AU8595898A - Novel diarylsulfone non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus - Google Patents

Novel diarylsulfone non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus

Info

Publication number: AU8595898A
Authority: AU; Australia
Prior art keywords: diarylsulfone; novel; reverse transcriptase; immunodeficiency virus; human immunodeficiency
Prior art date: 1997-07-29
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Abandoned

Application number

AU85958/98A

Inventor

Murray Zanger

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Philadelphia College of Pharmacy and Science

Original Assignee

Philadelphia College of Pharmacy and Science

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-07-29

Filing date

1998-07-29

Publication date

1999-02-22

1998-07-29 Application filed by Philadelphia College of Pharmacy and Science filed Critical Philadelphia College of Pharmacy and Science

1999-02-22 Publication of AU8595898A publication Critical patent/AU8595898A/en

Status Abandoned legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/58—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems with hetero atoms directly attached to the ring nitrogen atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/15—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings
- C07C311/21—Sulfonamides having sulfur atoms of sulfonamide groups bound to carbon atoms of six-membered aromatic rings having the nitrogen atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C311/00—Amides of sulfonic acids, i.e. compounds having singly-bound oxygen atoms of sulfo groups replaced by nitrogen atoms, not being part of nitro or nitroso groups
- C07C311/22—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms
- C07C311/29—Sulfonamides, the carbon skeleton of the acid part being further substituted by singly-bound oxygen atoms having the sulfur atom of at least one of the sulfonamide groups bound to a carbon atom of a six-membered aromatic ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/36—Sulfur atoms

Landscapes

Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Virology (AREA)
Chemical Kinetics & Catalysis (AREA)
Medicinal Chemistry (AREA)
Tropical Medicine & Parasitology (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
AIDS & HIV (AREA)
General Chemical & Material Sciences (AREA)
Molecular Biology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

AU85958/98A 1997-07-29 1998-07-29 Novel diarylsulfone non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus Abandoned AU8595898A (en)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
US08/901,919 US6063790A (en)	1997-07-29	1997-07-29	Diarylsulfone non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus
US08901919		1997-07-29
PCT/US1998/015577 WO1999006037A1 (en)	1997-07-29	1998-07-29	Novel diarylsulfone non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus

Publications (1)

Publication Number	Publication Date
AU8595898A true AU8595898A (en)	1999-02-22

Family

ID=25415059

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AU85958/98A Abandoned AU8595898A (en)	1997-07-29	1998-07-29	Novel diarylsulfone non-nucleoside reverse transcriptase inhibitors of human immunodeficiency virus

Country Status (5)

Country	Link
US (2)	US6063790A (en)
EP (1)	EP1011652A4 (en)
AU (1)	AU8595898A (en)
CA (1)	CA2303429A1 (en)
WO (1)	WO1999006037A1 (en)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US6586617B1 (en)	1999-04-28	2003-07-01	Sumitomo Chemical Takeda Agro Company, Limited	Sulfonamide derivatives
JP2001026506A (en) *	1999-04-28	2001-01-30	Takeda Chem Ind Ltd	Sulfonamide derivative
EP2925717A4 (en) *	2012-11-28	2016-08-03	Stichting Dienst Landbouwkundi	BENZENESULFONAMIDE COMPOUNDS FOR SOMATIC EMBRYOGENESIS IN PLANTS

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5142056A (en) *	1989-05-23	1992-08-25	Abbott Laboratories	Retroviral protease inhibiting compounds
US4505929A (en) *	1980-06-12	1985-03-19	The Dow Chemical Company	Sulfur-substituted diphenyl ethers having antiviral activity
JPS57167465A (en) *	1981-04-10	1982-10-15	Sumitomo Chemical Co	Dyeing of hydrophobic fiber
JPS613780A (en) *	1984-06-19	1986-01-09	Ricoh Co Ltd	heat sensitive recording material
US5017610A (en) *	1988-06-13	1991-05-21	Ono Pharmaceutical Co., Ltd.	Derivatives of p-substituted phenyl ester of pivalic acid
US5278173A (en) *	1988-06-30	1994-01-11	Davis Michael H	Method of inhibiting the activity of human immunodeficiency virus (HIV) in vivo
US5308854A (en) *	1990-06-18	1994-05-03	Merck & Co., Inc.	Inhibitors of HIV reverse transcriptase
US5230731A (en) *	1990-09-10	1993-07-27	Seiko Epson Corporation	Hot-melt ink composition
WO1992006683A1 (en) *	1990-10-22	1992-04-30	Research Corporation Technologies, Inc.	Aryl and heteroaryl compounds having anti-retrovirus activity
CA2147495A1 (en) *	1992-10-21	1994-04-28	Toshio Miyoshi	N-t-butylaniline analog and lipid level depressant containing the same
JPH06199047A (en) *	1993-01-08	1994-07-19	New Oji Paper Co Ltd	Heat-sensitive recording substance
US5565200A (en) *	1995-04-14	1996-10-15	University Of Southern California	Pharmaceutical preparations derived from korean mistletoe

1997
- 1997-07-29 US US08/901,919 patent/US6063790A/en not_active Expired - Fee Related
1998
- 1998-07-29 AU AU85958/98A patent/AU8595898A/en not_active Abandoned
- 1998-07-29 CA CA002303429A patent/CA2303429A1/en not_active Abandoned
- 1998-07-29 EP EP98937186A patent/EP1011652A4/en not_active Withdrawn
- 1998-07-29 WO PCT/US1998/015577 patent/WO1999006037A1/en not_active Ceased
2000
- 2000-04-11 US US09/547,820 patent/US6303630B1/en not_active Expired - Fee Related

Also Published As

Publication number	Publication date
CA2303429A1 (en)	1999-02-11
US6063790A (en)	2000-05-16
US6303630B1 (en)	2001-10-16
WO1999006037A1 (en)	1999-02-11
EP1011652A4 (en)	2004-12-22
EP1011652A1 (en)	2000-06-28

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Legal Events

Date	Code	Title	Description
2000-04-13	MK6	Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase