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BG108426A - Novel sulfonic acid derivatives - Google Patents

Novel sulfonic acid derivatives

Info

Publication number
BG108426A
BG108426A BG108426A BG10842603A BG108426A BG 108426 A BG108426 A BG 108426A BG 108426 A BG108426 A BG 108426A BG 10842603 A BG10842603 A BG 10842603A BG 108426 A BG108426 A BG 108426A
Authority
BG
Bulgaria
Prior art keywords
sulfonic acid
acid derivatives
novel sulfonic
novel
compound
Prior art date
Application number
BG108426A
Other languages
Bulgarian (bg)
English (en)
Inventor
Matthew Hayward
Original Assignee
Pfizer Products Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Products Inc. filed Critical Pfizer Products Inc.
Publication of BG108426A publication Critical patent/BG108426A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/04—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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    • A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
    • C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
    • C07D295/182—Radicals derived from carboxylic acids
    • C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers

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  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
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  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
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  • Communicable Diseases (AREA)
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  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Diabetes (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Neurology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Neurosurgery (AREA)
  • Hematology (AREA)
  • Vascular Medicine (AREA)
  • Pain & Pain Management (AREA)
  • AIDS & HIV (AREA)
  • Hospice & Palliative Care (AREA)
  • Biomedical Technology (AREA)
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BG108426A 2001-06-20 2003-12-08 Novel sulfonic acid derivatives BG108426A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US29946101P 2001-06-20 2001-06-20

Publications (1)

Publication Number Publication Date
BG108426A true BG108426A (en) 2005-01-31

Family

ID=23154893

Family Applications (1)

Application Number Title Priority Date Filing Date
BG108426A BG108426A (en) 2001-06-20 2003-12-08 Novel sulfonic acid derivatives

Country Status (35)

Country Link
US (2) US6974817B2 (xx)
EP (1) EP1430041A2 (xx)
JP (2) JP3829136B2 (xx)
KR (1) KR20040012956A (xx)
CN (1) CN1529699A (xx)
AP (1) AP1564A (xx)
AR (1) AR036094A1 (xx)
BG (1) BG108426A (xx)
BR (1) BR0210531A (xx)
CA (1) CA2447865C (xx)
CZ (1) CZ20033455A3 (xx)
DO (1) DOP2002000399A (xx)
EA (1) EA006447B1 (xx)
EC (1) ECSP034917A (xx)
EE (1) EE200400023A (xx)
GT (1) GT200200095A (xx)
HR (1) HRP20030834A2 (xx)
HU (1) HUP0400369A2 (xx)
IL (1) IL158461A0 (xx)
IS (1) IS6987A (xx)
MA (1) MA27033A1 (xx)
MX (1) MXPA03011954A (xx)
NO (1) NO20035694D0 (xx)
OA (1) OA12623A (xx)
PA (1) PA8548501A1 (xx)
PE (1) PE20030127A1 (xx)
PL (1) PL366900A1 (xx)
SK (1) SK15722003A3 (xx)
SV (1) SV2003001099A (xx)
TN (1) TNSN03140A1 (xx)
UA (1) UA74266C2 (xx)
UY (1) UY27338A1 (xx)
WO (1) WO2002102787A2 (xx)
YU (1) YU94103A (xx)
ZA (1) ZA200307736B (xx)

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CZ20033455A3 (en) * 2001-06-20 2004-06-16 Pfizer Products Inc. Novel sulfonic acid derivatives
US7456184B2 (en) * 2003-05-01 2008-11-25 Palatin Technologies Inc. Melanocortin receptor-specific compounds
US7732451B2 (en) * 2001-08-10 2010-06-08 Palatin Technologies, Inc. Naphthalene-containing melanocortin receptor-specific small molecule
US7718802B2 (en) 2001-08-10 2010-05-18 Palatin Technologies, Inc. Substituted melanocortin receptor-specific piperazine compounds
US7354923B2 (en) * 2001-08-10 2008-04-08 Palatin Technologies, Inc. Piperazine melanocortin-specific compounds
JP2005504043A (ja) * 2001-08-10 2005-02-10 パラチン テクノロジーズ インク． 生物学的に活性な金属ペプチド類のペプチド模倣体類
US7655658B2 (en) * 2001-08-10 2010-02-02 Palatin Technologies, Inc. Thieno [2,3-D]pyrimidine-2,4-dione melanocortin-specific compounds
US20040116441A1 (en) * 2002-10-30 2004-06-17 Pfizer Inc Methods of using sulfonic acid derivatives
MXPA05009771A (es) 2003-03-14 2005-10-26 Ono Pharmaceutical Co Derivados heterociclicos que contienen nitrogeno y medicamentos que los contienen como el ingrediente activo.
US7727990B2 (en) 2003-05-01 2010-06-01 Palatin Technologies, Inc. Melanocortin receptor-specific piperazine and keto-piperazine compounds
US7727991B2 (en) 2003-05-01 2010-06-01 Palatin Technologies, Inc. Substituted melanocortin receptor-specific single acyl piperazine compounds
US7968548B2 (en) 2003-05-01 2011-06-28 Palatin Technologies, Inc. Melanocortin receptor-specific piperazine compounds with diamine groups
US20050119275A1 (en) * 2003-06-24 2005-06-02 Pfizer Inc. Salt and crystal forms of (5-chloro-2-{2-[4-(4-fluoro-benzyl)-(2R,5S)-2,5-dimethyl-piperazin-1-yl]-2-oxo-ethoxy}-phenyl)-methanesulfonic acid
US7709484B1 (en) 2004-04-19 2010-05-04 Palatin Technologies, Inc. Substituted melanocortin receptor-specific piperazine compounds
US8188277B2 (en) 2004-08-06 2012-05-29 Otsuka Pharmaceutical Co., Ltd. Aromatic compounds for suppressing the generation of collagen
SG146673A1 (en) 2004-09-13 2008-10-30 Ono Pharmaceutical Co Nitrogenous heterocyclic derivative and medicine containing the same as an active ingredient
MY146514A (en) 2005-12-05 2012-08-15 Otsuka Pharma Co Ltd Diarylether derivatives as antitumor agents
WO2007105637A1 (ja) 2006-03-10 2007-09-20 Ono Pharmaceutical Co., Ltd. 含窒素複素環誘導体およびそれらを有効成分とする薬剤
US7834017B2 (en) 2006-08-11 2010-11-16 Palatin Technologies, Inc. Diamine-containing, tetra-substituted piperazine compounds having identical 1- and 4-substituents
UA95978C2 (xx) 2006-10-02 2011-09-26 Оцука Фармас'Ютікел Ко., Лтд. Інгібітор активації stat3/5$ингибитор активации stat3/5
US8716235B2 (en) * 2012-04-18 2014-05-06 Albert Einstein College Of Medicine Of Yeshiva University Method for inhibiting metastasis by using anti-CCL3 antibodies
FR3029112A1 (fr) * 2014-12-02 2016-06-03 Pf Medicament Dispersion solide a base de derives d'heteroarylsulfonamides a usage pharmaceutique

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CZ20033455A3 (en) * 2001-06-20 2004-06-16 Pfizer Products Inc. Novel sulfonic acid derivatives

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OA12623A (en) 2006-06-12
GT200200095A (es) 2003-02-27
AP2002002560A0 (en) 2002-06-30
JP3829136B2 (ja) 2006-10-04
WO2002102787A2 (en) 2002-12-27
IL158461A0 (en) 2004-05-12
KR20040012956A (ko) 2004-02-11
US20030083335A1 (en) 2003-05-01
HUP0400369A2 (hu) 2004-12-28
ECSP034917A (es) 2004-02-26
CN1529699A (zh) 2004-09-15
TNSN03140A1 (fr) 2005-12-23
JP2006232846A (ja) 2006-09-07
JP2005511486A (ja) 2005-04-28
CZ20033455A3 (en) 2004-06-16
CA2447865A1 (en) 2002-12-27
SV2003001099A (es) 2003-03-18
CA2447865C (en) 2010-07-20
EP1430041A2 (en) 2004-06-23
AP1564A (en) 2006-02-02
UA74266C2 (uk) 2005-11-15
EA006447B1 (ru) 2005-12-29
PE20030127A1 (es) 2003-02-22
PA8548501A1 (es) 2003-05-14
EE200400023A (et) 2004-06-15
ZA200307736B (en) 2004-10-04
HRP20030834A2 (en) 2004-08-31
PL366900A1 (en) 2005-02-07
UY27338A1 (es) 2003-10-31
YU94103A (sh) 2006-03-03
US20050250790A1 (en) 2005-11-10
SK15722003A3 (sk) 2004-08-03
MXPA03011954A (es) 2004-03-26
AR036094A1 (es) 2004-08-11
MA27033A1 (fr) 2004-12-20
BR0210531A (pt) 2004-06-22
DOP2002000399A (es) 2002-12-30
EA200301276A1 (ru) 2004-04-29
IS6987A (is) 2003-10-09
WO2002102787A3 (en) 2004-04-29
NO20035694D0 (no) 2003-12-19
US6974817B2 (en) 2005-12-13

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