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BR0111594A - Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local - Google Patents

Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local

Info

Publication number
BR0111594A
BR0111594A BR0111594-4A BR0111594A BR0111594A BR 0111594 A BR0111594 A BR 0111594A BR 0111594 A BR0111594 A BR 0111594A BR 0111594 A BR0111594 A BR 0111594A
Authority
BR
Brazil
Prior art keywords
pyrimidines
unsubstituted
substituted
alkyl
compounds
Prior art date
Application number
BR0111594-4A
Other languages
English (en)
Inventor
Klaus-Juergen Pees
Waldemar Pfrengle
Gavin Heffernan
Original Assignee
Basf Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Basf Ag filed Critical Basf Ag
Publication of BR0111594A publication Critical patent/BR0111594A/pt

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/40—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having a double or triple bond to nitrogen, e.g. cyanates, cyanamides
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/38—One sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

"PIRIMIDINAS, PROCESSO PARA A PREPARAçãO DE PIRIMIDINAS, COMPOSTOS, COMPOSIçãO FUNGICIDA, E, MéTODO PARA COMBATER FUNGO EM UM LOCAL". As pirimidinas da fórmula (I) em que R^ 1^ representa hidrogênio ou alquila, haloalquila, alquenila, alquinila, alcadienila, alcóxi, cicloalquila, fenila ou heteroarila de 5 ou 6 membros ou heterociclila de 5 ou 6 membros, contendo de um a quatro átomos de nitrogênio ou de um a três átomos de nitrogênio e um átomo de enxofre ou de oxigênio ou tri-alquil-silila, formila ou alcoxicarbonila, em que os grupos R^ 1^ são não substituídos ou substituídos como definido no relatório descritivo; R^ 2^ representa fenila, cicloalquila ou heteroarila de 5 ou 6 membros, contendo de um a quatro átomos de nitrogênio ou de um a três átomos de nitrogênio e um átomo de enxofre ou de oxigênio, que são não substituídos ou substituídos; R^ 3^ representa hidrogênio, halogênio ou alquila, alcóxi, alquiltio, alquilamino ou dialquilamino; que são não substituídos ou substituídos; R^ 4^ representa hidrogênio ou alquila, alquenila ou alquinila; que são não substituídos ou substituídos; e X representa O, S, NR^ 5^ ou uma ligação simples, em que R^ 5^ representa hidrogênio ou alquila; ou R^ 1^ e R^ 5^ juntos com o átomo de nitrogênio interjacente formam um anel heterocíclico; processos e intermediários para preparar estes compostos, a composições que os compreendam e ao seu uso para controlar fungos nocivos.
BR0111594-4A 2000-06-13 2001-06-11 Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local BR0111594A (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US21126200P 2000-06-13 2000-06-13
US23163200P 2000-09-11 2000-09-11
PCT/EP2001/006565 WO2001096314A1 (en) 2000-06-13 2001-06-11 Fungicidal 5-phenyl substituted 2-(cyanoamino) pyrimidines

Publications (1)

Publication Number Publication Date
BR0111594A true BR0111594A (pt) 2003-04-15

Family

ID=26905995

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0111594-4A BR0111594A (pt) 2000-06-13 2001-06-11 Pirimidinas, processo para a preparação de pirimidinas, compostos, composição fungicida, e, método papa combater fungo em um local

Country Status (19)

Country Link
US (5) US6632821B2 (pt)
EP (1) EP1289963B1 (pt)
JP (1) JP2004503542A (pt)
KR (1) KR20030011894A (pt)
CN (1) CN1279027C (pt)
AT (1) ATE303367T1 (pt)
AU (1) AU778913B2 (pt)
BR (1) BR0111594A (pt)
CA (1) CA2412010A1 (pt)
CZ (1) CZ20024041A3 (pt)
DE (1) DE60113104D1 (pt)
EA (1) EA005927B1 (pt)
ES (1) ES2246330T3 (pt)
HU (1) HUP0300649A3 (pt)
IL (2) IL153016A0 (pt)
MX (1) MXPA02012073A (pt)
PL (1) PL362551A1 (pt)
SK (1) SK17452002A3 (pt)
WO (1) WO2001096314A1 (pt)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL157723A0 (en) * 2001-03-15 2004-03-28 Basf Ag 5-phenylpyrimidine, methods and intermediate products for the production thereof and use of the same for controlling pathogenic fungi
GB0126914D0 (en) * 2001-11-08 2002-01-02 Syngenta Ltd Fungicides
HUP0402385A3 (en) 2001-11-19 2005-10-28 Basf Ag 5-phenylpyrimidines, fungicide compositions comprising the same, method for producing and use thereof
US20060058326A1 (en) * 2003-02-06 2006-03-16 Basf Aktiengesllschaft Pyrimidines, methods for the production thereof, and use thereof
BRPI0409159A (pt) * 2003-04-04 2006-05-02 Basf Ag composto, processo para preparar 2-pirimidinas substituìdas, agente adequado para combater fungos nocivos, e, processo para combater fungos fitopatogênicos nocivos
KR20060013665A (ko) * 2003-05-20 2006-02-13 바스프 악티엔게젤샤프트 2-치환 피리미딘
EP1651618B1 (de) 2003-07-24 2007-01-03 Basf Aktiengesellschaft 2-substituierte pyrimidine
BRPI0414736A (pt) 2003-09-24 2006-11-21 Wyeth Corp 5-aril-pirimidinas como agentes anticáncer
DE10360370A1 (de) * 2003-12-22 2005-07-14 Bayer Cropscience Ag Triazolopyrimidine
DE102004003493A1 (de) * 2004-01-23 2005-08-11 Bayer Cropscience Ag 5-Phenylpyrimidine
DE102004003428A1 (de) * 2004-01-23 2005-08-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue langwirksame Beta-2-Agonisten, und deren Verwendung als Arzneimittel
MX2007002590A (es) * 2004-09-17 2007-05-15 Basf Ag Uso de pirimidinas 2 - substituidas para combatir enfermedades de nematodo de plantas.
US20080176744A1 (en) * 2005-03-10 2008-07-24 Basf Aktiengesellschaft Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them
GB0512844D0 (en) * 2005-06-23 2005-08-03 Novartis Ag Organic compounds
US20110201496A1 (en) * 2006-03-27 2011-08-18 Joachim Rheinheimer Substituted 5-Hetaryl-4-Aminopyrimidines
WO2007113322A2 (de) * 2006-04-05 2007-10-11 Basf Se Substituierte 5-hetarylpyrimidine zur bekämpfung von pflanzenschädigenden pilzen und von krebserkrankungen
CL2007002231A1 (es) * 2006-08-02 2008-04-11 Basf Ag Uso de compuestos derivados de 5-(het) arilpirimidina para combatir hongos daninos; compuestos derivados de 5-(het) arilpirimidina; agente fungicida; y agente farmaceutico.
DE102007012908A1 (de) 2007-03-19 2008-09-25 Momentive Performance Materials Gmbh Neue Polyamid-Polysiloxan-Verbindungen
JP5731976B2 (ja) * 2008-08-20 2015-06-10 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． 置換ピリジン誘導体および置換ピリミジン誘導体ならびにそれらのウイルス感染の治療における使用
MA38246B1 (fr) * 2012-12-19 2017-12-29 Dow Agrosciences Llc Compositions pesticides et leurs procédés associés
CN104892528A (zh) * 2014-12-10 2015-09-09 上海工程技术大学 一种2-硫代巴比妥酸衍生物的制备方法
TWI820115B (zh) * 2018-04-13 2023-11-01 德商拜耳廠股份有限公司 殺昆蟲混合物之固體調配物

Family Cites Families (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2444606A (en) * 1945-12-15 1948-07-06 Gen Aniline & Film Corp Stabilizers for photographic emulsions
US3441560A (en) * 1967-03-14 1969-04-29 Geigy Chem Corp Cyclopropyl-2-sulphanilamido-pyrimidines
DD145913A1 (de) * 1979-02-27 1981-01-14 Horst Zaschke Verfahren zur herstellung von 2-cy n-5-eckige klammer auf 4-acyloxy-phenyl eckige klammer u-pyrimidinen
US4438117A (en) * 1980-09-03 1984-03-20 E. I. Du Pont De Nemours And Company 2-Substituted thio-4,5-diarylpyrimidines
US4504482A (en) * 1983-07-28 1985-03-12 Sterling Drug Inc. [5(or 4)-(Pyridinyl)-2-pyrimidinyl]ureas and cardiotonic use thereof
DE3525977A1 (de) 1985-07-20 1987-01-29 Bayer Ag Verfahren zur herstellung von 2-cyanamino-pyrimidin-derivaten
US4847258A (en) * 1986-08-26 1989-07-11 Ciba-Geigy Corporation Substituted benzoylphenylureas compounds useful as pesticides
DE3709549A1 (de) 1987-03-24 1988-10-06 Hoechst Ag Verwendung von 5-phenyl-pyrimidinderivaten als komponenten in smektischen fluessigkristallmischungen
DE3709618A1 (de) * 1987-03-24 1988-10-06 Hoechst Ag Neue fluessigkristalline 5-phenylpyrimidin-derivate mit s(pfeil abwaerts)c(pfeil abwaerts)-oder s(pfeil abwaerts)c(pfeil abwaerts) -phase und verfahren zu ihrer herstellung
DE3733818A1 (de) * 1987-10-07 1989-04-20 Merck Patent Gmbh Ferroelektrische fluessigkristalline phasen
DE3734158A1 (de) 1987-10-09 1989-04-20 Kugelfischer G Schaefer & Co Verfahren und vorrichtung zum ermitteln der tatsaechlichen kuenstlichen alpha-aerosolaktivitaets-konzentration in der luft
DE4003012A1 (de) 1990-02-02 1991-08-08 Hoechst Ag Geminale dimethylalkyl-verbindungen, verfahren zu ihrer herstellung und ihre verwendung in fluessigkristallinen mischungen
JPH06501926A (ja) * 1990-08-06 1994-03-03 藤沢薬品工業株式会社 複素環式化合物
JPH04300871A (ja) * 1991-03-28 1992-10-23 Canon Inc 光学活性化合物、これを含む液晶組成物、それを有する液晶素子、それ等を用いた表示方法及び表示装置
US5593996A (en) 1991-12-30 1997-01-14 American Cyanamid Company Triazolopyrimidine derivatives
IL108731A (en) 1993-03-04 1997-03-18 Shell Int Research 6, N-DISUBSTITUTED-£1, 2, 4| TRIAZOLO-£1, 5-a| PYRIMIDINE- 7-AMINE DERIVATIVES, THEIR PREPARATION AND THEIR USE AS FUNGICIDES
GB2277090A (en) * 1993-04-16 1994-10-19 Shell Int Research Fungicidal tetrahydropyrimidine and imidazoline derivatives
ES2079323B1 (es) * 1994-06-21 1996-10-16 Vita Invest Sa Derivados de indol utiles para el tratamiento de la migraña, composicion y uso correspondientes.
US6245774B1 (en) 1994-06-21 2001-06-12 Celltech Therapeutics Limited Tri-substituted phenyl or pyridine derivatives
US5739333A (en) * 1995-05-16 1998-04-14 Tanabe Seiyaku Co., Ltd. Sulfonamide derivative and process for preparing the same
US5935966A (en) * 1995-09-01 1999-08-10 Signal Pharmaceuticals, Inc. Pyrimidine carboxylates and related compounds and methods for treating inflammatory conditions
PL193686B1 (pl) * 1995-09-07 2007-03-30 Hoffmann La Roche Pochodne piperydyny, środki lecznicze zawierającepochodne piperydyny, sposoby wytwarzania tych pochodnych oraz zastosowanie pochodnych
TW460476B (en) 1997-04-14 2001-10-21 American Cyanamid Co Fungicidal trifluoromethylalkylamino-triazolopyrimidines
US5994360A (en) 1997-07-14 1999-11-30 American Cyanamid Company Fungicidal 5-alkyl-triazolopyrimidines
AU750489B2 (en) 1998-02-11 2002-07-18 Wyeth Holdings Corporation Fungicidal 7-alkyl-triazolopyrimidines
CZ291765B6 (cs) 1998-03-23 2003-05-14 American Cyanamid Company 6-(2-Halogen-4-alkoxyfenyl)triazolopyrimidin, způsob jeho přípravy, fungicidní prostředek s jeho obsahem, způsob potlačování hub a použití
JO2308B1 (en) * 1999-05-31 2005-09-12 اف. هوفمان- لاروش أيه جي‏ Derivatives of phenylpyrmidine

Also Published As

Publication number Publication date
CN1279027C (zh) 2006-10-11
US6632821B2 (en) 2003-10-14
SK17452002A3 (sk) 2003-06-03
EP1289963A1 (en) 2003-03-12
JP2004503542A (ja) 2004-02-05
US20040147744A1 (en) 2004-07-29
US7230104B2 (en) 2007-06-12
PL362551A1 (en) 2004-11-02
US6943252B2 (en) 2005-09-13
HUP0300649A2 (hu) 2003-07-28
CZ20024041A3 (cs) 2003-04-16
MXPA02012073A (es) 2003-04-25
AU778913B2 (en) 2004-12-23
DE60113104D1 (de) 2005-10-06
EA005927B1 (ru) 2005-08-25
EP1289963B1 (en) 2005-08-31
US20050282847A1 (en) 2005-12-22
KR20030011894A (ko) 2003-02-11
US20050282828A1 (en) 2005-12-22
ATE303367T1 (de) 2005-09-15
US20070208037A1 (en) 2007-09-06
US20030088096A1 (en) 2003-05-08
AU7056401A (en) 2001-12-24
IL153016A0 (en) 2003-06-24
CA2412010A1 (en) 2001-12-20
EA200201253A1 (ru) 2003-04-24
ES2246330T3 (es) 2006-02-16
CN1443174A (zh) 2003-09-17
IL176276A0 (en) 2006-10-05
WO2001096314A1 (en) 2001-12-20
HUP0300649A3 (en) 2003-10-28

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Legal Events

Date Code Title Description
B08F Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette]

Free format text: REFERENTE A 8A ANUIDADE.

B08K Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette]

Free format text: REFERENTE AO DESPACHO 8.6 DA RPI 2016 DE 25/08/2009.