BR0012058A - Combinação sinérgica: gabapentina e pregabalina - Google Patents
Combinação sinérgica: gabapentina e pregabalinaInfo
- Publication number
- BR0012058A BR0012058A BR0012058-8A BR0012058A BR0012058A BR 0012058 A BR0012058 A BR 0012058A BR 0012058 A BR0012058 A BR 0012058A BR 0012058 A BR0012058 A BR 0012058A
- Authority
- BR
- Brazil
- Prior art keywords
- pregabalin
- gabapentin
- synergistic combination
- pregabalina
- gabapentina
- Prior art date
Links
- UGJMXCAKCUNAIE-UHFFFAOYSA-N Gabapentin Chemical compound OC(=O)CC1(CN)CCCCC1 UGJMXCAKCUNAIE-UHFFFAOYSA-N 0.000 title abstract 5
- AYXYPKUFHZROOJ-ZETCQYMHSA-N pregabalin Chemical compound CC(C)C[C@H](CN)CC(O)=O AYXYPKUFHZROOJ-ZETCQYMHSA-N 0.000 title abstract 3
- 229960002870 gabapentin Drugs 0.000 title abstract 2
- 229960001233 pregabalin Drugs 0.000 title abstract 2
- 239000011885 synergistic combination Substances 0.000 title 1
- 230000002195 synergetic effect Effects 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
Landscapes
- Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Pain & Pain Management (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Epidemiology (AREA)
- Neurology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Patente de Invenção: "COMBINAçãO SINéRGICA : GABAPENTINA E PREGABALINA". A presente invenção é uma composição farmacêutica sinérgica de gabapentina e pregabalina que compreende um método melhorado para o tratamento de dor.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US14221599P | 1999-07-02 | 1999-07-02 | |
| PCT/US2000/017039 WO2001001983A1 (en) | 1999-07-02 | 2000-06-21 | A synergistic combination: gabapentin and pregabalin |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BR0012058A true BR0012058A (pt) | 2002-05-14 |
Family
ID=22499016
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BR0012058-8A BR0012058A (pt) | 1999-07-02 | 2000-06-21 | Combinação sinérgica: gabapentina e pregabalina |
Country Status (14)
| Country | Link |
|---|---|
| EP (1) | EP1196160B1 (pt) |
| JP (1) | JP2003503453A (pt) |
| AR (1) | AR030024A1 (pt) |
| AT (1) | ATE313322T1 (pt) |
| AU (1) | AU5753900A (pt) |
| BR (1) | BR0012058A (pt) |
| CA (1) | CA2373953A1 (pt) |
| CO (1) | CO5210869A1 (pt) |
| DE (1) | DE60024995T2 (pt) |
| ES (1) | ES2255500T3 (pt) |
| MX (1) | MXPA02000170A (pt) |
| PE (1) | PE20010331A1 (pt) |
| UY (1) | UY26230A1 (pt) |
| WO (1) | WO2001001983A1 (pt) |
Families Citing this family (11)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN1094757C (zh) | 1996-07-24 | 2002-11-27 | 沃尼尔·朗伯公司 | 用于治疗疼痛的异丁基γ-氨基丁酸及其衍生物 |
| WO2003066040A1 (en) | 2002-02-05 | 2003-08-14 | Ajinomoto Co.,Inc. | Medicinal compositions containing gabapentin or pregabalin and n-type calcium channel antagonist |
| US7687080B2 (en) * | 2002-11-25 | 2010-03-30 | Taraxos Inc. | Treatment of neuropathy |
| WO2004084881A1 (en) * | 2003-03-21 | 2004-10-07 | Dynogen Pharmaceuticals, Inc. | METHODS FOR TREATING FUNCTIONAL BOWEL DISORDERS USING α2δ SUBUNIT CALCIUM CHANNEL MODULATORS WITH SMOOTH MUSCLE MODULATORS |
| CN1791399A (zh) * | 2003-03-21 | 2006-06-21 | 戴诺根医药品公司 | 用α2δ亚基钙通道调节剂和平滑肌调节剂一起治疗下泌尿道病症的方法 |
| WO2004084880A1 (en) * | 2003-03-21 | 2004-10-07 | Dynogen Pharmaceuticals, Inc. | METHODS FOR TREATING PAIN USING SMOOTH MUSCLE MODULATORS AND α2δ SUBUNIT CALCIUM CHANNEL MODULATORS |
| JP2005060311A (ja) * | 2003-08-13 | 2005-03-10 | Mochida Pharmaceut Co Ltd | N−(ベンゾイル)アミノ酸誘導体を有効成分とするニューロパシー性疼痛治療剤 |
| DE102007019071A1 (de) * | 2007-04-23 | 2008-10-30 | Ratiopharm Gmbh | Stabilisierte pharmazeutische Zusammensetzung enthaltend Pregabalin |
| EP2334176A4 (en) | 2008-09-27 | 2012-05-02 | Taraxos Inc | TOPICAL FORMULATIONS FOR THE TREATMENT OF NERVE DISEASES |
| WO2010115612A2 (en) * | 2009-04-10 | 2010-10-14 | Synthon B.V. | Pregabalin compositions |
| WO2011069063A2 (en) | 2009-12-04 | 2011-06-09 | Sunovion Pharmaceuticals, Inc. | Multicyclic compounds and methods of use thereof |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO1999008667A2 (en) * | 1997-08-19 | 1999-02-25 | Warner-Lambert Company | Methods for treating physiological conditions associated with the use, or sequelae of use, of cocaine or other psychomotor stimulants |
| DE19802327A1 (de) * | 1998-01-23 | 1999-07-29 | Goedecke Ag | Synergistische Arzneimittelzubereitung mit analgetischer Wirkung |
| EP1161263A1 (en) * | 1999-03-10 | 2001-12-12 | Warner-Lambert Company Llc | Analgesic compositions comprising anti-epileptic compounds and methods of using same |
-
2000
- 2000-06-21 EP EP00943001A patent/EP1196160B1/en not_active Expired - Lifetime
- 2000-06-21 AT AT00943001T patent/ATE313322T1/de not_active IP Right Cessation
- 2000-06-21 ES ES00943001T patent/ES2255500T3/es not_active Expired - Lifetime
- 2000-06-21 BR BR0012058-8A patent/BR0012058A/pt not_active Application Discontinuation
- 2000-06-21 WO PCT/US2000/017039 patent/WO2001001983A1/en not_active Ceased
- 2000-06-21 JP JP2001507475A patent/JP2003503453A/ja not_active Abandoned
- 2000-06-21 MX MXPA02000170A patent/MXPA02000170A/es active IP Right Grant
- 2000-06-21 CA CA002373953A patent/CA2373953A1/en not_active Abandoned
- 2000-06-21 DE DE60024995T patent/DE60024995T2/de not_active Expired - Fee Related
- 2000-06-21 AU AU57539/00A patent/AU5753900A/en not_active Abandoned
- 2000-06-28 PE PE2000000651A patent/PE20010331A1/es not_active Application Discontinuation
- 2000-06-30 CO CO00049385A patent/CO5210869A1/es not_active Application Discontinuation
- 2000-06-30 AR ARP000103359A patent/AR030024A1/es unknown
- 2000-06-30 UY UY26230A patent/UY26230A1/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| MXPA02000170A (es) | 2002-07-02 |
| AU5753900A (en) | 2001-01-22 |
| CO5210869A1 (es) | 2002-10-30 |
| CA2373953A1 (en) | 2001-01-11 |
| ES2255500T3 (es) | 2006-07-01 |
| UY26230A1 (es) | 2001-03-16 |
| DE60024995T2 (de) | 2006-06-22 |
| JP2003503453A (ja) | 2003-01-28 |
| EP1196160B1 (en) | 2005-12-21 |
| DE60024995D1 (de) | 2006-01-26 |
| EP1196160A1 (en) | 2002-04-17 |
| PE20010331A1 (es) | 2001-03-22 |
| AR030024A1 (es) | 2003-08-13 |
| ATE313322T1 (de) | 2006-01-15 |
| WO2001001983A1 (en) | 2001-01-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B06A | Patent application procedure suspended [chapter 6.1 patent gazette] | ||
| B11B | Dismissal acc. art. 36, par 1 of ipl - no reply within 90 days to fullfil the necessary requirements |