BR0113731A - Comprimidos contendo epinastina produzidos por compressão direta - Google Patents
Comprimidos contendo epinastina produzidos por compressão diretaInfo
- Publication number
- BR0113731A BR0113731A BR0113731-0A BR0113731A BR0113731A BR 0113731 A BR0113731 A BR 0113731A BR 0113731 A BR0113731 A BR 0113731A BR 0113731 A BR0113731 A BR 0113731A
- Authority
- BR
- Brazil
- Prior art keywords
- epinastine
- direct compression
- containing tablets
- tablets produced
- produced
- Prior art date
Links
- 238000007907 direct compression Methods 0.000 title abstract 3
- WHWZLSFABNNENI-UHFFFAOYSA-N epinastine Chemical compound C1C2=CC=CC=C2C2CN=C(N)N2C2=CC=CC=C21 WHWZLSFABNNENI-UHFFFAOYSA-N 0.000 title abstract 2
- 229960003449 epinastine Drugs 0.000 title abstract 2
- 238000000034 method Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2095—Tabletting processes; Dosage units made by direct compression of powders or specially processed granules, by eliminating solvents, by melt-extrusion, by injection molding, by 3D printing
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Immunology (AREA)
- Pulmonology (AREA)
- Medicinal Preparation (AREA)
- Enzymes And Modification Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Plant Substances (AREA)
Abstract
"COMPRIMIDOS CONTENDO EPINASTINA PRODUZIDOS POR COMPRESSãO DIRETA". A invenção refere-se a um comprimido produzido por um processo de compressão direta compreendendo Epinastina como agente com uma estabilidade a armazenamento aperfeiçoada.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2000315849A JP2002087963A (ja) | 2000-09-08 | 2000-09-08 | 直接打錠により製造されたエピナスチン含有錠剤 |
| PCT/EP2001/010139 WO2002020018A1 (en) | 2000-09-08 | 2001-09-04 | Tablets containing epinastine manufactured by direct compression |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0113731A true BR0113731A (pt) | 2003-07-29 |
Family
ID=18794888
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0113731-0A BR0113731A (pt) | 2000-09-08 | 2001-09-04 | Comprimidos contendo epinastina produzidos por compressão direta |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JP2002087963A (pt) |
| AU (1) | AU2001291820A1 (pt) |
| BR (1) | BR0113731A (pt) |
| EC (1) | ECSP034501A (pt) |
| MX (1) | MXPA03002013A (pt) |
| WO (1) | WO2002020018A1 (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2494065A1 (en) * | 2002-08-02 | 2004-02-19 | Boehringer Ingelheim International Gmbh | Pharmaceutical formulations comprising combinations of epinastine, pseudoephedrine and methylephedrine |
| JP5162141B2 (ja) * | 2007-02-20 | 2013-03-13 | エスエス製薬株式会社 | フィルムコーティング用組成物 |
| JP5291324B2 (ja) * | 2007-11-01 | 2013-09-18 | 沢井製薬株式会社 | 口腔内崩壊錠 |
| JP5806490B2 (ja) * | 2011-03-31 | 2015-11-10 | エスエス製薬株式会社 | フィルムコーティング用組成物 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19542281C2 (de) * | 1995-11-14 | 1997-12-04 | Boehringer Ingelheim Kg | Verwendung von Epinastin für die Behandlung der Migräne |
| CN1283115A (zh) * | 1997-12-23 | 2001-02-07 | 先灵公司 | 用于治疗呼吸道和皮肤病的含有至少一种白三烯拮抗剂和至少一种抗组胺药的组合物 |
| EP1000623A1 (en) * | 1998-09-29 | 2000-05-17 | BOEHRINGER INGELHEIM INTERNATIONAL GmbH | Use of epinastine as antitussivum |
| JP4016128B2 (ja) * | 1999-09-09 | 2007-12-05 | 東和薬品株式会社 | 耐光性塩酸エピナスチンフィルムコート錠 |
-
2000
- 2000-09-08 JP JP2000315849A patent/JP2002087963A/ja active Pending
-
2001
- 2001-09-04 WO PCT/EP2001/010139 patent/WO2002020018A1/en not_active Ceased
- 2001-09-04 BR BR0113731-0A patent/BR0113731A/pt not_active IP Right Cessation
- 2001-09-04 AU AU2001291820A patent/AU2001291820A1/en not_active Abandoned
- 2001-09-04 MX MXPA03002013A patent/MXPA03002013A/es not_active Application Discontinuation
-
2003
- 2003-03-05 EC EC2003004501A patent/ECSP034501A/es unknown
Also Published As
| Publication number | Publication date |
|---|---|
| WO2002020018A1 (en) | 2002-03-14 |
| ECSP034501A (es) | 2003-04-25 |
| AU2001291820A1 (en) | 2002-03-22 |
| MXPA03002013A (es) | 2003-07-24 |
| JP2002087963A (ja) | 2002-03-27 |
| WO2002020018A8 (en) | 2002-09-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 7A E 8A ANUIDADES |
|
| B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2021 DE 29/09/2009. |