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BR0215281A - Fused heterocyclic succinimide compounds and their analogues, modulators of nuclear hormone receptor function - Google Patents

Fused heterocyclic succinimide compounds and their analogues, modulators of nuclear hormone receptor function

Info

Publication number
BR0215281A
BR0215281A BR0215281-9A BR0215281A BR0215281A BR 0215281 A BR0215281 A BR 0215281A BR 0215281 A BR0215281 A BR 0215281A BR 0215281 A BR0215281 A BR 0215281A
Authority
BR
Brazil
Prior art keywords
analogues
modulators
compounds
hormone receptor
fused heterocyclic
Prior art date
Application number
BR0215281-9A
Other languages
Portuguese (pt)
Inventor
Mark E Salvati
James Aaron Balog
Darcia A Pickering
Soren Giese
Aberra Fura
Wenying Li
Ramesh N Patel
Ronald L Hanson
Toomas Mitt
Jacques Roberge
James R Corte
Steven H Spergel
Richard A Rampulla
Raj Misra
Hai-Yun Xiao
Original Assignee
Bristol Myers Squibb Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bristol Myers Squibb Co filed Critical Bristol Myers Squibb Co
Publication of BR0215281A publication Critical patent/BR0215281A/en

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    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D495/18—Bridged systems
    • A—HUMAN NECESSITIES
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    • A61P5/32—Antioestrogens
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/22—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains four or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/08—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

"COMPOSTOS DE SUCCINIMIDA HETEROCìCLICOS FUNDIDOS E SEUS ANáLOGOS, MODULADORES DA FUNçãO DO RECEPTOR DE HORMÈNIO NUCLEAR". Compostos cíclicos fundidos, métodos de usar tais compostos no tratamento de condições associadas ao receptor de hormónio nuclear, tais como o câncer e os distúrbios imunes, e composições farmacêuticas contendo tais compostos."Fused Heterocyclic Succinaminide Compounds and Their Analogues, Modulators of NUCLEAR HORMEN RECEPTOR FUNCTION". Fused cyclic compounds, methods of using such compounds in the treatment of nuclear hormone receptor associated conditions, such as cancer and immune disorders, and pharmaceutical compositions containing such compounds.

BR0215281-9A 2001-12-19 2002-12-18 Fused heterocyclic succinimide compounds and their analogues, modulators of nuclear hormone receptor function BR0215281A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US2511601A 2001-12-19 2001-12-19
PCT/US2002/040598 WO2003062241A1 (en) 2001-12-19 2002-12-18 Fused heterocyclic succinimidecompounds and analogs thereof, modulators of nuclear hormone receptor function

Publications (1)

Publication Number Publication Date
BR0215281A true BR0215281A (en) 2004-10-19

Family

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Family Applications (1)

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BR0215281-9A BR0215281A (en) 2001-12-19 2002-12-18 Fused heterocyclic succinimide compounds and their analogues, modulators of nuclear hormone receptor function

Country Status (31)

Country Link
EP (1) EP1458723B1 (en)
JP (1) JP2005523257A (en)
KR (1) KR20040086248A (en)
CN (1) CN1589271A (en)
AR (1) AR037950A1 (en)
AT (1) ATE411319T1 (en)
AU (1) AU2002361785B2 (en)
BR (1) BR0215281A (en)
CA (1) CA2471342A1 (en)
CO (1) CO5640082A2 (en)
DE (1) DE60229435D1 (en)
DK (1) DK1458723T3 (en)
ES (1) ES2314127T3 (en)
GE (1) GEP20063817B (en)
HR (1) HRP20040567A2 (en)
HU (1) HUP0402554A3 (en)
IL (1) IL162547A0 (en)
IS (1) IS7324A (en)
MX (1) MXPA04005876A (en)
NO (1) NO20043068L (en)
NZ (1) NZ533471A (en)
PL (1) PL370904A1 (en)
PT (1) PT1458723E (en)
RU (1) RU2330038C2 (en)
SI (1) SI1458723T1 (en)
TW (1) TWI263640B (en)
UA (1) UA78265C2 (en)
UY (1) UY27595A1 (en)
WO (1) WO2003062241A1 (en)
YU (1) YU53604A (en)
ZA (1) ZA200404812B (en)

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