BR0110642A - Processo para preparação de sais de sulfonilbenzoilguanidìnio - Google Patents
Processo para preparação de sais de sulfonilbenzoilguanidìnioInfo
- Publication number
- BR0110642A BR0110642A BR0110642-2A BR0110642A BR0110642A BR 0110642 A BR0110642 A BR 0110642A BR 0110642 A BR0110642 A BR 0110642A BR 0110642 A BR0110642 A BR 0110642A
- Authority
- BR
- Brazil
- Prior art keywords
- salts
- preparation
- sulfonylbenzoylguanidium
- sulphonylbenzoilguanidine
- alkyl
- Prior art date
Links
- 150000003839 salts Chemical class 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 1
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 125000004432 carbon atom Chemical group C* 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Patente de Invenção: "PROCESSO PARA PREPARAçãO DE SAIS DE SULFONILBENZOILGUANIDìNIO". A invenção refere-se a um processo para a preparação de sais de adição ácidos dos compostos de fórmula(I) em que R^ 1^, R^ 2^ e R^ 3^ são alquila tendo de 1 a 12 átomos de carbono.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10023405A DE10023405A1 (de) | 2000-05-12 | 2000-05-12 | Verfahren zur Herstellung von Sulfonyl-benzoylguanidinum-Salzen |
| PCT/EP2001/004294 WO2001085679A1 (de) | 2000-05-12 | 2001-04-17 | Verfahren zur herstellung von sulfonyl-benzoylguanidinium-salzen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0110642A true BR0110642A (pt) | 2003-03-18 |
Family
ID=7641866
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0110642-2A BR0110642A (pt) | 2000-05-12 | 2001-04-17 | Processo para preparação de sais de sulfonilbenzoilguanidìnio |
Country Status (24)
| Country | Link |
|---|---|
| US (1) | US6706921B2 (pt) |
| EP (1) | EP1282598B1 (pt) |
| JP (1) | JP2003532704A (pt) |
| KR (1) | KR20030007599A (pt) |
| CN (1) | CN1193011C (pt) |
| AR (1) | AR028442A1 (pt) |
| AT (1) | ATE280151T1 (pt) |
| AU (1) | AU783369B2 (pt) |
| BR (1) | BR0110642A (pt) |
| CA (1) | CA2408640A1 (pt) |
| CZ (1) | CZ20023647A3 (pt) |
| DE (2) | DE10023405A1 (pt) |
| DK (1) | DK1282598T3 (pt) |
| ES (1) | ES2228897T3 (pt) |
| HU (1) | HUP0301936A2 (pt) |
| MX (1) | MXPA02011069A (pt) |
| MY (1) | MY133941A (pt) |
| NO (1) | NO20025385L (pt) |
| PL (1) | PL358690A1 (pt) |
| PT (1) | PT1282598E (pt) |
| RU (1) | RU2258699C2 (pt) |
| SK (1) | SK15812002A3 (pt) |
| WO (1) | WO2001085679A1 (pt) |
| ZA (1) | ZA200210050B (pt) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003272967A1 (en) * | 2002-10-28 | 2004-05-13 | Kaneka Corporation | Processes for producing optically active n-(2,3-epoxypropan-1-yl)phthalimide |
| JP5634985B2 (ja) | 2008-05-09 | 2014-12-03 | メルク パテント ゲゼルシャフト ミット ベシュレンクテル ハフツングMerck Patent Gesellschaft mit beschraenkter Haftung | インスリン抵抗性およびβ−細胞機能障害に関連する疾患を治療するためのリメポリドを含む医薬組成物 |
| CN108602767A (zh) * | 2016-02-08 | 2018-09-28 | 默克专利股份有限公司 | N-(4,5-双甲磺酰基-2-甲基苯甲酰基)胍盐酸盐和n-(4,5-双甲磺酰基-2-甲基苯甲酰基)胍盐的结晶变体 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS6248648A (ja) * | 1985-08-28 | 1987-03-03 | Fujisawa Pharmaceut Co Ltd | ジアルコキシ酢酸エステル化合物の製造法 |
| ATE147375T1 (de) * | 1992-09-22 | 1997-01-15 | Hoechst Ag | Benzoylguanidine, verfahren zu ihrer herstellung, sowie ihre verwendung als antiarrhythmika |
| DE4437874A1 (de) * | 1994-10-22 | 1996-04-25 | Merck Patent Gmbh | Alkyl-5-methylsulfonyl-benzoylguanidin-Derivate |
| DE19502644A1 (de) * | 1995-01-28 | 1996-08-01 | Merck Patent Gmbh | 4-Amino-benzoylguanidin-Derivate |
| DE19526381A1 (de) * | 1995-07-19 | 1997-01-23 | Hoechst Ag | 4-Fluoralkyl-substituierte Benzoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| DE19529612A1 (de) * | 1995-08-11 | 1997-02-13 | Merck Patent Gmbh | Sulfonyl- oder Sulfinyl-benzoylguanidin-Derivate |
| DE19621482A1 (de) * | 1996-05-29 | 1997-12-04 | Hoechst Ag | Substituierte 1-Naphthoylguanidine, Verfahren zu ihrer Herstellung, ihre Verwendung als Medikament oder Diagnostikum sowie sie enthaltendes Medikament |
| DE19951418A1 (de) * | 1999-10-26 | 2001-05-03 | Merck Patent Gmbh | Verfahren zur Herstellung von N-(4,5-Bismethansulfonyl-2-methyl-benzoyl) -guanidin, Hydrochlorid |
| JP2001247557A (ja) * | 1999-12-27 | 2001-09-11 | Sagami Chem Res Center | 5−オキシ−7−オキサビシクロ[4.1.0]ヘプト−3−エン−3−カルボン酸エステルの製造方法 |
-
2000
- 2000-05-12 DE DE10023405A patent/DE10023405A1/de active Pending
-
2001
- 2001-04-17 PT PT01947223T patent/PT1282598E/pt unknown
- 2001-04-17 RU RU2002133235/04A patent/RU2258699C2/ru not_active IP Right Cessation
- 2001-04-17 PL PL01358690A patent/PL358690A1/xx unknown
- 2001-04-17 AU AU68969/01A patent/AU783369B2/en not_active Ceased
- 2001-04-17 EP EP01947223A patent/EP1282598B1/de not_active Expired - Lifetime
- 2001-04-17 CN CNB018094058A patent/CN1193011C/zh not_active Expired - Fee Related
- 2001-04-17 MX MXPA02011069A patent/MXPA02011069A/es active IP Right Grant
- 2001-04-17 ES ES01947223T patent/ES2228897T3/es not_active Expired - Lifetime
- 2001-04-17 CZ CZ20023647A patent/CZ20023647A3/cs unknown
- 2001-04-17 KR KR1020027015038A patent/KR20030007599A/ko not_active Withdrawn
- 2001-04-17 HU HU0301936A patent/HUP0301936A2/hu unknown
- 2001-04-17 BR BR0110642-2A patent/BR0110642A/pt not_active Application Discontinuation
- 2001-04-17 SK SK1581-2002A patent/SK15812002A3/sk unknown
- 2001-04-17 DK DK01947223T patent/DK1282598T3/da active
- 2001-04-17 JP JP2001582280A patent/JP2003532704A/ja active Pending
- 2001-04-17 AT AT01947223T patent/ATE280151T1/de not_active IP Right Cessation
- 2001-04-17 WO PCT/EP2001/004294 patent/WO2001085679A1/de not_active Ceased
- 2001-04-17 US US10/275,484 patent/US6706921B2/en not_active Expired - Fee Related
- 2001-04-17 CA CA002408640A patent/CA2408640A1/en not_active Abandoned
- 2001-04-17 DE DE50104219T patent/DE50104219D1/de not_active Expired - Lifetime
- 2001-05-09 MY MYPI20012143 patent/MY133941A/en unknown
- 2001-05-11 AR ARP010102230A patent/AR028442A1/es unknown
-
2002
- 2002-11-11 NO NO20025385A patent/NO20025385L/no not_active Application Discontinuation
- 2002-12-11 ZA ZA200210050A patent/ZA200210050B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| NO20025385D0 (no) | 2002-11-11 |
| KR20030007599A (ko) | 2003-01-23 |
| ZA200210050B (en) | 2003-09-10 |
| ATE280151T1 (de) | 2004-11-15 |
| DK1282598T3 (da) | 2005-02-07 |
| MXPA02011069A (es) | 2003-03-10 |
| WO2001085679A1 (de) | 2001-11-15 |
| ES2228897T3 (es) | 2005-04-16 |
| JP2003532704A (ja) | 2003-11-05 |
| US6706921B2 (en) | 2004-03-16 |
| CZ20023647A3 (cs) | 2003-02-12 |
| AR028442A1 (es) | 2003-05-07 |
| AU783369B2 (en) | 2005-10-20 |
| HUP0301936A2 (hu) | 2003-09-29 |
| DE10023405A1 (de) | 2001-11-15 |
| PT1282598E (pt) | 2005-03-31 |
| EP1282598B1 (de) | 2004-10-20 |
| CA2408640A1 (en) | 2002-11-08 |
| NO20025385L (no) | 2002-11-11 |
| EP1282598A1 (de) | 2003-02-12 |
| CN1429207A (zh) | 2003-07-09 |
| CN1193011C (zh) | 2005-03-16 |
| RU2258699C2 (ru) | 2005-08-20 |
| AU6896901A (en) | 2001-11-20 |
| US20030162999A1 (en) | 2003-08-28 |
| SK15812002A3 (sk) | 2003-03-04 |
| PL358690A1 (en) | 2004-08-09 |
| DE50104219D1 (de) | 2004-11-25 |
| MY133941A (en) | 2007-11-30 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B07A | Application suspended after technical examination (opinion) [chapter 7.1 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] | ||
| B09B | Patent application refused [chapter 9.2 patent gazette] |
Free format text: MANTIDO O INDEFERIMENTO UMA VEZ QUE NAO FOI APRESENTADO RECURSO DENTRO DO PRAZO LEGAL. |