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AU7414300A - Method for the production of substituted pyrimidine derivatives - Google Patents

Method for the production of substituted pyrimidine derivatives

Info

Publication number
AU7414300A
AU7414300A AU74143/00A AU7414300A AU7414300A AU 7414300 A AU7414300 A AU 7414300A AU 74143/00 A AU74143/00 A AU 74143/00A AU 7414300 A AU7414300 A AU 7414300A AU 7414300 A AU7414300 A AU 7414300A
Authority
AU
Australia
Prior art keywords
production
pyrimidine derivatives
substituted pyrimidine
substituted
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU74143/00A
Inventor
Cristina Alonso-Alija
Jan Janichen
Michael Preiss
Alexander Straub
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of AU7414300A publication Critical patent/AU7414300A/en
Abandoned legal-status Critical Current

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C255/00Carboxylic acid nitriles
    • C07C255/01Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms
    • C07C255/31Carboxylic acid nitriles having cyano groups bound to acyclic carbon atoms having cyano groups bound to acyclic carbon atoms of a carbon skeleton containing rings other than six-membered aromatic rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2601/00Systems containing only non-condensed rings
    • C07C2601/02Systems containing only non-condensed rings with a three-membered ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
AU74143/00A 1999-09-08 2000-08-28 Method for the production of substituted pyrimidine derivatives Abandoned AU7414300A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE19942809A DE19942809A1 (en) 1999-09-08 1999-09-08 Process for the preparation of substituted pyrimidine derivatives
DE19942809 1999-09-08
PCT/EP2000/008362 WO2001017998A2 (en) 1999-09-08 2000-08-28 Method for the production of substituted pyrimidine derivatives

Publications (1)

Publication Number Publication Date
AU7414300A true AU7414300A (en) 2001-04-10

Family

ID=7921171

Family Applications (1)

Application Number Title Priority Date Filing Date
AU74143/00A Abandoned AU7414300A (en) 1999-09-08 2000-08-28 Method for the production of substituted pyrimidine derivatives

Country Status (3)

Country Link
AU (1) AU7414300A (en)
DE (1) DE19942809A1 (en)
WO (1) WO2001017998A2 (en)

Families Citing this family (37)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE10122894A1 (en) * 2001-05-11 2002-11-14 Bayer Ag New pyrazolo(3,4-b)pyridin-3-yl)-5-pyrimidinyl sulfonates, are soluble guanyl cyclase stimulants useful e.g. for treating cardiovascular, thromboembolic or central nervous system diseases
DE102007028319A1 (en) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituted oxazolidinones and their use
DE102007028406A1 (en) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituted oxazolidinones and their use
DE102007028407A1 (en) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituted oxazolidinones and their use
DE102007028320A1 (en) 2007-06-20 2008-12-24 Bayer Healthcare Ag Substituted oxazolidinones and their use
EP2138178A1 (en) 2008-06-28 2009-12-30 Bayer Schering Pharma Aktiengesellschaft Oxazolidninones for the treatment fo chronic obstructive pulmonary disease (COPD) and/or asthma
US20130178475A1 (en) 2010-03-17 2013-07-11 Ironwood Pharmaceuticals, Inc. sGC STIMULATORS
DK2588465T3 (en) 2010-06-30 2017-05-01 Ironwood Pharmaceuticals Inc SGC stimulators
RU2582679C2 (en) 2010-11-09 2016-04-27 Айронвуд Фармасьютикалз, Инк. sGC STIMULATORS
EP2797915B1 (en) 2011-12-27 2016-07-13 Ironwood Pharmaceuticals, Inc. 2-benzyl-3-(oxazole/thiazole)-5-(pyrimidin-2-yl)-1(H)-pyrazole derivatives as stimulators of the soluble guanylate cyclase (sGC) for the treatment of e.g. hypertension or heart failure
WO2013167669A1 (en) 2012-05-10 2013-11-14 Bayer Pharma Aktiengesellschaft Antibodies capable of binding to the coagulation factor xi and/or its activated form factor xia and uses thereof
US9309235B2 (en) 2012-09-18 2016-04-12 Ironwood Pharmaceuticals, Inc. SGC stimulators
CA2885645A1 (en) 2012-09-19 2014-03-27 Ironwood Pharmaceuticals, Inc. Sgc stimulators
LT3660013T (en) 2013-03-15 2022-04-11 Cyclerion Therapeutics, Inc. Sgc stimulators
MX2016007522A (en) 2013-12-11 2017-12-15 Ironwood Pharmaceuticals Inc Sgc stimulators.
EP3094327A1 (en) 2014-01-13 2016-11-23 Ironwood Pharmaceuticals, Inc. USE OF sGC STIMULATORS FOR THE TREATMENT OF NEUROMUSCULAR DISORDERS
US10844064B2 (en) 2014-09-17 2020-11-24 Cyclerion Therapeutics, Inc. sGC stimulators
US20170291889A1 (en) 2014-09-17 2017-10-12 Ironwood Pharmaceuticals, Inc. Pyrazole derivatives as sgc stimulators
WO2016044445A2 (en) 2014-09-17 2016-03-24 Ironwood Pharmaceuticals, Inc. sGC STIMULATORS
CA3006764A1 (en) 2015-12-14 2017-06-22 Ironwood Pharmaceuticals, Inc. Use of sgc stimulators for the treatment of gastrointestinal sphincter dysfunction
US10889577B2 (en) 2016-07-07 2021-01-12 Cyclerion Therapeutics, Inc. Solid forms of an sGC stimulator
KR102513343B1 (en) 2016-07-07 2023-03-22 사이클리온 테라퓨틱스, 인크. Phosphorus prodrugs of sGC stimulators
WO2018045276A1 (en) 2016-09-02 2018-03-08 Ironwood Pharmaceuticals, Inc. Fused bicyclic sgc stimulators
MA46752A (en) 2016-11-08 2019-09-18 Cyclerion Therapeutics Inc TREATMENT OF CNS DISEASES USING GCS STIMULATORS
IL266372B2 (en) 2016-11-08 2023-11-01 Cyclerion Therapeutics Inc Sgc stimulators
US20190381039A1 (en) 2016-12-13 2019-12-19 Cyclerion Therapeutics, Inc. USE OF sGC STIMULATORS FOR THE TREATMENT OF ESOPHAGEAL MOTILITY DISORDERS
EP3727388A1 (en) 2017-12-19 2020-10-28 Cyclerion Therapeutics, Inc. Sgc stimulators
MX2023004858A (en) 2018-03-07 2023-11-24 Cyclerion Therapeutics Inc Crystalline forms of an sgc stimulator.
KR20250141845A (en) 2018-07-11 2025-09-29 티센토 쎄라퓨틱스 인크. USE OF sGC STIMULATORS FOR THE TREATMENT OF MITOCHONRIAL DISORDERS
MX2021005892A (en) 2018-11-28 2021-06-23 Topadur Pharma Ag NOVEL ACTIVATORS OF SOLUBLE GUANYLATE CYCLASE AND INHIBITORS OF PHOSPHODIESTERASE WITH DUAL MODE OF ACTION AND THEIR USES.
WO2021195403A1 (en) 2020-03-26 2021-09-30 Cyclerion Therapeutics, Inc. Deuterated sgc stimulators
WO2021202546A1 (en) 2020-03-31 2021-10-07 Cyclerion Therapeutics, Inc. Early drug interventions to reduce covid-19 related respiratory distress, need for ventilator assistance and death
US20240207265A1 (en) 2021-04-20 2024-06-27 Tisento Therapeutics Inc. TREATMENT OF CNS DISEASES WITH sGC STIMULATORS
BR112023021851A2 (en) 2021-04-20 2024-02-06 Tisento Therapeutics Inc SGC STIMULANTS
JP2025536343A (en) 2022-10-18 2025-11-05 ティセント セラピューティクス インコーポレーテッド Pyrimidine SGC stimulators
WO2024086182A1 (en) 2022-10-18 2024-04-25 Tisento Therapeutics Inc. Treatment of mitochondrial diseases with sgc stimulators
CN118772140A (en) * 2023-04-07 2024-10-15 四川大学 A class of compounds and their use in treating hDHODH-mediated diseases

Also Published As

Publication number Publication date
WO2001017998A2 (en) 2001-03-15
WO2001017998A3 (en) 2001-10-11
DE19942809A1 (en) 2001-03-15

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Legal Events

Date Code Title Description
MK6 Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase