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AU569494B2 - 1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids - Google Patents

1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids

Info

Publication number
AU569494B2
AU569494B2 AU25516/84A AU2551684A AU569494B2 AU 569494 B2 AU569494 B2 AU 569494B2 AU 25516/84 A AU25516/84 A AU 25516/84A AU 2551684 A AU2551684 A AU 2551684A AU 569494 B2 AU569494 B2 AU 569494B2
Authority
AU
Australia
Prior art keywords
optionally substituted
carbon atoms
cyclopropyl
dihydro
oxo
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
AU25516/84A
Other versions
AU2551684A (en
Inventor
Klaus Grohe
Karl-Heinz Kuck
Engelbert Kuhle
Uwe Petersen
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Bayer AG
Original Assignee
Bayer AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer AG filed Critical Bayer AG
Publication of AU2551684A publication Critical patent/AU2551684A/en
Application granted granted Critical
Publication of AU569494B2 publication Critical patent/AU569494B2/en
Anticipated expiration legal-status Critical
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Quinoline Compounds (AREA)

Abstract

1. Use of 1-cyclopropyl-1,4-dihydro-4-oxo-3-quinolinecarboxylic acid derivatives of the formula (l) see diagramm : EP0121727,P34,F1 in which R**1 represents a CO-R**6, CN, SO2 -R**7 or S-R**8 radical, wherein R**6 represents hydrogen, optionally substituted straight-chain or branched alkyl with 1 to 6 carbon atoms, optionally substituted aryl with 6 or 10 carbon atoms, optionally substituted aralkyl with 6 carbon atoms in the aryl part and 1 to 3 carbon atoms in the alkyl part, optionally substituted alkoxy or alkylthio with 1 to 6 carbon atoms, optionally substituted phenoxy, optionally substituted benzyloxy, amino, optionally substituted alkylamino or dialkylamino with 1 to 6 carbon atoms per alkyl radical or optionally substituted phenylamino, R**7 represents optionally substituted straightchain or branched alkyl with 1 to 5 carbon atoms, phenyl or methylphenyl, R**8 represents methoxycarbonyl, trichloromethyl, trifluoromethyl or dichlorofluoromethyl, R**2, R**3, R**4 and R**5 can be identical or different and represent hydrogen, methyl, ethyl or n- or i-propyl and X represents hydrogen, halogen or nitro, and their acid addition, alkali metal and alkaline earth metal salts, zinc, manganese and copper salts and hydrates, for combating bacteria in plant protection.
AU25516/84A 1983-03-12 1984-03-12 1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids Ceased AU569494B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3308909 1983-03-12
DE19833308909 DE3308909A1 (en) 1983-03-12 1983-03-12 BACTERICIDALS BASED ON CHINOLONIC CARBONIC ACID

Publications (2)

Publication Number Publication Date
AU2551684A AU2551684A (en) 1984-09-13
AU569494B2 true AU569494B2 (en) 1988-02-04

Family

ID=6193319

Family Applications (1)

Application Number Title Priority Date Filing Date
AU25516/84A Ceased AU569494B2 (en) 1983-03-12 1984-03-12 1-cyclopropyl-1,4-dihydro-4-oxo-3-quinoline carboxylic acids

Country Status (12)

Country Link
EP (1) EP0121727B1 (en)
JP (1) JPS59170069A (en)
AT (1) ATE22387T1 (en)
AU (1) AU569494B2 (en)
BR (1) BR8401084A (en)
CA (1) CA1222249A (en)
DE (2) DE3308909A1 (en)
DK (1) DK148384A (en)
GR (1) GR81891B (en)
HU (1) HU194024B (en)
IL (1) IL71200A (en)
ZA (1) ZA841764B (en)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NZ217650A (en) * 1985-09-24 1989-09-27 Hoffmann La Roche Quinoline derivatives and pharmaceutical compositions
DE3542002A1 (en) * 1985-11-28 1987-06-04 Bayer Ag 1-CYCLOPROPYL-6-FLUOR-1,4-DIHYDRO-4-OXO-7- (1-PIPERAZINYL) -3-QUINOLINE CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THEIR ANTIBACTERIAL AGENTS CONTAINING THEM
US4788320A (en) * 1986-01-20 1988-11-29 Kyorin Pharmaceutical Co., Ltd. Benzoylacetic acid ester derivatives and process for their preparations
DE3705621C2 (en) * 1986-02-25 1997-01-09 Otsuka Pharma Co Ltd Heterocyclic substituted quinolonecarboxylic acid derivatives
SI8712447A8 (en) 1987-12-31 1995-12-31 Krka Tovarna Zdravil Process for preparing 1-substituted 6-fluoro-4-oxo-7-(1-piperazinyl) -1,4-dihydroquinoline-3-carboxylic acid and new intermediate used in this process
US5328908A (en) * 1988-10-24 1994-07-12 Procter & Gamble Pharmaceuticals, Inc. Antimicrobial quinolone thioureas
SI9200377A (en) 1992-12-11 1994-06-30 Krka Process for the preparation of 1-substituted 6-fluoro-4-oxo-7-(1-piperazinyl)-1,4-dihydroquinoline-3-carboxilic acid, novel intermediate used in this process and process for its preparation
CA2114981A1 (en) * 1993-02-09 1994-08-10 Kazumi Ogata Quinolonecarboxylic acid derivatives
SE9904108D0 (en) * 1999-11-15 1999-11-15 New Pharma Research Ab New compounds

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2428484A (en) * 1983-02-25 1984-08-30 Bayer Aktiengesellschaft Quinolone carboxylic acids

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS604820B2 (en) * 1979-02-26 1985-02-06 大塚製薬株式会社 Quinoline carboxylic acid derivative
DE3033157A1 (en) * 1980-09-03 1982-04-01 Bayer Ag, 5090 Leverkusen 7-AMINO-1-CYCLOPROPYL-4-OXO-1,4-DIHYDRO-NAPHTHYRIDINE-3-CARBONIC ACIDS, METHOD FOR THE PRODUCTION THEREOF AND THE ANTIBACTERIAL AGENTS CONTAINING THEM

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2428484A (en) * 1983-02-25 1984-08-30 Bayer Aktiengesellschaft Quinolone carboxylic acids

Also Published As

Publication number Publication date
HU194024B (en) 1988-01-28
EP0121727B1 (en) 1986-09-24
AU2551684A (en) 1984-09-13
IL71200A0 (en) 1984-06-29
DK148384D0 (en) 1984-02-29
BR8401084A (en) 1984-10-16
EP0121727A1 (en) 1984-10-17
GR81891B (en) 1984-12-12
DE3308909A1 (en) 1984-09-13
HUT34665A (en) 1985-04-28
IL71200A (en) 1988-03-31
ATE22387T1 (en) 1986-10-15
JPS59170069A (en) 1984-09-26
DK148384A (en) 1984-09-13
CA1222249A (en) 1987-05-26
ZA841764B (en) 1984-10-31
DE3460791D1 (en) 1986-10-30

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