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AU584861B2 - N-(2-Nitrophenyl)-4-aminopyrimidine derivatives, the preparation thereof and use thereof - Google Patents

N-(2-Nitrophenyl)-4-aminopyrimidine derivatives, the preparation thereof and use thereof

Info

Publication number
AU584861B2
AU584861B2 AU32450/84A AU3245084A AU584861B2 AU 584861 B2 AU584861 B2 AU 584861B2 AU 32450/84 A AU32450/84 A AU 32450/84A AU 3245084 A AU3245084 A AU 3245084A AU 584861 B2 AU584861 B2 AU 584861B2
Authority
AU
Australia
Prior art keywords
nitrophenyl
preparation
aminopyrimidine derivatives
aminopyrimidine
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU32450/84A
Other versions
AU3245084A (en
Inventor
Wolfgang Eckhardt
Adolf Hubele
Elmar Sturm
Helmut Zondler
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of AU3245084A publication Critical patent/AU3245084A/en
Application granted granted Critical
Publication of AU584861B2 publication Critical patent/AU584861B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/32—One oxygen, sulfur or nitrogen atom
    • C07D239/42—One nitrogen atom
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/48—Two nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/52—Two oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/56—One oxygen atom and one sulfur atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
AU32450/84A 1983-08-29 1984-08-28 N-(2-Nitrophenyl)-4-aminopyrimidine derivatives, the preparation thereof and use thereof Ceased AU584861B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
CH4723/83 1983-08-29
CH472383 1983-08-29

Publications (2)

Publication Number Publication Date
AU3245084A AU3245084A (en) 1985-03-07
AU584861B2 true AU584861B2 (en) 1989-06-08

Family

ID=4281386

Family Applications (1)

Application Number Title Priority Date Filing Date
AU32450/84A Ceased AU584861B2 (en) 1983-08-29 1984-08-28 N-(2-Nitrophenyl)-4-aminopyrimidine derivatives, the preparation thereof and use thereof

Country Status (12)

Country Link
EP (1) EP0139613A1 (en)
JP (1) JPS6072867A (en)
AU (1) AU584861B2 (en)
BR (1) BR8404295A (en)
CA (1) CA1254560A (en)
DK (1) DK410384A (en)
ES (1) ES8506288A1 (en)
GR (1) GR80171B (en)
IL (1) IL72771A (en)
NZ (1) NZ209356A (en)
PT (1) PT79137B (en)
ZA (1) ZA846706B (en)

Families Citing this family (34)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH21918A (en) * 1983-07-25 1988-04-08 Ciba Geigy Ag N-(2-nitrophenyl)-5-aminopyrimidine derivatives,the preparation and use thereof
US4659363A (en) * 1983-07-25 1987-04-21 Ciba-Geigy Corporation N-(2-nitrophenyl)-2-aminopyrimidine derivatives, the preparation and use thereof
US4694009A (en) * 1984-06-25 1987-09-15 Ciba-Geigy Corporation Pesticidal compositions
DE3618353A1 (en) * 1986-05-31 1987-12-03 Hoechst Ag PEST CONTROLS BASED ON AMINOPYRIMIDINE DERIVATIVES AND NEW AMINOPYRIMIDINE COMPOUNDS
DE3717480A1 (en) * 1987-05-23 1988-12-01 Shell Agrar Gmbh & Co Kg Novel herbicidal and microbicidal 2,6-diaminopyrimidines
ES2057172T3 (en) * 1988-03-09 1994-10-16 Ciba Geigy Ag AGENT FOR THE PROTECTION OF PLANTS AGAINST DISEASES.
DE3808739A1 (en) * 1988-03-16 1989-09-28 Bayer Ag PYRIMIDINE DERIVATIVES
IE63502B1 (en) * 1989-04-21 1995-05-03 Zeneca Ltd Aminopyrimidine derivatives useful for treating cardiovascular disorders
US5117097A (en) * 1990-02-27 1992-05-26 Kabushiki Kaisha Tokai Rika Denki Seisakusho Key system for a vehicle
KR910021383A (en) * 1990-02-27 1991-12-20 베그르 발데크 N- (2, 6-dinitro-3-chloro-4-trifluoromethylphenyl) -4-amino-6-fluoropyrimidine derivative and preparation method thereof
GB9008818D0 (en) * 1990-04-19 1990-06-13 Ici Plc Amine derivatives
DE4029648A1 (en) * 1990-09-19 1992-03-26 Hoechst Ag 4-ANILINO-PYRIMIDINE, METHOD FOR THE PRODUCTION THEREOF, AGENTS CONTAINING IT AND THEIR USE AS FUNGICIDES
WO1992008461A1 (en) * 1990-11-14 1992-05-29 Protos Corporation Specific inhibition of dihydrofolate reductase and compounds therefor
GB9325217D0 (en) * 1993-12-09 1994-02-09 Zeneca Ltd Pyrimidine derivatives
DE19917785A1 (en) * 1999-04-20 2000-10-26 Bayer Ag New 2,4-diamino-pyrimidine derivatives useful as microbicides in protection of plants and materials and as herbicides
TWI329105B (en) 2002-02-01 2010-08-21 Rigel Pharmaceuticals Inc 2,4-pyrimidinediamine compounds and their uses
JP2006514989A (en) 2002-07-29 2006-05-18 ライジェル ファーマシューティカルズ Method for treating and preventing autoimmune diseases with 2,4-pyrimidinediamine compounds
AU2004265288A1 (en) 2003-07-30 2005-02-24 Rigel Pharmaceuticals, Inc. 2,4-pyrimidinediamine compounds for use in the treatment or prevention of autoimmune diseases
EP1814878B1 (en) 2004-11-24 2012-01-04 Rigel Pharmaceuticals, Inc. Spiro-2, 4-pyrimidinediamine compounds and their uses
US7449458B2 (en) 2005-01-19 2008-11-11 Rigel Pharmaceuticals, Inc. Prodrugs of 2,4-pyrimidinediamine compounds and their uses
PT2562162E (en) * 2008-01-22 2015-10-21 Dow Agrosciences Llc N-cyano-4-amino-5-fluoro-pyrimidine derivatives as fungicides
JP5580310B2 (en) * 2008-08-01 2014-08-27 ダウ アグロサイエンシィズ エルエルシー Use of 5-fluorocytosine as a fungicide
CA2769073C (en) 2009-08-07 2018-07-24 Dow Agrosciences Llc N1-sulfonyl-5-fluoropyrimidinone derivatives
UA106889C2 (en) 2009-08-07 2014-10-27 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі N1-ACYL-5-FLORPYRIMIDINONE DERIVATIVES
UA107671C2 (en) 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
UA112284C2 (en) 2009-08-07 2016-08-25 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі 5-fluoro-pyrimidinone derivatives
EP2521452B1 (en) 2010-01-07 2014-12-24 Dow AgroSciences LLC THIAZOLO[5,4-d]PYRIMIDINES AND THEIR USE AS AGROCHEMICALS
CN103874413B (en) 2011-08-17 2017-03-08 阿达玛马克西姆股份有限公司 5‑Fluoro‑4‑imino‑3‑(substituted)‑3,4‑dihydropyrimidin‑2(1H)one derivatives
KR20150100869A (en) 2012-12-28 2015-09-02 다우 아그로사이언시즈 엘엘씨 N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxamides derivatives
CN110003118A (en) 2012-12-28 2019-07-12 阿达玛马克西姆股份有限公司 The method for preparing carboxylic ester derivative
CA2893776A1 (en) 2012-12-28 2014-07-03 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1h)-one derivatives
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
HUE072634T2 (en) 2013-12-31 2025-11-28 Adama Makhteshim Ltd Synergistic fungicidal mixtures for fungal control in cereals
SG11201605372QA (en) 2013-12-31 2016-08-30 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation

Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2687384A (en) * 1983-04-22 1984-10-25 Shell Internationale Research Maatschappij B.V. Biologically active (N-Heterocyclic) anilines
AU3099884A (en) * 1983-07-25 1985-02-14 Ciba-Geigy Ag N-(2-nitrophenyl)-5-aminopyrimidine derivatives
AU4398885A (en) * 1984-06-25 1986-01-02 Ciba-Geigy Ag Pesticidal compositions

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PH20344A (en) * 1981-01-29 1986-12-04 Sankyo Co Aminopyrimidine derivatives, processes for their preparation, and fungicidal, insecticidal and acaricidal compositions containing them
JPS57203072A (en) * 1981-06-05 1982-12-13 Sankyo Co Ltd 4-anilinopyrimidine derivative, its preparation, antidepressant comprising it as active ingredient

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2687384A (en) * 1983-04-22 1984-10-25 Shell Internationale Research Maatschappij B.V. Biologically active (N-Heterocyclic) anilines
AU3099884A (en) * 1983-07-25 1985-02-14 Ciba-Geigy Ag N-(2-nitrophenyl)-5-aminopyrimidine derivatives
AU4398885A (en) * 1984-06-25 1986-01-02 Ciba-Geigy Ag Pesticidal compositions

Also Published As

Publication number Publication date
PT79137A (en) 1984-09-01
IL72771A0 (en) 1984-11-30
CA1254560A (en) 1989-05-23
AU3245084A (en) 1985-03-07
PT79137B (en) 1986-11-14
JPS6072867A (en) 1985-04-24
BR8404295A (en) 1985-07-23
DK410384A (en) 1985-03-01
GR80171B (en) 1985-01-02
DK410384D0 (en) 1984-08-28
ZA846706B (en) 1985-04-24
NZ209356A (en) 1988-01-08
ES535469A0 (en) 1985-07-16
ES8506288A1 (en) 1985-07-16
IL72771A (en) 1988-03-31
EP0139613A1 (en) 1985-05-02

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