BR9105371A - Formulacao apropriada para a administracao transdermica de dobutamina e processo para aumentar a contratilidade cardiaca - Google Patents
Formulacao apropriada para a administracao transdermica de dobutamina e processo para aumentar a contratilidade cardiacaInfo
- Publication number
- BR9105371A BR9105371A BR919105371A BR9105371A BR9105371A BR 9105371 A BR9105371 A BR 9105371A BR 919105371 A BR919105371 A BR 919105371A BR 9105371 A BR9105371 A BR 9105371A BR 9105371 A BR9105371 A BR 9105371A
- Authority
- BR
- Brazil
- Prior art keywords
- contratility
- dobutamine
- transdermal administration
- appropriate formulation
- increase cardiac
- Prior art date
Links
- JRWZLRBJNMZMFE-UHFFFAOYSA-N Dobutamine Chemical compound C=1C=C(O)C(O)=CC=1CCNC(C)CCC1=CC=C(O)C=C1 JRWZLRBJNMZMFE-UHFFFAOYSA-N 0.000 title 1
- 230000000747 cardiac effect Effects 0.000 title 1
- 229960001089 dobutamine Drugs 0.000 title 1
- 238000009472 formulation Methods 0.000 title 1
- 238000000034 method Methods 0.000 title 1
- 239000000203 mixture Substances 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0014—Skin, i.e. galenical aspects of topical compositions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/20—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing sulfur, e.g. dimethyl sulfoxide [DMSO], docusate, sodium lauryl sulfate or aminosulfonic acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Dermatology (AREA)
- Hospice & Palliative Care (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63048090A | 1990-12-20 | 1990-12-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR9105371A true BR9105371A (pt) | 1992-08-25 |
Family
ID=24527346
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR919105371A BR9105371A (pt) | 1990-12-20 | 1991-12-12 | Formulacao apropriada para a administracao transdermica de dobutamina e processo para aumentar a contratilidade cardiaca |
Country Status (12)
| Country | Link |
|---|---|
| EP (1) | EP0492930A3 (pt) |
| JP (1) | JPH04275219A (pt) |
| KR (1) | KR920011479A (pt) |
| AU (1) | AU8985791A (pt) |
| BR (1) | BR9105371A (pt) |
| CA (1) | CA2057647A1 (pt) |
| CS (1) | CS379491A3 (pt) |
| HU (1) | HU914012D0 (pt) |
| IE (1) | IE914453A1 (pt) |
| IL (1) | IL100367A0 (pt) |
| MX (1) | MX9102627A (pt) |
| ZA (1) | ZA919853B (pt) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2014505726A (ja) * | 2011-02-15 | 2014-03-06 | イーライ リリー アンド カンパニー | フェンタニルの経皮溶液を使用してイヌにおける疼痛を抑制するための方法 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3527864A (en) * | 1966-11-18 | 1970-09-08 | Procter & Gamble | Compositions for topical application to animal tissue and method of enhancing penetration thereof |
| US3551554A (en) * | 1968-08-16 | 1970-12-29 | Crown Zellerbach Corp | Enhancing tissue penetration of physiologically active agents with dmso |
| US3987200A (en) * | 1972-04-12 | 1976-10-19 | Eli Lilly And Company | Method for increasing cardiac contractility |
| US4581225A (en) * | 1984-04-25 | 1986-04-08 | Eli Lilly And Company | Sustained release intranasal formulation and method of use thereof |
| US4704407A (en) * | 1984-12-20 | 1987-11-03 | Eli Lilly And Company | Soluble dobutamine salts |
| ATE77962T1 (de) * | 1985-02-25 | 1992-07-15 | Univ Rutgers | Dosierungssystem fuer transdermale absorption von arzneimittelwirkstoffen. |
| JPS62169723A (ja) * | 1986-01-22 | 1987-07-25 | Teisan Seiyaku Kk | 徐放化製剤 |
| US4814173A (en) * | 1987-09-08 | 1989-03-21 | Warner-Lambert Company | Silicone elastomer transdermal matrix system |
-
1991
- 1991-12-12 BR BR919105371A patent/BR9105371A/pt unknown
- 1991-12-13 IL IL100367A patent/IL100367A0/xx unknown
- 1991-12-13 ZA ZA919853A patent/ZA919853B/xx unknown
- 1991-12-13 CA CA002057647A patent/CA2057647A1/en not_active Abandoned
- 1991-12-13 CS CS913794A patent/CS379491A3/cs unknown
- 1991-12-17 MX MX9102627A patent/MX9102627A/es unknown
- 1991-12-17 JP JP3333268A patent/JPH04275219A/ja not_active Withdrawn
- 1991-12-17 EP EP19910311691 patent/EP0492930A3/en not_active Withdrawn
- 1991-12-18 AU AU89857/91A patent/AU8985791A/en not_active Abandoned
- 1991-12-18 HU HU914012A patent/HU914012D0/hu unknown
- 1991-12-18 KR KR1019910023332A patent/KR920011479A/ko not_active Withdrawn
- 1991-12-19 IE IE445391A patent/IE914453A1/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CS379491A3 (en) | 1992-07-15 |
| ZA919853B (en) | 1993-06-14 |
| EP0492930A3 (en) | 1992-10-14 |
| HU914012D0 (en) | 1992-03-30 |
| AU8985791A (en) | 1992-06-25 |
| IL100367A0 (en) | 1992-09-06 |
| MX9102627A (es) | 1992-06-01 |
| JPH04275219A (ja) | 1992-09-30 |
| EP0492930A2 (en) | 1992-07-01 |
| IE914453A1 (en) | 1992-07-01 |
| CA2057647A1 (en) | 1992-06-21 |
| KR920011479A (ko) | 1992-07-24 |
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