BR0208508A - Cyclopropylindole derivatives as selective serotonin uptake inhibitors - Google Patents
Cyclopropylindole derivatives as selective serotonin uptake inhibitorsInfo
- Publication number
- BR0208508A BR0208508A BR0208508-9A BR0208508A BR0208508A BR 0208508 A BR0208508 A BR 0208508A BR 0208508 A BR0208508 A BR 0208508A BR 0208508 A BR0208508 A BR 0208508A
- Authority
- BR
- Brazil
- Prior art keywords
- disorders
- derivatives
- selective serotonin
- cyclopropylindole
- uptake inhibitors
- Prior art date
Links
- INCAQIRDTKGRNM-UHFFFAOYSA-N 2-cyclopropyl-1h-indole Chemical class C1CC1C1=CC2=CC=CC=C2N1 INCAQIRDTKGRNM-UHFFFAOYSA-N 0.000 title 1
- 239000003772 serotonin uptake inhibitor Substances 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 208000019901 Anxiety disease Diseases 0.000 abstract 1
- 208000020925 Bipolar disease Diseases 0.000 abstract 1
- 208000000094 Chronic Pain Diseases 0.000 abstract 1
- 208000020401 Depressive disease Diseases 0.000 abstract 1
- 208000030814 Eating disease Diseases 0.000 abstract 1
- 208000019454 Feeding and Eating disease Diseases 0.000 abstract 1
- 208000021384 Obsessive-Compulsive disease Diseases 0.000 abstract 1
- 208000002193 Pain Diseases 0.000 abstract 1
- 208000028017 Psychotic disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 208000035475 disorder Diseases 0.000 abstract 1
- 235000014632 disordered eating Nutrition 0.000 abstract 1
- 230000001544 dysphoric effect Effects 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 208000019906 panic disease Diseases 0.000 abstract 1
- 206010036596 premature ejaculation Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 201000000980 schizophrenia Diseases 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
DERIVADOS DE CICLOPROPILINDOL COMO INIBIDORES SELETIVOS DA CAPTAçãO DE SEROTONINA. A presente invenção está relacionada aos compostos de fórmula (I) e seus sais ou solvatos farmaceuticamente aceitáveis e formulações farmaceuticamente aceitáveis que compreendem os citados composoto úteis para o tratamento da depressão, de distúrbios da ansiedade, ejaculação precoce, dor crónica, distúrbios compulsivo-obssessivo, distúrbios alimentares, distúrbios pré-mestrual disfórico, distúrbios do pânico e distúrbios psicóticos incluindo distúrbios bipolares e esquizofrenia.CYCLOPROPILINDOL DERIVATIVES AS SELECTIVE SEROTONIN-INHIBITORS. The present invention relates to the compounds of formula (I) and their pharmaceutically acceptable salts or solvates and pharmaceutically acceptable formulations comprising said compounds useful for the treatment of depression, anxiety disorders, premature ejaculation, chronic pain, obsessive compulsive disorders , eating disorders, dysphoric premenstrual disorders, panic disorders and psychotic disorders including bipolar disorders and schizophrenia.
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US27988801P | 2001-03-29 | 2001-03-29 | |
| US29312201P | 2001-05-23 | 2001-05-23 | |
| US23780401P | 2001-10-09 | 2001-10-09 | |
| PCT/US2002/006627 WO2002079152A1 (en) | 2001-03-29 | 2002-03-05 | Cyclopropylindole derivatives as selective serotonin reuptake inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0208508A true BR0208508A (en) | 2004-04-20 |
Family
ID=32234124
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0208508-9A BR0208508A (en) | 2001-03-29 | 2002-03-05 | Cyclopropylindole derivatives as selective serotonin uptake inhibitors |
Country Status (1)
| Country | Link |
|---|---|
| BR (1) | BR0208508A (en) |
-
2002
- 2002-03-05 BR BR0208508-9A patent/BR0208508A/en not_active Application Discontinuation
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B11A | Dismissal acc. art.33 of ipl - examination not requested within 36 months of filing | ||
| B11Y | Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette] |