BE884848A - Sel mixte d'acide valproique utile notamment pour le traitement de l'epilepsie, presentant des caracteristiques tres superieures de stabilite - Google Patents
Sel mixte d'acide valproique utile notamment pour le traitement de l'epilepsie, presentant des caracteristiques tres superieures de stabiliteInfo
- Publication number
- BE884848A BE884848A BE0/201805A BE201805A BE884848A BE 884848 A BE884848 A BE 884848A BE 0/201805 A BE0/201805 A BE 0/201805A BE 201805 A BE201805 A BE 201805A BE 884848 A BE884848 A BE 884848A
- Authority
- BE
- Belgium
- Prior art keywords
- eplepsy
- treatment
- valproic acid
- mixed salt
- stability characteristics
- Prior art date
Links
- NIJJYAXOARWZEE-UHFFFAOYSA-N di-n-propyl-acetic acid Natural products CCCC(C(O)=O)CCC NIJJYAXOARWZEE-UHFFFAOYSA-N 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- MSRILKIQRXUYCT-UHFFFAOYSA-M valproate semisodium Chemical compound [Na+].CCCC(C(O)=O)CCC.CCCC(C([O-])=O)CCC MSRILKIQRXUYCT-UHFFFAOYSA-M 0.000 title 1
- 229960000604 valproic acid Drugs 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
- C07C53/126—Acids containing more than four carbon atoms
- C07C53/128—Acids containing more than four carbon atoms the carboxylic group being bound to a carbon atom bound to at least two other carbon atoms, e.g. neo-acids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pain & Pain Management (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6828479A | 1979-08-20 | 1979-08-20 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BE884848A true BE884848A (fr) | 1981-02-20 |
Family
ID=22081599
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BE0/201805A BE884848A (fr) | 1979-08-20 | 1980-08-20 | Sel mixte d'acide valproique utile notamment pour le traitement de l'epilepsie, presentant des caracteristiques tres superieures de stabilite |
Country Status (8)
| Country | Link |
|---|---|
| EP (1) | EP0034172B1 (fr) |
| AU (1) | AU538751B2 (fr) |
| BE (1) | BE884848A (fr) |
| CA (1) | CA1136151A (fr) |
| DE (1) | DE3063328D1 (fr) |
| IT (1) | IT1148718B (fr) |
| WO (1) | WO1981000562A1 (fr) |
| ZA (1) | ZA804636B (fr) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR2547499A1 (fr) * | 1983-06-15 | 1984-12-21 | Opochimiotherapie Lab | Medicaments contenant du dipropylacetate de calcium |
| IL72381A (en) * | 1983-07-20 | 1988-03-31 | Sanofi Sa | Pharmaceutical composition based on valproic acid |
| FR2549374B1 (fr) * | 1983-07-20 | 1985-10-18 | Sanofi Sa | Compositions medicamenteuses a base d'acide valproique modifiant favorablement leur cinetique et leur procede de fabrication galenique |
| US4558070A (en) * | 1983-10-26 | 1985-12-10 | Abbott Laboratories | Acid salts of valproic acid |
| CA1242738A (fr) * | 1983-10-26 | 1988-10-04 | Abbott Laboratories | Sels acides de l'acide valproique |
| DE3709230A1 (de) * | 1987-03-20 | 1988-10-06 | Desitin Arzneimittel Gmbh | Neues calciumsalz der valproinsaeure |
| FR2643556B1 (fr) * | 1989-02-27 | 1993-03-05 | Sanofi Sa | Composition pharmaceutique a liberation prolongee d'acide valproique |
| DE19840152A1 (de) * | 1998-09-03 | 2000-03-09 | Dresden Arzneimittel | Calciumvalproat enthaltende pharmazeutische Zusammensetzungen mit retardierter Wirkstoff-Freisetzung, Verfahren zu deren Herstellung und deren Verwendung |
| US6753349B1 (en) * | 1999-11-02 | 2004-06-22 | Cilag Ag | Method of preparing valproinic acid compounds |
| AR057882A1 (es) | 2005-11-09 | 2007-12-26 | Novartis Ag | Compuestos de accion doble de bloqueadores del receptor de angiotensina e inhibidores de endopeptidasa neutra |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1295343A (fr) * | 1959-08-03 | 1962-06-08 | Chugai Pharmaceutical Co Ltd | Procédé de fabrication de dérivés de glucosamine |
| FR2442M (fr) * | 1962-10-17 | 1964-04-06 | Henry Eugene | L'acide dipropylacétique et ses dérivés en tant que nouveuax médicaments dépresseurs du systeme nerveux central. |
| FR2383907A1 (fr) * | 1977-03-15 | 1978-10-13 | Labaz | Procede de preparation de derives de l'acide acetique et derives obtenus par ce procede |
-
1980
- 1980-07-28 DE DE8080901740T patent/DE3063328D1/de not_active Expired
- 1980-07-28 AU AU63329/80A patent/AU538751B2/en not_active Expired
- 1980-07-28 CA CA000357148A patent/CA1136151A/fr not_active Expired
- 1980-07-28 WO PCT/US1980/000954 patent/WO1981000562A1/fr not_active Ceased
- 1980-07-30 ZA ZA00804636A patent/ZA804636B/xx unknown
- 1980-08-18 IT IT24207/80A patent/IT1148718B/it active
- 1980-08-20 BE BE0/201805A patent/BE884848A/fr not_active IP Right Cessation
-
1981
- 1981-03-09 EP EP80901740A patent/EP0034172B1/fr not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ZA804636B (en) | 1981-11-25 |
| EP0034172B1 (fr) | 1983-05-18 |
| CA1136151A (fr) | 1982-11-23 |
| IT8024207A0 (it) | 1980-08-18 |
| WO1981000562A1 (fr) | 1981-03-05 |
| EP0034172A4 (fr) | 1981-12-10 |
| IT1148718B (it) | 1986-12-03 |
| DE3063328D1 (en) | 1983-07-07 |
| EP0034172A1 (fr) | 1981-08-26 |
| AU6332980A (en) | 1981-03-18 |
| AU538751B2 (en) | 1984-08-23 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RE | Patent lapsed |
Owner name: ABBOTT LABORATORIES Effective date: 19890831 |