/351,852 patent/US5556863A/en not_active Expired - Fee Related
-
1995
- 1995-11-08 AR ARP950100099A patent/AR001996A1/es unknown
- 1995-11-17 CN CN95196698A patent/CN1169142A/zh active Pending
- 1995-11-17 BR BR9509888A patent/BR9509888A/pt not_active Application Discontinuation
- 1995-11-17 PL PL95320754A patent/PL320754A1/xx unknown
- 1995-11-17 FI FI972410A patent/FI972410L/fi unknown
- 1995-11-17 CA CA002205896A patent/CA2205896A1/en not_active Abandoned
- 1995-11-17 JP JP8517523A patent/JPH10510259A/ja active Pending
- 1995-11-17 HU HU9800175A patent/HUT77949A/hu unknown
- 1995-11-17 MX MX9704136A patent/MX9704136A/es unknown
- 1995-11-17 SK SK637-97A patent/SK63797A3/sk unknown
- 1995-11-17 NZ NZ297566A patent/NZ297566A/xx unknown
- 1995-11-17 WO PCT/SE1995/001369 patent/WO1996017830A1/en not_active Ceased
- 1995-11-17 EP EP95941272A patent/EP0796249A1/en not_active Ceased
- 1995-11-17 EE EE9700131A patent/EE9700131A/xx unknown
- 1995-11-27 ZA ZA9510066A patent/ZA9510066B/xx unknown
- 1995-12-05 TR TR95/01536A patent/TR199501536A2/xx unknown
- 1995-12-07 IL IL11628595A patent/IL116285A0/xx unknown
-
1997
- 1997-05-22 IS IS4485A patent/IS4485A/is unknown
- 1997-06-03 NO NO972529A patent/NO972529L/no unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CA2205896A1 (en) | 1996-06-13 |
| IL116285A0 (en) | 1996-03-31 |
| AU697006B2 (en) | 1998-09-24 |
| AR001996A1 (es) | 1998-01-07 |
| ZA9510066B (en) | 1996-06-10 |
| FI972410A0 (fi) | 1997-06-06 |
| PL320754A1 (en) | 1997-10-27 |
| NO972529D0 (no) | 1997-06-03 |
| AU4274896A (en) | 1996-06-26 |
| EP0796249A1 (en) | 1997-09-24 |
| SK63797A3 (en) | 1998-07-08 |
| JPH10510259A (ja) | 1998-10-06 |
| HUT77949A (hu) | 1998-12-28 |
| MX9704136A (es) | 1998-02-28 |
| CN1169142A (zh) | 1997-12-31 |
| FI972410A7 (fi) | 1997-06-06 |
| NZ297566A (en) | 1998-12-23 |
| FI972410L (fi) | 1997-06-06 |
| US5556863A (en) | 1996-09-17 |
| IS4485A (is) | 1997-05-22 |
| WO1996017830A1 (en) | 1996-06-13 |
| EE9700131A (et) | 1997-12-15 |
| NO972529L (no) | 1997-06-03 |
| TR199501536A2 (tr) | 1996-07-21 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| Hawkey et al. | Prostaglandins and the gastrointestinal mucosa: are they important in its function, disease, or treatment? | |
| ITMI951359A0 (it) | Formulazioni farmaceutiche e dietetiche per la profilassi e la cura di affezioni gastrointestinali | |
| BR9607367A (pt) | Forma de múltipla dosagem unitária em tablete efervecente processos para preparação da mesma para a inibição de secreção de ácido gástrico em mamíferos e no homem e para o tratamento de doenças gastrointestinais inflamatórias em maniferos e no homem e uso da forma de dosagem em tablete efervecente | |
| FI940629A7 (fi) | Valmiste ruoansulatuskanavan sisäiseen ravitsemukseen | |
| AU1063201A (en) | Use of tgf beta and growth factors in the treatment and prevention of diseases of the intestinal mucosa | |
| ITRM920270A1 (it) | Composizione farmaceutica per il trattamento e la prevenzione delle infiammazioni cutanee e della mucosa orale. | |
| BR9814378A (pt) | Forma de dosagem de liberação prolongada farmacêutica revestida entérica de um inibidor de h+, k+-atpase, processos para a manufatura da mesma, para melhorar a inibição de secreção de ácido gástrico, para melhorar o efeito terapêutico no tratamento de distúrbios gastrointentinais, para receber um perfil de plasma prolongado de um inibidor da h+, k+-atpase, e, usos de uma composição farmacêutica e de inibidor da h+, k+-atpase | |
| CY1105834T1 (el) | Χρηση παρασκευασματων για την εφαρμογη, στον κατω αναπνευστικο σωληνα αντισηπτικων παραγοντων και/ή παραγοντων που προαγουν την επουλωση των πληγων | |
| PT1042324E (pt) | Compostos heterociclicos para inibicao da secrecaode acido gastrico processis para a sua prepara cao e suas composicoes farmaceuticas | |
| HUP0000450A2 (hu) | 7-(2-Oxa-5,8-diazabiciklo[4.3.0]non-8-il)-kinolon-karbonsav és -naftiridon-karbonsav-származékok alkalmazása Helicobacter pylori fertőzések, és az ezzel kapcsolatos gyomor-bél megbetegedések gyógyítására szolgáló gyógyszerkészítmények előállítására | |
| BR9913103A (pt) | Composto, processo para a preparação do mesmo, formulação farmacêutica, uso do composto, processos para inibir a secreção do ácido gástrico, para o tratamento de doenças inflamatórias gastrointestinal, e para o tratamento ou profilaxia de condições que envolvem a infeção por helicobacter pylori da mucosa gástrica humana, e, formulações farmacêuticas para o uso na inibição da secreção de ácido gástrico, para o uso no tratamento de doenças inflamatórias gastrointestinais, e para o uso no tratamento ou profilaxia de condições que envolvem a infecção por helicobacter pylori da mucosa gástrica humana | |
| NO973243D0 (no) | Anvendelse av 3,4-difenylkromaner til fremstilling av et farmasöytisk preparat for behandling eller profylakse av gynekologiske sykdommer | |
| BR0211846A (pt) | Composto, processo para a preparação do mesmo, formulação farmacêutica, uso de um composto, e, métodos para inibir a secreção de ácido gástrico, para tratar doenças gastrintestinais inflamatórias, e para tratar ou profilaxia de condições envolvendo infecção por helicobacter pylori de mucosa gástrica humana | |
| IL113263A0 (en) | Imidazo pyridine compounds and pharmaceutical compositions for the treatment of gastrointestinal diseases | |
| SE9201930D0 (sv) | Gastric antibacterial treatment | |
| DK0616802T3 (da) | Oralt præparat til frigivelse i de nedre fordøjelseskanaler | |
| EP0161817A3 (en) | Urogastrone | |
| BR9506235A (pt) | Compostos enanciométricos únicos uso dos mesmos processos para sua preparação e de(+)-e-(-)-5-carbometoxi-6-metail-2-((3,4-dimetoxi-2-piridinil)metil )1-h-benzimidazol ou seu sal de sódio em suas for mas cristalinas para inibição de secreção de ácido gástrico e para o tratamento de doenças inflamatórias gastrointestinais e preparação farmacêutica | |
| IL85963A0 (en) | Pharmaceutical compositions for the prophylaxis or treatment of disorders or diseases of the gastrointestinal tract,comprising antigenic substances | |
| CA2353048A1 (en) | Pharmaceutical composition useful in the prevention or treatment of peptic ulcers | |
| BR9509888A (pt) | Composto formulação farmacéutica uso do composto e processos para a inibição de secreção de ácido gástrico para o tratamento das doenças inflamatórias gastrointestinais e para o tratamento ou profilaxia das condições envolvendo a infecção por helicobacter pylori da mucosa gástrica humana | |
| KR930701166A (ko) | 5-디플루오로메톡시-2-[메틸설피닐] 벤즈이미다졸을 함유하는 약학 조성물 및 위장 질환 치료용 항헬리코박터제 | |
| AU1395583A (en) | Use of oleanolic acid for ulcer treatment | |
| ES2123004T3 (es) | Uso de factor de crecimiento derivado de plaquetas en la preparacion de un medicamento para el tratamiento de ulceras gastrointestinales. | |
| IT8219482A0 (it) | Composizione farmaceutica per la cura di affezioni della cavita'orale. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] |