BG26526A3 - METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES - Google Patents

METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES

Info

Publication number: BG26526A3
Authority: BG; Bulgaria
Prior art keywords: benzazolylalkyl; preparation; piperidine derivatives; piperidine; derivatives
Prior art date: 1975-07-21

Application number

BG033791A

Other languages

Bulgarian (bg)

Inventor

Jan Vandenberk

Ludo Edmond Kennis

Marcel Van

Albert M.

Original Assignee

Неизвестен

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1975-07-21

Filing date

1976-07-20

Publication date

1979-04-12

1976-05-17 Priority claimed from US05/687,139 external-priority patent/US4066772A/en

1976-07-20 Application filed by Неизвестен filed Critical Неизвестен

1979-04-12 Publication of BG26526A3 publication Critical patent/BG26526A3/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
- C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D211/36—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D211/56—Nitrogen atoms
- C07D211/58—Nitrogen atoms attached in position 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Hospice & Palliative Care (AREA)
Otolaryngology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Hydrogenated Pyridines (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

BG033791A 1975-07-21 1976-07-20 METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES BG26526A3 (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US59779375A	1975-07-21	1975-07-21
US05/687,139 US4066772A (en)	1975-07-21	1976-05-17	1,3-Dihydro-1-[3-(1-piperidinyl)propyl]-2H-benzimidazol-2-ones and related compounds
KR7601697A KR810000334B1 (en)	1975-07-21	1976-07-12	Process for preparation 1-(benzazolylalkyl)-piperidine derivatives

Publications (1)

Publication Number	Publication Date
BG26526A3 true BG26526A3 (en)	1979-04-12

Family

ID=27348142

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BG033791A BG26526A3 (en)	1975-07-21	1976-07-20	METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES

Country Status (25)

Country	Link
JP (1)	JPS5217475A (en)
AT (1)	AT364358B (en)
AU (1)	AU511027B2 (en)
BG (1)	BG26526A3 (en)
CA (1)	CA1085852A (en)
CH (1)	CH623820A5 (en)
CS (1)	CS202550B2 (en)
DE (1)	DE2632870A1 (en)
DK (1)	DK154950C (en)
ES (3)	ES449740A1 (en)
FI (1)	FI62667C (en)
GB (1)	GB1542514A (en)
HK (1)	HK14180A (en)
IE (1)	IE43496B1 (en)
IT (1)	IT1062614B (en)
KE (1)	KE3215A (en)
LU (1)	LU75354A1 (en)
MY (1)	MY8100017A (en)
NL (1)	NL187442C (en)
NZ (1)	NZ181256A (en)
PH (1)	PH13710A (en)
PT (1)	PT65387B (en)
RO (1)	RO70566A (en)
SE (2)	SE426490B (en)
YU (1)	YU39969B (en)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4501749A (en) *	1983-10-31	1985-02-26	Merck & Co., Inc.	Peripherally selective dopamine antagonists in the treatment of ocular hypertension
JPS6248684A (en) *	1985-08-26	1987-03-03	Sumitomo Chem Co Ltd	Novel iodobutyrophenone derivative and production thereof
JPS62251313A (en) *	1986-04-25	1987-11-02	信越ポリマー株式会社	Bundling device
US6355659B1 (en)	1994-07-29	2002-03-12	Laboratorios Del Dr. Esteve, S.A.	4-(4-Chlorophenyl)-1236-tetrahydro-1(1H-124-triazol-1-yl)butty)pyrideine and salts thereof; pharmaceutical compositions and method of treating psychoses utilizing same
FR2723091B1 (en) *	1994-07-29	1996-11-08	Esteve Labor Dr	TETRAHYDROPYRIDINE- (6,4-HYDROXYPIPERIDINE) ALKYLAZOLES
RU2192848C1 (en) *	2001-10-30	2002-11-20	Закрытое акционерное общество "ВЕРОФАРМ"	Antiemetic remedy
PA8603801A1 (en) *	2003-05-27	2004-12-16	Janssen Pharmaceutica Nv	DERIVATIVES OF QUINAZOLINE
RU2268047C2 (en) *	2003-12-15	2006-01-20	Закрытое акционерное общество "Фармацевтическое предприятие "Оболенское"	Medicinal formulation possessing anti-vomiting effect and method for its preparing
WO2005058913A1 (en)	2003-12-18	2005-06-30	Janssen Pharmaceutica N.V.	Pyrido- and pyrimidopyrimidine derivatives as anti- proliferative agents
NI200700147A (en)	2004-12-08	2019-05-10	Janssen Pharmaceutica Nv	QUINAZOLINE DERIVATIVES KINE INHIBITORS TARGETING MULTIP
AU2007274284B2 (en)	2006-07-13	2012-04-26	Janssen Pharmaceutica N.V.	Mtki quinazoline derivatives
EP1997805A1 (en) *	2007-06-01	2008-12-03	Commissariat à l'Energie Atomique	Compounds with antiparasitic activity, applications thereof to the treatment of infectious diseases caused by apicomplexans
ES2562218T3 (en)	2007-07-27	2016-03-03	Janssen Pharmaceutica, N.V.	Pyrrolopyrimidines useful for the treatment of proliferative diseases
EP2433935A1 (en)	2007-08-31	2012-03-28	Purdue Pharma LP	Substituted-quinoxaline-type-piperidine compounds and the uses thereof
WO2014102594A2 (en)	2012-12-27	2014-07-03	Purdue Pharma L.P.	Substituted benzimidazole-type piperidine compounds and uses thereof
CN108697700B (en) *	2016-02-04	2021-08-17	辛多美制药有限公司	Deuterated domperidone composition and method for treating disorders
KR20240125702A (en)	2017-06-30	2024-08-19	신돔 파마, 인크.	Deuterated domperidone compositions, methods, and preparation
US12478612B2 (en)	2017-06-30	2025-11-25	Cindome Pharma, Inc.	Deuterated domperidone compositions, methods, and preparation

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
BE633495A (en) *	1962-06-13
BE633914A (en) *	1962-06-22
US3629267A (en) *	1968-10-28	1971-12-21	Smith Kline French Lab	Benzoheterocyclicalkyl derivatives of 4-(2-keto -1-benzimidazolinyl)-piperidine 4-(2-keto - 1 - benzimidazolinyl) -1 2 3 6 tetrahydropyridine 1 - phenyl - 1 3 8-triazaspiro(4 5)decan - 4 - one and 2 4 9-triazaspiro(5 5)undecan-1 3 5-trione
AU4698672A (en) *	1972-09-22	1972-11-09	Ciba-Geigy Ag	Azacycloaliphatic compounds, process for their manufacture and compositions containing them
FR2218100A1 (en) *	1973-02-20	1974-09-13	Janssen Pharmaceutica Nv	Neuroleptic tricyclic derivs. - of benzimidazolinones and triazaspiro-4,5-decan-4-ones
US3989707A (en) *	1974-06-21	1976-11-02	Janssen Pharmaceutica N.V.	Benzimidazolinone derivatives

1976
- 1976-06-23 NZ NZ181256A patent/NZ181256A/en unknown
- 1976-06-30 GB GB7627242A patent/GB1542514A/en not_active Expired
- 1976-07-07 RO RO7686860A patent/RO70566A/en unknown
- 1976-07-07 CA CA256,450A patent/CA1085852A/en not_active Expired
- 1976-07-08 PH PH18663A patent/PH13710A/en unknown
- 1976-07-09 LU LU75354A patent/LU75354A1/xx unknown
- 1976-07-09 ES ES449740A patent/ES449740A1/en not_active Expired
- 1976-07-16 AU AU15964/76A patent/AU511027B2/en not_active Expired
- 1976-07-16 CS CS764688A patent/CS202550B2/en unknown
- 1976-07-19 JP JP51085216A patent/JPS5217475A/en active Granted
- 1976-07-19 IT IT50499/76A patent/IT1062614B/en active
- 1976-07-20 IE IE1602/76A patent/IE43496B1/en not_active IP Right Cessation
- 1976-07-20 CH CH929176A patent/CH623820A5/en not_active IP Right Cessation
- 1976-07-20 BG BG033791A patent/BG26526A3/en unknown
- 1976-07-20 FI FI762086A patent/FI62667C/en not_active IP Right Cessation
- 1976-07-20 AT AT0534776A patent/AT364358B/en not_active IP Right Cessation
- 1976-07-20 DK DK327576A patent/DK154950C/en not_active IP Right Cessation
- 1976-07-20 SE SE7608265A patent/SE426490B/en not_active IP Right Cessation
- 1976-07-20 NL NLAANVRAGE7608023,A patent/NL187442C/en not_active IP Right Cessation
- 1976-07-20 PT PT65387A patent/PT65387B/en unknown
- 1976-07-21 YU YU1794/76A patent/YU39969B/en unknown
- 1976-07-21 DE DE19762632870 patent/DE2632870A1/en active Granted
1977
- 1977-08-16 ES ES461631A patent/ES461631A1/en not_active Expired
- 1977-08-16 ES ES461630A patent/ES461630A1/en not_active Expired
1980
- 1980-03-20 HK HK141/80A patent/HK14180A/en unknown
- 1980-12-11 SE SE8008713A patent/SE435621B/en not_active IP Right Cessation
1981
- 1981-12-30 MY MY17/81A patent/MY8100017A/en unknown
1982
- 1982-05-21 KE KE3215A patent/KE3215A/en unknown

Also Published As

Publication number	Publication date
PH13710A (en)	1980-09-09
DK327576A (en)	1977-01-22
DE2632870A1 (en)	1977-02-10
AU1596476A (en)	1978-01-19
FI762086A7 (en)	1977-01-22
CS202550B2 (en)	1981-01-30
ES449740A1 (en)	1978-02-16
KE3215A (en)	1982-07-09
DE2632870C2 (en)	1989-02-16
DK154950C (en)	1989-05-29
ATA534776A (en)	1981-03-15
MY8100017A (en)	1981-12-31
AT364358B (en)	1981-10-12
SE435621B (en)	1984-10-08
JPS5217475A (en)	1977-02-09
YU39969B (en)	1985-06-30
IE43496L (en)	1977-01-21
RO70566A (en)	1982-10-11
DK154950B (en)	1989-01-09
SE426490B (en)	1983-01-24
NZ181256A (en)	1978-04-28
CA1085852A (en)	1980-09-16
HK14180A (en)	1980-03-28
YU179476A (en)	1983-01-21
JPS6131109B2 (en)	1986-07-17
PT65387A (en)	1976-08-01
ES461630A1 (en)	1978-06-16
PT65387B (en)	1978-06-09
NL187442C (en)	1991-10-01
IE43496B1 (en)	1981-03-11
NL187442B (en)	1991-05-01
AU511027B2 (en)	1980-07-24
FI62667B (en)	1982-10-29
LU75354A1 (en)	1977-02-28
IT1062614B (en)	1984-10-20
SE7608265L (en)	1977-01-22
SE8008713L (en)	1980-12-11
ES461631A1 (en)	1978-12-01
GB1542514A (en)	1979-03-21
NL7608023A (en)	1977-01-25
FI62667C (en)	1983-02-10
CH623820A5 (en)	1981-06-30

Publication	Publication Date	Title
SE437022B (en)	1985-02-04	PROCEDURE FOR THE PREPARATION OF N-SUBSTITUTED MORPHOLINE DERIVATIVES RESPECTIVE PIPERIDINE DERIVATIVES
SE434049B (en)	1984-07-02	PROCEDURE FOR PREPARING 1,4-DIHYDROPYRIDINE DERIVATIVES
BG27380A3 (en)	1979-10-12	METHOD FOR OBTAINING ERYTHROMYCYLAMINE DERIVATIVES
BG24673A3 (en)	1978-04-12	METHOD FOR OBTAINING QUINAZOLONE DERIVATIVES
ZA764322B (en)	1978-03-29	Novel 1-(benzazolyalkyl)piperidine derivatives
BG26515A3 (en)	1979-04-12	METHOD FOR OBTAINING ACYLAMINO DERIVATIVES
BG26526A3 (en)	1979-04-12	METHOD FOR THE PREPARATION OF 1-(BENZAZOLYLALKYL)PIPERIDINE DERIVATIVES
BG27362A3 (en)	1979-10-12	METHOD FOR OBTAINING N-PHENYL-N-BENZOYL-UREAS
BG26518A3 (en)	1979-04-12	METHOD FOR OBTAINING PHENYL-ALKANE DERIVATIVES
BG25517A3 (en)	1978-10-10	METHOD FOR OBTAINING IMIDAZOLE DERIVATIVES
BG27542A3 (en)	1979-11-12	METHOD FOR THE PREPARATION OF 1-BENZAZOLYLALKYL-4-SUBSTITUTED PIPERIDINES
BG25074A3 (en)	1978-07-12	METHOD FOR PREPARING SUBSTITUTED PERHALOALKYLAMIDINES
BG27368A3 (en)	1979-10-12	METHOD FOR OBTAINING SUBSTITUTED PYRIDINES
BG24810A3 (en)	1978-05-12	METHOD FOR OBTAINING BENZIZYTHIAZONES
BG24799A3 (en)	1978-05-12	METHOD FOR OBTAINING BENZOYLUREIDO-DIPHENYLETHERS
SE433745B (en)	1984-06-12	PROCEDURE FOR PREPARING TETRAHYDROISOKINOLIN DERIVATIVES
BG27355A3 (en)	1979-10-12	METHOD FOR THE PREPARATION OF 11-DESOXY-16-ARYLOXY-W-TETRANORPROSTAGLANDINS
BG27543A3 (en)	1979-11-12	METHOD FOR THE PREPARATION OF N-ARYL-N-(1-L-4-PIPERIDINYL)- ARYLACET-AMIDES
MX4118E (en)	1981-12-14	PROCEDURE FOR PREPARING PIPERIDINE COMPOUND
BG27359A3 (en)	1979-10-12	METHOD FOR OBTAINING ACYLAMINE DERIVATIVES
SE423902B (en)	1982-06-14	PROCEDURE FOR PURINATE DERIVATIVES
BG24801A3 (en)	1978-05-12	METHOD FOR OBTAINING L-PYROGLUTAMYLL-PROLINAMIDE
BG27361A3 (en)	1979-10-12	METHOD FOR OBTAINING SUBSTITUTED UREA DERIVATIVES
BG26535A3 (en)	1979-04-12	METHOD FOR OBTAINING INDOLQUINOLYSINES
RO73050A (en)	1981-08-30	PROCESS FOR PREPARATION OF SUBSTITUTED AMINOCHINESOLINE DERIVATIVES