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BR0111594A - Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local - Google Patents

Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local

Info

Publication number
BR0111594A
BR0111594A BR0111594-4A BR0111594A BR0111594A BR 0111594 A BR0111594 A BR 0111594A BR 0111594 A BR0111594 A BR 0111594A BR 0111594 A BR0111594 A BR 0111594A
Authority
BR
Brazil
Prior art keywords
pyrimidines
unsubstituted
substituted
alkyl
compounds
Prior art date
Application number
BR0111594-4A
Other languages
English (en)
Inventor
Klaus-Juergen Pees
Waldemar Pfrengle
Gavin Heffernan
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of BR0111594A publication Critical patent/BR0111594A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

"PIRIMIDINAS, PROCESSO PARA A PREPARAçãO DE PIRIMIDINAS, COMPOSTOS, COMPOSIçãO FUNGICIDA, E, MéTODO PARA COMBATER FUNGO EM UM LOCAL". As pirimidinas da fórmula (I) em que R^ 1^ representa hidrogênio ou alquila, haloalquila, alquenila, alquinila, alcadienila, alcóxi, cicloalquila, fenila ou heteroarila de 5 ou 6 membros ou heterociclila de 5 ou 6 membros, contendo de um a quatro átomos de nitrogênio ou de um a três átomos de nitrogênio e um átomo de enxofre ou de oxigênio ou tri-alquil-silila, formila ou alcoxicarbonila, em que os grupos R^ 1^ são não substituídos ou substituídos como definido no relatório descritivo; R^ 2^ representa fenila, cicloalquila ou heteroarila de 5 ou 6 membros, contendo de um a quatro átomos de nitrogênio ou de um a três átomos de nitrogênio e um átomo de enxofre ou de oxigênio, que são não substituídos ou substituídos; R^ 3^ representa hidrogênio, halogênio ou alquila, alcóxi, alquiltio, alquilamino ou dialquilamino; que são não substituídos ou substituídos; R^ 4^ representa hidrogênio ou alquila, alquenila ou alquinila; que são não substituídos ou substituídos; e X representa O, S, NR^ 5^ ou uma ligação simples, em que R^ 5^ representa hidrogênio ou alquila; ou R^ 1^ e R^ 5^ juntos com o átomo de nitrogênio interjacente formam um anel heterocíclico; processos e intermediários para preparar estes compostos, a composições que os compreendam e ao seu uso para controlar fungos nocivos.
BR0111594-4A 2000-06-13 2001-06-11 Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local BR0111594A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21126200P 2000-06-13 2000-06-13
US23163200P 2000-09-11 2000-09-11
PCT/EP2001/006565 WO2001096314A1 (en) 2000-06-13 2001-06-11 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines

Publications (1)

Publication Number Publication Date
BR0111594A true BR0111594A (pt) 2003-04-15

Family

ID=26905995

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0111594-4A BR0111594A (pt) 2000-06-13 2001-06-11 Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local

Country Status (19)

Country Link
US (5) US6632821B2 (pt)
EP (1) EP1289963B1 (pt)
JP (1) JP2004503542A (pt)
KR (1) KR20030011894A (pt)
CN (1) CN1279027C (pt)
AT (1) ATE303367T1 (pt)
AU (1) AU778913B2 (pt)
BR (1) BR0111594A (pt)
CA (1) CA2412010A1 (pt)
CZ (1) CZ20024041A3 (pt)
DE (1) DE60113104D1 (pt)
EA (1) EA005927B1 (pt)
ES (1) ES2246330T3 (pt)
HU (1) HUP0300649A3 (pt)
IL (2) IL153016A0 (pt)
MX (1) MXPA02012073A (pt)
PL (1) PL362551A1 (pt)
SK (1) SK17452002A3 (pt)
WO (1) WO2001096314A1 (pt)

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KR100849311B1 (ko) 2001-03-15 2008-07-29 바스프 에스이 5-페닐피리미딘, 그의 제조를 위한 방법 및 중간 생성물,및 병원성 진균을 방제하기 위한 그의 용도
GB0126914D0 (en) * 2001-11-08 2002-01-02 Syngenta Ltd Fungicides
PL371059A1 (en) * 2001-11-19 2005-06-13 Basf Aktiengesellschaft 5-phenylpyrimidines, agents comprising the same, method for production and use thereof
JP2006518717A (ja) * 2003-02-06 2006-08-17 ビーエーエスエフ　アクチェンゲゼルシャフト ピリミジン類、製造およびそれの使用
JP2006522045A (ja) 2003-04-04 2006-09-28 ビーエーエスエフ　アクチェンゲゼルシャフト ２−置換ピリミジン
CA2525762A1 (en) * 2003-05-20 2004-12-02 Basf Aktiengesellschaft 2-substituted pyrimidines
SI1651618T1 (sl) 2003-07-24 2007-06-30 Basf Ag 2-substituirani pirimidini
MXPA06003207A (es) * 2003-09-24 2006-06-23 Wyeth Corp 5-arilpirimidinas como agentes anti-cancer.
DE10360370A1 (de) * 2003-12-22 2005-07-14 Bayer Cropscience Ag Triazolopyrimidine
DE102004003428A1 (de) * 2004-01-23 2005-08-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue langwirksame Beta-2-Agonisten, und deren Verwendung als Arzneimittel
DE102004003493A1 (de) * 2004-01-23 2005-08-11 Bayer Cropscience Ag 5-Phenylpyrimidine
BRPI0515405A (pt) * 2004-09-17 2008-07-22 Basf Ag uso de compostos, método para a proteção de plantas de ataque ou infestação por pragas nematódeas, e, semente
BRPI0608411A2 (pt) * 2005-03-10 2009-12-29 Basf Ag uso de um composto, composto, processo para preparar compostos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos
GB0512844D0 (en) * 2005-06-23 2005-08-03 Novartis Ag Organic compounds
EP2001298A2 (de) * 2006-03-27 2008-12-17 Basf Se Substituierte 5-hetaryl-4-aminopyrimidine
WO2007113322A2 (de) * 2006-04-05 2007-10-11 Basf Se Substituierte 5-hetarylpyrimidine zur bekämpfung von pflanzenschädigenden pilzen und von krebserkrankungen
CL2007002231A1 (es) * 2006-08-02 2008-04-11 Basf Ag Uso de compuestos derivados de 5-(het) arilpirimidina para combatir hongos daninos; compuestos derivados de 5-(het) arilpirimidina; agente fungicida; y agente farmaceutico.
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JP5731976B2 (ja) * 2008-08-20 2015-06-10 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． 置換ピリジン誘導体および置換ピリミジン誘導体ならびにそれらのウイルス感染の治療における使用
TWI602802B (zh) * 2012-12-19 2017-10-21 陶氏農業科學公司 殺蟲組成物及其相關之方法（四）
CN104892528A (zh) * 2014-12-10 2015-09-09 上海工程技术大学 一种2-硫代巴比妥酸衍生物的制备方法
JP7560359B2 (ja) * 2018-04-13 2024-10-02 バイエル アクチェンゲゼルシャフト 殺虫混合物の固体製剤

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Also Published As

Publication number Publication date
EP1289963A1 (en) 2003-03-12
US20040147744A1 (en) 2004-07-29
US6632821B2 (en) 2003-10-14
ES2246330T3 (es) 2006-02-16
CZ20024041A3 (cs) 2003-04-16
US6943252B2 (en) 2005-09-13
SK17452002A3 (sk) 2003-06-03
AU7056401A (en) 2001-12-24
EA005927B1 (ru) 2005-08-25
EP1289963B1 (en) 2005-08-31
EA200201253A1 (ru) 2003-04-24
KR20030011894A (ko) 2003-02-11
MXPA02012073A (es) 2003-04-25
WO2001096314A1 (en) 2001-12-20
IL153016A0 (en) 2003-06-24
CN1443174A (zh) 2003-09-17
ATE303367T1 (de) 2005-09-15
JP2004503542A (ja) 2004-02-05
CN1279027C (zh) 2006-10-11
US7230104B2 (en) 2007-06-12
US20050282847A1 (en) 2005-12-22
AU778913B2 (en) 2004-12-23
HUP0300649A2 (hu) 2003-07-28
CA2412010A1 (en) 2001-12-20
PL362551A1 (en) 2004-11-02
US20030088096A1 (en) 2003-05-08
HUP0300649A3 (en) 2003-10-28
DE60113104D1 (de) 2005-10-06
IL176276A0 (en) 2006-10-05
US20050282828A1 (en) 2005-12-22
US20070208037A1 (en) 2007-09-06

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2016 DE 25/08/2009.