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BR0012481A - Processo para desacilação de lipodepsipeptìdeos - Google Patents

Processo para desacilação de lipodepsipeptìdeos

Info

Publication number
BR0012481A
BR0012481A BR0012481-8A BR0012481A BR0012481A BR 0012481 A BR0012481 A BR 0012481A BR 0012481 A BR0012481 A BR 0012481A BR 0012481 A BR0012481 A BR 0012481A
Authority
BR
Brazil
Prior art keywords
lipodepsipeptides
deacylation process
deacylation
dilopilation
lipodepsipeptide
Prior art date
Application number
BR0012481-8A
Other languages
English (en)
Inventor
Adam Joseph Kreuzman
Palaniappan Kulanthaivel
Michael John Rodriguez
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Publication of BR0012481A publication Critical patent/BR0012481A/pt

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/64Cyclic peptides containing only normal peptide links
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10Antimycotics
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Peptides Or Proteins (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Patente de Invenção: "PROCESSO PARA DESACILAçãO DE LIPODEPSIPEPTìDEOS". é descrito um processo para desacilação de um lipodepsipeptídeo para produzir o correspondente núcleo. Os produtos produzidos a partir deste processo também são descritos (por exemplo, um núcleo pseudomicina representado por estruturas (I) ou (II)).
BR0012481-8A 1999-07-15 2000-06-08 Processo para desacilação de lipodepsipeptìdeos BR0012481A (pt)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14396899P 1999-07-15 1999-07-15
PCT/US2000/015018 WO2001005815A1 (en) 1999-07-15 2000-06-08 Process for deacylation of lipodepsipeptides

Publications (1)

Publication Number Publication Date
BR0012481A true BR0012481A (pt) 2002-04-02

Family

ID=22506494

Family Applications (1)

Application Number Title Priority Date Filing Date
BR0012481-8A BR0012481A (pt) 1999-07-15 2000-06-08 Processo para desacilação de lipodepsipeptìdeos

Country Status (11)

Country Link
EP (1) EP1198471A1 (pt)
JP (1) JP2003505042A (pt)
CN (1) CN1361791A (pt)
AU (1) AU5310600A (pt)
BR (1) BR0012481A (pt)
CA (1) CA2378868A1 (pt)
EA (1) EA200200162A1 (pt)
HU (1) HUP0202315A2 (pt)
MX (1) MXPA02000458A (pt)
NO (1) NO20020183L (pt)
WO (1) WO2001005815A1 (pt)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1362865A4 (en) 2001-02-19 2004-05-06 Takara Bio Inc CYCLIC PEPTIDE
DE10335584B4 (de) * 2003-07-31 2006-06-29 Philipps-Universität Marburg Verfahren zur Herstellung zyklischer Moleküle
US20060004185A1 (en) * 2004-07-01 2006-01-05 Leese Richard A Peptide antibiotics and peptide intermediates for their prepartion
DE102004060750A1 (de) * 2004-12-15 2006-07-13 Sanofi-Aventis Deutschland Gmbh Verfahren zur Deacylierung von Lipopeptiden
TW201035111A (en) 2008-12-23 2010-10-01 Biosource Pharm Inc Antibiotic compositions for the treatment of gram negative infections
US8415307B1 (en) 2010-06-23 2013-04-09 Biosource Pharm, Inc. Antibiotic compositions for the treatment of gram negative infections
WO2014044803A1 (en) * 2012-09-24 2014-03-27 Dsm Sinochem Pharmaceuticals Netherlands B.V. Method for producing a cyclic peptide

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DK0460882T3 (da) * 1990-06-07 1996-08-26 Lilly Co Eli Lipopeptiddeacylase

Also Published As

Publication number Publication date
EP1198471A1 (en) 2002-04-24
HUP0202315A2 (en) 2002-10-28
MXPA02000458A (es) 2002-07-02
CN1361791A (zh) 2002-07-31
NO20020183D0 (no) 2002-01-14
JP2003505042A (ja) 2003-02-12
NO20020183L (no) 2002-03-13
AU5310600A (en) 2001-02-05
EA200200162A1 (ru) 2002-06-27
CA2378868A1 (en) 2001-01-25
WO2001005815A1 (en) 2001-01-25

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Legal Events

Date Code Title Description
FA10 Dismissal: dismissal - article 33 of industrial property law
B11Y Definitive dismissal - extension of time limit for request of examination expired [chapter 11.1.1 patent gazette]