BG27902A3 - Метод за получаване на n-(метокси-метил-фуриметил)-6,7-бензоморфани и морфипани - Google Patents
Метод за получаване на n-(метокси-метил-фуриметил)-6,7-бензоморфани и морфипаниInfo
- Publication number
- BG27902A3 BG27902A3 BG028037A BG2803774A BG27902A3 BG 27902 A3 BG27902 A3 BG 27902A3 BG 028037 A BG028037 A BG 028037A BG 2803774 A BG2803774 A BG 2803774A BG 27902 A3 BG27902 A3 BG 27902A3
- Authority
- BG
- Bulgaria
- Prior art keywords
- benzomorphanes
- morphipanes
- furimethyl
- methoxy
- methyl
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
Landscapes
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Organic Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Other In-Based Heterocyclic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Метод за получаване на охарактеризирани и доказани в описанието n-(метоксиметил-фурилметил)-6, 7-бензоморфани и -морфинани с обща формула........ Патентните претенции са формулирани в 2 точки
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE19732354002 DE2354002A1 (de) | 1973-10-27 | 1973-10-27 | Neue n-(methoxymethyl-furylmethyl)6,7-benzomorphane und -morphinane, deren saeureadditionssalze, ihre verwendung als arzneimittel und verfahren zu deren herstellung |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BG27902A3 true BG27902A3 (bg) | 1980-01-15 |
Family
ID=5896658
Family Applications (3)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG028036A BG27901A3 (bg) | 1973-10-27 | 1974-10-25 | Метод за получаване на n-(метокси-метил-фурил-метил)-6-7-бензоморфани и бензоморфинапи |
| BG028037A BG27902A3 (bg) | 1973-10-27 | 1974-10-25 | Метод за получаване на n-(метокси-метил-фуриметил)-6,7-бензоморфани и морфипани |
| BG028038A BG27903A3 (bg) | 1973-10-27 | 1974-10-25 | Метод за получаване на n-(метокси-метил-фурилметил)-6,7-бензоморфани и морфипани и техните присъединителни с киселина соли |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG028036A BG27901A3 (bg) | 1973-10-27 | 1974-10-25 | Метод за получаване на n-(метокси-метил-фурил-метил)-6-7-бензоморфани и бензоморфинапи |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BG028038A BG27903A3 (bg) | 1973-10-27 | 1974-10-25 | Метод за получаване на n-(метокси-метил-фурилметил)-6,7-бензоморфани и морфипани и техните присъединителни с киселина соли |
Country Status (27)
| Country | Link |
|---|---|
| US (1) | US3981874A (bg) |
| JP (1) | JPS5738590B2 (bg) |
| AT (6) | AT335634B (bg) |
| BE (1) | BE821505A (bg) |
| BG (3) | BG27901A3 (bg) |
| CA (1) | CA1056377A (bg) |
| CH (6) | CH609340A5 (bg) |
| CS (3) | CS171195B2 (bg) |
| DD (1) | DD115909A5 (bg) |
| DE (1) | DE2354002A1 (bg) |
| DK (1) | DK138325C (bg) |
| ES (6) | ES431056A1 (bg) |
| FI (1) | FI62079C (bg) |
| FR (1) | FR2248838B1 (bg) |
| GB (1) | GB1482552A (bg) |
| HU (1) | HU176479B (bg) |
| IE (1) | IE41528B1 (bg) |
| IL (1) | IL45938A (bg) |
| NL (1) | NL7413980A (bg) |
| NO (1) | NO140859C (bg) |
| PH (1) | PH11894A (bg) |
| PL (3) | PL92086B1 (bg) |
| RO (5) | RO65656A (bg) |
| SE (1) | SE422791B (bg) |
| SU (6) | SU510999A3 (bg) |
| YU (5) | YU36949B (bg) |
| ZA (1) | ZA746790B (bg) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1513961A (en) * | 1975-02-25 | 1978-06-14 | Acf Chemiefarma Nv | 6,7-benzomorphans method for their preparation and intermediates |
| US4208523A (en) * | 1978-11-30 | 1980-06-17 | Sterling Drug Inc. | 11-Lower-alkyl-, 11-phenyl-lower-alkyl- and 11-cyclo-lower-alkyl-lower-alkyl-hexahydro-2,6-methano-3-benzazocines |
| EP2183229B1 (en) | 2007-07-26 | 2012-04-18 | Vitae Pharmaceuticals, Inc. | Synthesis of inhibitors of 11beta-hydroxysteroid dehydrogenase type 1 |
| TW200927115A (en) * | 2007-11-16 | 2009-07-01 | Boehringer Ingelheim Int | Aryl-and heteroarylcarbonyl derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| WO2009075835A1 (en) | 2007-12-11 | 2009-06-18 | Vitae Pharmaceutical, Inc | CYCLIC UREA INHIBITORS OF 11β-HYDROXYSTEROID DEHYDROGENASE 1 |
| TW200934490A (en) | 2008-01-07 | 2009-08-16 | Vitae Pharmaceuticals Inc | Lactam inhibitors of 11 &abgr;-hydroxysteroid dehydrogenase 1 |
| WO2009094169A1 (en) | 2008-01-24 | 2009-07-30 | Vitae Pharmaceuticals, Inc. | Cyclic carbazate and semicarbazide inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| EP2245014B1 (en) * | 2008-02-12 | 2011-11-02 | Boehringer Ingelheim International GmbH | Urea derivatives of benzomorphanes and related scaffolds, medicaments containing such compounds and their use |
| US8598160B2 (en) | 2008-02-15 | 2013-12-03 | Vitae Pharmaceuticals, Inc. | Cycloalkyl lactame derivatives as inhibitors of 11-beta-hydroxysteroid dehydrogenase 1 |
| ES2421537T3 (es) | 2008-05-01 | 2013-09-03 | Vitae Pharmaceuticals Inc | Inhibidores cíclicos de la 11beta-hidroxiesteroide deshidrogenasa 1 |
| CA2723034A1 (en) | 2008-05-01 | 2009-11-05 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| CA2723039A1 (en) | 2008-05-01 | 2009-11-05 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| JP5711115B2 (ja) | 2008-05-13 | 2015-04-30 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | ベンゾモルファン及び関連骨格のアリサイクリックカルボン酸誘導体、そのような化合物を含有する医薬及びその使用 |
| US8846668B2 (en) | 2008-07-25 | 2014-09-30 | Vitae Pharmaceuticals, Inc. | Inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| DK2324018T3 (da) | 2008-07-25 | 2013-10-14 | Boehringer Ingelheim Int | Cykliske inhibitorer af 11 beta-hydroxysteroid dehydrogenase 1 |
| US8680093B2 (en) | 2009-04-30 | 2014-03-25 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 |
| EP2440537A1 (en) | 2009-06-11 | 2012-04-18 | Vitae Pharmaceuticals, Inc. | Cyclic inhibitors of 11beta-hydroxysteroid dehydrogenase 1 based on the 1,3 -oxazinan- 2 -one structure |
| TWI531571B (zh) | 2009-11-06 | 2016-05-01 | 維它藥物公司 | 六氫茚并吡啶及八氫苯并喹啉之芳基－及雜芳基羰基衍生物 |
| WO2011159760A1 (en) | 2010-06-16 | 2011-12-22 | Vitae Pharmaceuticals, Inc. | Substituted 5-,6- and 7-membered heterocycles, medicaments containing such compounds, and their use |
| TWI537258B (zh) | 2010-11-05 | 2016-06-11 | 百靈佳殷格翰國際股份有限公司 | 六氫茚并吡啶及八氫苯并喹啉之芳基－及雜環芳基羰基衍生物 |
| JP2014524438A (ja) | 2011-08-17 | 2014-09-22 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | インデノピリジン誘導体 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3632591A (en) * | 1968-07-19 | 1972-01-04 | Sterling Drug Inc | 1 2 3 4 5 6 - hexahydro-3-(cycloaliphatic or cycloaliphatic 11-dimethyl-2 alkyl)-66-methano-3-benzazocines |
| US3833595A (en) * | 1968-12-26 | 1974-09-03 | Sumitomo Chemical Co | 2-aroylalkyl benzomorphans |
| CS166803B2 (bg) * | 1971-02-08 | 1976-03-29 | Boehringer Sohn Ingelheim |
-
1973
- 1973-10-25 SU SU2069684A patent/SU510999A3/ru active
- 1973-10-25 SU SU2069691A patent/SU511005A3/ru active
- 1973-10-27 DE DE19732354002 patent/DE2354002A1/de not_active Withdrawn
-
1974
- 1974-01-25 RO RO7480315A patent/RO65656A/ro unknown
- 1974-10-02 CS CS6768A patent/CS171195B2/cs unknown
- 1974-10-02 CS CS6767A patent/CS171194B2/cs unknown
- 1974-10-02 CS CS6769A patent/CS171196B2/cs unknown
- 1974-10-15 US US05/514,474 patent/US3981874A/en not_active Expired - Lifetime
- 1974-10-16 AT AT829074A patent/AT335634B/de not_active IP Right Cessation
- 1974-10-16 ES ES431056A patent/ES431056A1/es not_active Expired
- 1974-10-16 ES ES431058A patent/ES431058A1/es not_active Expired
- 1974-10-16 AT AT828974A patent/AT336202B/de not_active IP Right Cessation
- 1974-10-16 AT AT828774A patent/AT335633B/de not_active IP Right Cessation
- 1974-10-16 AT AT828574A patent/AT335631B/de not_active IP Right Cessation
- 1974-10-16 ES ES431057A patent/ES431057A1/es not_active Expired
- 1974-10-16 ES ES431054A patent/ES431054A1/es not_active Expired
- 1974-10-16 AT AT828874A patent/AT335076B/de active
- 1974-10-16 ES ES431055A patent/ES431055A1/es not_active Expired
- 1974-10-16 ES ES431059A patent/ES431059A1/es not_active Expired
- 1974-10-16 AT AT828674A patent/AT335632B/de not_active IP Right Cessation
- 1974-10-24 YU YU2854/74A patent/YU36949B/xx unknown
- 1974-10-24 YU YU2851/74A patent/YU36951B/xx unknown
- 1974-10-24 CH CH1426574A patent/CH609340A5/xx not_active IP Right Cessation
- 1974-10-24 CH CH1426274A patent/CH609046A5/xx not_active IP Right Cessation
- 1974-10-24 CH CH1426474A patent/CH609048A5/xx not_active IP Right Cessation
- 1974-10-24 CH CH1426374A patent/CH609047A5/xx not_active IP Right Cessation
- 1974-10-24 YU YU02852/74A patent/YU36519B/xx unknown
- 1974-10-24 YU YU2853/74A patent/YU36952B/xx unknown
- 1974-10-24 PH PH16448A patent/PH11894A/en unknown
- 1974-10-24 YU YU2856/74A patent/YU36950B/xx unknown
- 1974-10-25 RO RO7480314A patent/RO65655A/ro unknown
- 1974-10-25 NO NO743845A patent/NO140859C/no unknown
- 1974-10-25 BG BG028036A patent/BG27901A3/bg unknown
- 1974-10-25 BE BE149902A patent/BE821505A/xx not_active IP Right Cessation
- 1974-10-25 CH CH1437074A patent/CH609686A5/xx not_active IP Right Cessation
- 1974-10-25 IL IL45938A patent/IL45938A/en unknown
- 1974-10-25 SU SU2070657A patent/SU508193A3/ru active
- 1974-10-25 NL NL7413980A patent/NL7413980A/xx unknown
- 1974-10-25 RO RO7480317A patent/RO65658A/ro unknown
- 1974-10-25 FI FI3141/74A patent/FI62079C/fi active
- 1974-10-25 GB GB46323/74A patent/GB1482552A/en not_active Expired
- 1974-10-25 ZA ZA00746790A patent/ZA746790B/xx unknown
- 1974-10-25 IE IE2206/74A patent/IE41528B1/en unknown
- 1974-10-25 CA CA212,340A patent/CA1056377A/en not_active Expired
- 1974-10-25 JP JP12261074A patent/JPS5738590B2/ja not_active Expired
- 1974-10-25 DK DK559874A patent/DK138325C/da not_active IP Right Cessation
- 1974-10-25 HU HU74BO1521A patent/HU176479B/hu unknown
- 1974-10-25 RO RO7480318A patent/RO65659A/ro unknown
- 1974-10-25 BG BG028037A patent/BG27902A3/bg unknown
- 1974-10-25 SE SE7413485A patent/SE422791B/xx unknown
- 1974-10-25 SU SU2069689A patent/SU508192A3/ru active
- 1974-10-25 RO RO7480316A patent/RO65657A/ro unknown
- 1974-10-25 BG BG028038A patent/BG27903A3/bg unknown
- 1974-10-25 SU SU2070713A patent/SU512707A3/ru active
- 1974-10-25 SU SU7402069685A patent/SU578870A3/ru active
- 1974-10-25 FR FR7435890A patent/FR2248838B1/fr not_active Expired
- 1974-10-25 DD DD181929A patent/DD115909A5/xx unknown
- 1974-10-25 CH CH1436974A patent/CH609685A5/xx not_active IP Right Cessation
- 1974-10-26 PL PL1974175144A patent/PL92086B1/pl unknown
- 1974-10-26 PL PL1974175142A patent/PL92053B1/pl unknown
- 1974-10-26 PL PL1974175143A patent/PL92052B1/pl unknown
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